Novel highly selective inhibitors of ubiquitin specific protease 30 (USP30) accelerate mitophagy
Kluge, Arthur F., Lagu, Bharat R., Maiti, Pranab, Jaleel, Mahaboobi, Webb, Michael, Malhotra, Jyoti, Mallat, Ashley, Srinivas, P. Akhila, Thompson, James E.
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
Published in Bioorganic & medicinal chemistry letters (15.08.2018)
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Targeted covalent drugs of the kinase family
Singh, Juswinder, Petter, Russell C, Kluge, Arthur F
Published in Current opinion in chemical biology (01.08.2010)
Published in Current opinion in chemical biology (01.08.2010)
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Journal Article
Addressing hERG activity while maintaining favorable potency, selectivity and pharmacokinetic properties of PPARδ modulators
Lagu, Bharat, Senaiar, Ramesh S., Kluge, Arthur F., Mallesh, B., Ramakrishna, M., Bhat, Raveendra, Patane, Michael A.
Published in Bioorganic & medicinal chemistry letters (15.02.2020)
Published in Bioorganic & medicinal chemistry letters (15.02.2020)
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Journal Article
Novel highly selective peroxisome proliferator-activated receptor δ (PPARδ) modulators with pharmacokinetic properties suitable for once-daily oral dosing
Lagu, Bharat, Kluge, Arthur F., Fredenburg, Ross A., Tozzo, Effie, Senaiar, Ramesh S., Jaleel, Mahaboobi, Panigrahi, Sunil K., Tiwari, Nirbhay K., Krishnamurthy, Narasimha R., Takahashi, Taisuke, Patane, Michael A.
Published in Bioorganic & medicinal chemistry letters (01.12.2017)
Published in Bioorganic & medicinal chemistry letters (01.12.2017)
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Journal Article
Highly selective peroxisome proliferator-activated receptor δ (PPARδ) modulator demonstrates improved safety profile compared to GW501516
Lagu, Bharat, Kluge, Arthur F., Goddeeris, Matthew M., Tozzo, Effie, Fredenburg, Ross A., Chellur, Shekar, Senaiar, Ramesh S., Jaleel, Mahaboobi, Babu, D. Ravi Krishna, Tiwari, Nirbhay K., Takahashi, Taisuke, Patane, Michael A.
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
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Journal Article
Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)
Lagu, Bharat, Kluge, Arthur F, Tozzo, Effie, Fredenburg, Ross, Bell, Eric L, Goddeeris, Matthew M, Dwyer, Peter, Basinski, Andrew, Senaiar, Ramesh S, Jaleel, Mahaboobi, Tiwari, Nirbhay Kumar, Panigrahi, Sunil K, Krishnamurthy, Narasimha Rao, Takahashi, Taisuke, Patane, Michael A
Published in ACS medicinal chemistry letters (13.09.2018)
Published in ACS medicinal chemistry letters (13.09.2018)
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Journal Article
Author Correction: Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
Lasko, Loren M, Jakob, Clarissa G, Edalji, Rohinton P, Qiu, Wei, Montgomery, Debra, Digiammarino, Enrico L, Hansen, T Matt, Risi, Roberto M, Frey, Robin, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Hessler, Paul, Lam, Lloyd T, Uziel, Tamar, Faivre, Emily, Ferguson, Debra, Buchanan, Fritz G, Martin, Ruth L, Torrent, Maricel, Chiang, Gary G, Karukurichi, Kannan, Langston, J William, Weinert, Brian T, Choudhary, Chunaram, de Vries, Peter, Kluge, Arthur F, Patane, Michael A, Van Drie, John H, Wang, Ce, McElligott, David, Kesicki, Edward A, Marmorstein, Ronen, Sun, Chaohong, Cole, Philip A, Rosenberg, Saul H, Michaelides, Michael R, Lai, Albert, Bromberg, Kenneth D
Published in Nature (London) (01.06.2018)
Published in Nature (London) (01.06.2018)
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Journal Article
Correction to “Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)”
Lagu, Bharat, Kluge, Arthur F, Tozzo, Effie, Fredenburg, Ross, Bell, Eric L, Goddeeris, Matthew M, Dwyer, Peter, Basinski, Andrew, Senaiar, Ramesh S, Jaleel, Mahaboobi, Tiwari, Nirbhay Kumar, Panigrahi, Sunil K, Krishnamurthy, Narasimha Rao, Takahashi, Taisuke, Patane, Michael A
