Gasdermin D plays a vital role in the generation of neutrophil extracellular traps
Sollberger, Gabriel, Choidas, Axel, Burn, Garth Lawrence, Habenberger, Peter, Di Lucrezia, Raffaella, Kordes, Susanne, Menninger, Sascha, Eickhoff, Jan, Nussbaumer, Peter, Klebl, Bert, Krüger, Renate, Herzig, Alf, Zychlinsky, Arturo
Published in Science immunology (24.08.2018)
Published in Science immunology (24.08.2018)
Get more information
Journal Article
Small-molecule inhibitors of human mitochondrial DNA transcription
Bonekamp, Nina A, Peter, Bradley, Hillen, Hauke S, Felser, Andrea, Bergbrede, Tim, Choidas, Axel, Horn, Moritz, Unger, Anke, Di Lucrezia, Raffaella, Atanassov, Ilian, Li, Xinping, Koch, Uwe, Menninger, Sascha, Boros, Joanna, Habenberger, Peter, Giavalisco, Patrick, Cramer, Patrick, Denzel, Martin S, Nussbaumer, Peter, Klebl, Bert, Falkenberg, Maria, Gustafsson, Claes M, Larsson, Nils-Göran
Published in Nature (London) (24.12.2020)
Published in Nature (London) (24.12.2020)
Get full text
Journal Article
Pyrrolopyrimidine based CSF1R inhibitors: Attempted departure from Flatland
Bjørnstad, Frithjof, Havik, Simen, Aarhus, Thomas Ihle, Mahdi, Iktedar, Unger, Anke, Habenberger, Peter, Degenhart, Carsten, Eickhoff, Jan, Klebl, Bert M., Sundby, Eirik, Hoff, Bård Helge
Published in European journal of medicinal chemistry (05.02.2024)
Published in European journal of medicinal chemistry (05.02.2024)
Get full text
Journal Article
A novel CDK7 inhibitor of the Pyrazolotriazine class exerts broad-spectrum antiviral activity at nanomolar concentrations
Hutterer, Corina, Eickhoff, Jan, Milbradt, Jens, Korn, Klaus, Zeitträger, Isabel, Bahsi, Hanife, Wagner, Sabrina, Zischinsky, Gunther, Wolf, Alexander, Degenhart, Carsten, Unger, Anke, Baumann, Matthias, Klebl, Bert, Marschall, Manfred
Published in Antimicrobial agents and chemotherapy (01.04.2015)
Published in Antimicrobial agents and chemotherapy (01.04.2015)
Get full text
Journal Article
Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer
Lücking, Ulrich, Scholz, Arne, Lienau, Philip, Siemeister, Gerhard, Kosemund, Dirk, Bohlmann, Rolf, Briem, Hans, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Denner, Karsten, Bömer, Ulf, Schäfer, Martina, Eis, Knut, Valencia, Ray, Ince, Stuart, von Nussbaum, Franz, Mumberg, Dominik, Ziegelbauer, Karl, Klebl, Bert, Choidas, Axel, Nussbaumer, Peter, Baumann, Matthias, Schultz‐Fademrecht, Carsten, Rühter, Gerd, Eickhoff, Jan, Brands, Michael
Published in ChemMedChem (08.11.2017)
Published in ChemMedChem (08.11.2017)
Get full text
Journal Article
Cytomegalovirus cyclin-dependent kinase ortholog vCDK/pUL97 undergoes regulatory interaction with human cyclin H and CDK7 to codetermine viral replication efficiency
Schütz, Martin, Wangen, Christina, Sommerer, Mona, Kögler, Melanie, Eickhoff, Jan, Degenhart, Carsten, Klebl, Bert, Naing, Zin, Egilmezer, Ece, Hamilton, Stuart T., Rawlinson, William D., Sticht, Heinrich, Marschall, Manfred
Published in Virus research (02.10.2023)
Published in Virus research (02.10.2023)
Get full text
Journal Article
Insight into Targeting Exon20 Insertion Mutations of the Epidermal Growth Factor Receptor with Wild Type-Sparing Inhibitors
Lategahn, Jonas, Tumbrink, Hannah L., Schultz-Fademrecht, Carsten, Heimsoeth, Alena, Werr, Lisa, Niggenaber, Janina, Keul, Marina, Parmaksiz, Fatma, Baumann, Matthias, Menninger, Sascha, Zent, Eldar, Landel, Ina, Weisner, Jörn, Jeyakumar, Kirujan, Heyden, Leonie, Russ, Nicole, Müller, Fabienne, Lorenz, Carina, Brägelmann, Johannes, Spille, Inga, Grabe, Tobias, Müller, Matthias P., Heuckmann, Johannes M., Klebl, Bert M., Nussbaumer, Peter, Sos, Martin L., Rauh, Daniel
