Catalytic promiscuity in the biosynthesis of cyclic peptide secondary metabolites in planktonic marine cyanobacteria
Li, Bo, Sher, Daniel, Kelly, Libusha, Shi, Yanxiang, Huang, Katherine, Knerr, Patrick J, Joewono, Ike, Rusch, Doug, Chisholm, Sallie W, van der Donk, Wilfred A
Published in Proceedings of the National Academy of Sciences - PNAS (08.06.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (08.06.2010)
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Journal Article
Next generation GLP-1/GIP/glucagon triple agonists normalize body weight in obese mice
Knerr, Patrick J., Mowery, Stephanie A., Douros, Jonathan D., Premdjee, Bhavesh, Hjøllund, Karina Rahr, He, Yantao, Kruse Hansen, Ann Maria, Olsen, Anette K., Perez-Tilve, Diego, DiMarchi, Richard D., Finan, Brian
Published in Molecular metabolism (Germany) (01.09.2022)
Published in Molecular metabolism (Germany) (01.09.2022)
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Journal Article
Spatiotemporal GLP-1 and GIP receptor signaling and trafficking/recycling dynamics induced by selected receptor mono- and dual-agonists
Novikoff, Aaron, O'Brien, Shannon L., Bernecker, Miriam, Grandl, Gerald, Kleinert, Maximilian, Knerr, Patrick J., Stemmer, Kerstin, Klingenspor, Martin, Zeigerer, Anja, DiMarchi, Richard, Tschöp, Matthias H., Finan, Brian, Calebiro, Davide, Müller, Timo D.
Published in Molecular metabolism (Germany) (01.07.2021)
Published in Molecular metabolism (Germany) (01.07.2021)
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Journal Article
Discovery of a potent GIPR peptide antagonist that is effective in rodent and human systems
Yang, Bin, Gelfanov, Vasily M, El, Kimberley, Chen, Alex, Rohlfs, Rebecca, DuBois, Barent, Kruse Hansen, Ann Maria, Perez-Tilve, Diego, Knerr, Patrick J, D'Alessio, David, Campbell, Jonathan E, Douros, Jonathan D, Finan, Brian
Published in Molecular metabolism (Germany) (01.12.2022)
Published in Molecular metabolism (Germany) (01.12.2022)
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Journal Article
Experimental colonization with H. hepaticus, S. aureus and R. pneumotropicus does not influence the metabolic response to high-fat diet or incretin-analogues in wildtype SOPF mice
Wunderlich, Margit, Miller, Manuel, Ritter, Bärbel, Le Gleut, Ronan, Marchi, Hannah, Majzoub-Altweck, Monir, Knerr, Patrick J., Douros, Jonathan D., Müller, Timo D., Brielmeier, Markus
Published in Molecular metabolism (Germany) (01.09.2024)
Published in Molecular metabolism (Germany) (01.09.2024)
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Journal Article
The glucose-dependent insulinotropic polypeptide (GIP) regulates body weight and food intake via CNS-GIPR signaling
Zhang, Qian, Delessa, Challa Tenagne, Augustin, Robert, Bakhti, Mostafa, Colldén, Gustav, Drucker, Daniel J., Feuchtinger, Annette, Caceres, Cristina Garcia, Grandl, Gerald, Harger, Alexandra, Herzig, Stephan, Hofmann, Susanna, Holleman, Cassie Lynn, Jastroch, Martin, Keipert, Susanne, Kleinert, Maximilian, Knerr, Patrick J., Kulaj, Konxhe, Legutko, Beata, Lickert, Heiko, Liu, Xue, Luippold, Gerd, Lutter, Dominik, Malogajski, Emilija, Medina, Marta Tarquis, Mowery, Stephanie A., Blutke, Andreas, Perez-Tilve, Diego, Salinno, Ciro, Sehrer, Laura, DiMarchi, Richard D., Tschöp, Matthias H., Stemmer, Kerstin, Finan, Brian, Wolfrum, Christian, Müller, Timo D.
Published in Cell metabolism (06.04.2021)
Published in Cell metabolism (06.04.2021)
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Journal Article
Chemical Synthesis and Biological Activity of Analogues of the Lantibiotic Epilancin 15X
Knerr, Patrick J, van der Donk, Wilfred A
Published in Journal of the American Chemical Society (09.05.2012)
Published in Journal of the American Chemical Society (09.05.2012)
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Journal Article
Selection and progression of unimolecular agonists at the GIP, GLP-1, and glucagon receptors as drug candidates
Knerr, Patrick J., Mowery, Stephanie A., Finan, Brian, Perez-Tilve, Diego, Tschöp, Matthias H., DiMarchi, Richard D.
Published in Peptides (New York, N.Y. : 1980) (01.03.2020)
Published in Peptides (New York, N.Y. : 1980) (01.03.2020)
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Journal Article
Glucose-dependent insulinotropic polypeptide regulates body weight and food intake via GABAergic neurons in mice
Liskiewicz, Arkadiusz, Khalil, Ahmed, Liskiewicz, Daniela, Novikoff, Aaron, Grandl, Gerald, Maity-Kumar, Gandhari, Gutgesell, Robert M, Bakhti, Mostafa, Bastidas-Ponce, Aimée, Czarnecki, Oliver, Makris, Konstantinos, Lickert, Heiko, Feuchtinger, Annette, Tost, Monica, Coupland, Callum, Ständer, Lisa, Akindehin, Seun, Prakash, Sneha, Abrar, Faiyaz, Castelino, Russell L, He, Yantao, Knerr, Patrick J, Yang, Bin, Hogendorf, Wouter F J, Zhang, Shiqi, Hofmann, Susanna M, Finan, Brian, DiMarchi, Richard D, Tschöp, Matthias H, Douros, Jonathan D, Müller, Timo D
Published in Nature metabolism (01.12.2023)
Published in Nature metabolism (01.12.2023)
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Journal Article
Conjugation to Albumin-Binding Molecule Tags as a Strategy to Improve Both Efficacy and Pharmacokinetic Properties of the Complement Inhibitor Compstatin
Huang, Yijun, Reis, Edimara S., Knerr, Patrick J., van der Donk, Wilfred A., Ricklin, Daniel, Lambris, John D.
Published in ChemMedChem (01.10.2014)
Published in ChemMedChem (01.10.2014)
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Journal Article
Non-proteinogenic Amino Acids in Lacticin 481 Analogues Result in More Potent Inhibition of Peptidoglycan Transglycosylation
Knerr, Patrick J, Oman, Trent J, Garcia De Gonzalo, Chantal V, Lupoli, Tania J, Walker, Suzanne, van der Donk, Wilfred A
Published in ACS chemical biology (16.11.2012)
Published in ACS chemical biology (16.11.2012)
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Journal Article
Cover Picture: Conjugation to Albumin-Binding Molecule Tags as a Strategy to Improve Both Efficacy and Pharmacokinetic Properties of the Complement Inhibitor Compstatin (ChemMedChem 10/2014)
Huang, Yijun, Reis, Edimara S., Knerr, Patrick J., van der Donk, Wilfred A., Ricklin, Daniel, Lambris, John D.
Published in ChemMedChem (01.10.2014)
Published in ChemMedChem (01.10.2014)
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