Published in ACS medicinal chemistry letters (13.06.2019)
Published in ACS medicinal chemistry letters (13.06.2019)
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Journal Article
IRAK 분해제 및 이의 용도
JI NAN, MAINOLFI NELLO, WEISS MATTHEW M, ZHENG XIAOZHANG, ZHANG YI, KLUGE ARTHUR F
Year of Publication 10.09.2021
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Year of Publication 10.09.2021
Patent
A Three-Hybrid Approach to Scanning the Proteome for Targets of Small Molecule Kinase Inhibitors
Becker, Frank, Murthi, Krishna, Smith, Chase, Come, Jon, Costa-Roldán, Nuria, Kaufmann, Christine, Hanke, Urs, Degenhart, Carsten, Baumann, Sabine, Wallner, Wolfgang, Huber, Andrea, Dedier, Severine, Dill, Simone, Kinsman, David, Hediger, Mark, Bockovich, Nicholas, Meier-Ewert, Sebastian, Kluge, Arthur F, Kley, Nikolai
Published in Chemistry & biology (01.02.2004)
Published in Chemistry & biology (01.02.2004)
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HETEROARYL COMPOUNDS AND USES THEREOF
HORMOZ MAZDIYASNI, RICHLAND WAYNE TESTER, RUSSELL C PETTER, SINGH JUSWINDER, QIAO LIXIN, NIU DEQIANG, WILLIAM FREDERICK WESTLIN, KLUGE ARTHUR F
Year of Publication 07.11.2019
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Year of Publication 07.11.2019
Patent
Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
Lasko, Loren M, Jakob, Clarissa G, Edalji, Rohinton P, Qiu, Wei, Montgomery, Debra, Digiammarino, Enrico L, Hansen, T Matt, Risi, Roberto M, Frey, Robin, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Hessler, Paul, Lam, Lloyd T, Uziel, Tamar, Faivre, Emily, Ferguson, Debra, Buchanan, Fritz G, Martin, Ruth L, Torrent, Maricel, Chiang, Gary G, Karukurichi, Kannan, Langston, J William, Weinert, Brian T, Choudhary, Chunaram, de Vries, Peter, Van Drie, John H, McElligott, David, Kesicki, Ed, Marmorstein, Ronen, Sun, Chaohong, Cole, Philip A, Rosenberg, Saul H, Michaelides, Michael R, Lai, Albert, Bromberg, Kenneth D
Published in Nature (London) (05.10.2017)
Published in Nature (London) (05.10.2017)
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Journal Article
Heteroaryl compounds and uses thereof
MAZDIYASNI HORMOZ, SINGH JUSWINDER, WESTLIN WILLIAM FREDERICK, QIAO LIXIN, NIU DEQIANG, TESTER RICHLAND WAYNE, PETTER RUSSELL C, KLUGE ARTHUR F
Year of Publication 03.05.2018
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Year of Publication 03.05.2018
Patent
A series of quinoline analogues as potent inhibitors of C. albicans prolyl tRNA synthetase
Yu, Xiang Y., Hill, Jason M., Yu, Guixue, Yang, Yifeng, Kluge, Arthur F., Keith, Dennis, Finn, John, Gallant, Paul, Silverman, Jared, Lim, Audrey
Published in Bioorganic & medicinal chemistry letters (26.02.2001)
Published in Bioorganic & medicinal chemistry letters (26.02.2001)
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Journal Article
HETEROARYL COMPOUNDS AND USES THEREOF
HORMOZ MAZDIYASNI, RICHLAND WAYNE TESTER, RUSSELL C PETTER, SINGH JUSWINDER, QIAO LIXIN, NIU DEQIANG, WILLIAM FREDERICK WESTLIN, KLUGE ARTHUR F
Year of Publication 10.08.2017
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Year of Publication 10.08.2017
Patent
HETEROARYL COMPOUNDS AND USES THEREOF
PETTER RUSSELL, WESTLIN III WILLIAM FREDERICK, MAZDIYASNI HORMOZ, SINGH JUSWINDER, NIU DEQIANG, QIAO LIXIN, TESTER RICHLAND WAYNE, KLUGE ARTHUR F
Year of Publication 26.07.2017
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Year of Publication 26.07.2017
Patent
Antifungal activity of a Candida albicans GGTase I inhibitor-Alanine conjugate. inhibition of Rho1p prenylation in C. albicans
Murthi, Krishna K, Smith, Susan E, Kluge, Arthur F, Bergnes, Gustave, Bureau, Patrick, Berlin, Vivian
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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