Published in Journal of medicinal chemistry (12.05.2022)
Published in Journal of medicinal chemistry (12.05.2022)
Get full text
Journal Article
Amorfrutins are potent antidiabetic dietary natural products
Weidner, Christopher, de Groot, Jens C, Prasad, Aman, Freiwald, Anja, Quedenau, Claudia, Kliem, Magdalena, Witzke, Annabell, Kodelja, Vitam, Han, Chung-Ting, Giegold, Sascha, Baumann, Matthias, Klebl, Bert, Siems, Karsten, Müller-Kuhrt, Lutz, Schürmann, Annette, Schüler, Rita, Pfeiffer, Andreas F. H, Schroeder, Frank C, Büssow, Konrad, Sauer, Sascha
Published in Proceedings of the National Academy of Sciences - PNAS (08.05.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (08.05.2012)
Get full text
Journal Article
Cyclin-Dependent Kinase 7 Controls mRNA Synthesis by Affecting Stability of Preinitiation Complexes, Leading to Altered Gene Expression, Cell Cycle Progression, and Survival of Tumor Cells
Kelso, Timothy W. R., Baumgart, Karen, Eickhoff, Jan, Albert, Thomas, Antrecht, Claudia, Lemcke, Sarah, Klebl, Bert, Meisterernst, Michael
Published in Molecular and cellular biology (01.10.2014)
Published in Molecular and cellular biology (01.10.2014)
Get full text
Journal Article
ComplexEye: a multi-lens array microscope for high-throughput embedded immune cell migration analysis
Cibir, Zülal, Hassel, Jacqueline, Sonneck, Justin, Kowitz, Lennart, Beer, Alexander, Kraus, Andreas, Hallekamp, Gabriel, Rosenkranz, Martin, Raffelberg, Pascal, Olfen, Sven, Smilowski, Kamil, Burkard, Roman, Helfrich, Iris, Tuz, Ali Ata, Singh, Vikramjeet, Ghosh, Susmita, Sickmann, Albert, Klebl, Anne-Kathrin, Eickhoff, Jan Eike, Klebl, Bert, Seidl, Karsten, Chen, Jianxu, Grabmaier, Anton, Viga, Reinhard, Gunzer, Matthias
Published in Nature communications (11.12.2023)
Published in Nature communications (11.12.2023)
Get full text
Journal Article
Protein Kinase G from Pathogenic Mycobacteria Promotes Survival within Macrophages
Walburger, Anne, Koul, Anil, Ferrari, Giorgio, Nguyen, Liem, Prescianotto-Baschong, Cristina, Huygen, Kris, Klebl, Bert, Thompson, Charles, Bacher, Gerald, Pieters, Jean
Published in Science (American Association for the Advancement of Science) (18.06.2004)
Published in Science (American Association for the Advancement of Science) (18.06.2004)
Get full text
Journal Article
Discovery of tetrazolo-pyridazine-based small molecules as inhibitors of MACC1-driven cancer metastasis
Yan, Shixian, Schöpe, Paul Curtis, Lewis, Joe, Putzker, Kerstin, Uhrig, Ulrike, Specker, Edgar, von Kries, Jens Peter, Lindemann, Peter, Omran, Anahid, Sanchez-Ibarra, Hector E., Unger, Anke, Zischinsky, Mia-Lisa, Klebl, Bert, Walther, Wolfgang, Nazaré, Marc, Kobelt, Dennis, Stein, Ulrike
Published in Biomedicine & pharmacotherapy (01.12.2023)
Published in Biomedicine & pharmacotherapy (01.12.2023)
Get full text
Journal Article
Dual Inhibition of GSK3β and CDK5 Protects the Cytoskeleton of Neurons from Neuroinflammatory-Mediated Degeneration In Vitro and In Vivo
Reinhardt, Lydia, Kordes, Susanne, Reinhardt, Peter, Glatza, Michael, Baumann, Matthias, Drexler, Hannes C.A., Menninger, Sascha, Zischinsky, Gunther, Eickhoff, Jan, Fröb, Claudia, Bhattarai, Prabesh, Arulmozhivarman, Guruchandar, Marrone, Lara, Janosch, Antje, Adachi, Kenjiro, Stehling, Martin, Anderson, Eric N., Abo-Rady, Masin, Bickle, Marc, Pandey, Udai Bhan, Reimer, Michell M., Kizil, Caghan, Schöler, Hans R., Nussbaumer, Peter, Klebl, Bert, Sterneckert, Jared L.
Published in Stem cell reports (05.03.2019)
Published in Stem cell reports (05.03.2019)
Get full text
Journal Article
Anti-leukemic effect of CDK9 inhibition in T-cell prolymphocytic leukemia
Johansson, Patricia, Dierichs, Laura, Klein-Hitpass, Ludger, Bergmann, Anke K., Möllmann, Michael, Menninger, Sascha, Habenberger, Peter, Klebl, Bert, Siveke, Jens T., Dührsen, Ulrich, Choidas, Axel, Dürig, Jan
Published in Therapeutic advances in hematology (01.10.2020)
Published in Therapeutic advances in hematology (01.10.2020)
Get full text
Journal Article
Profiling of ERBB receptors and downstream pathways reveals selectivity and hidden properties of ERBB4 antagonists
Popović, Lukša, Wintgens, Jan P., Wu, Yuxin, Brankatschk, Ben, Menninger, Sascha, Degenhart, Carsten, Jensen, Niels, Wichert, Sven P., Klebl, Bert, Rossner, Moritz J., Wehr, Michael C.
Published in iScience (16.02.2024)
Published in iScience (16.02.2024)
Get full text
Journal Article
An Antiherpesviral Host-Directed Strategy Based on CDK7 Covalently Binding Drugs: Target-Selective, Picomolar-Dose, Cross-Virus Reactivity
Yu, DongHoon, Wagner, Sabrina, Schütz, Martin, Jeon, Yeejin, Seo, Mooyoung, Kim, Jaeseung, Brückner, Nadine, Kicuntod, Jintawee, Tillmanns, Julia, Wangen, Christina, Hahn, Friedrich, Kaufer, Benedikt B, Neipel, Frank, Eickhoff, Jan, Klebl, Bert, Nam, Kiyean, Marschall, Manfred
Published in Pharmaceutics (23.01.2024)
Published in Pharmaceutics (23.01.2024)
Get full text
Journal Article
Assessment of Covalently Binding Warhead Compounds in the Validation of the Cytomegalovirus Nuclear Egress Complex as an Antiviral Target
Tillmanns, Julia, Häge, Sigrun, Borst, Eva Maria, Wardin, Julia, Eickhoff, Jan, Klebl, Bert, Wagner, Sabrina, Wangen, Christina, Hahn, Friedrich, Socher, Eileen, Marschall, Manfred
Published in Cells (Basel, Switzerland) (01.04.2023)
Published in Cells (Basel, Switzerland) (01.04.2023)
Get full text
Journal Article
The E3 ligase Cbl-b and TAM receptors regulate cancer metastasis via natural killer cells
Paolino, Magdalena, Choidas, Axel, Wallner, Stephanie, Pranjic, Blanka, Uribesalgo, Iris, Loeser, Stefanie, Jamieson, Amanda M, Langdon, Wallace Y, Ikeda, Fumiyo, Fededa, Juan Pablo, Cronin, Shane J, Nitsch, Roberto, Schultz-Fademrecht, Carsten, Eickhoff, Jan, Menninger, Sascha, Unger, Anke, Torka, Robert, Gruber, Thomas, Hinterleitner, Reinhard, Baier, Gottfried, Wolf, Dominik, Ullrich, Axel, Klebl, Bert M, Penninger, Josef M
Published in Nature (London) (27.03.2014)
Published in Nature (London) (27.03.2014)
Get full text
Journal Article
Characterization of the Antibacterial Activity of Quinone-Based Compounds Originating from the Alnumycin Biosynthetic Gene Cluster of a Streptomyces Isolate
Sagurna, Leonie, Heinrich, Sascha, Kaufmann, Lara-Sophie, Rückert-Reed, Christian, Busche, Tobias, Wolf, Alexander, Eickhoff, Jan, Klebl, Bert, Kalinowski, Jörn, Bandow, Julia E
Published in Antibiotics (Basel) (28.06.2023)
Published in Antibiotics (Basel) (28.06.2023)
Get full text
Journal Article