Potent and Selective BACE-1 Peptide Inhibitors Lower Brain Aβ Levels Mediated by Brain Shuttle Transport
Ruderisch, Nadine, Schlatter, Daniel, Kuglstatter, Andreas, Guba, Wolfgang, Huber, Sylwia, Cusulin, Carlo, Benz, Jörg, Rufer, Arne Christian, Hoernschemeyer, Joerg, Schweitzer, Christophe, Bülau, Tina, Gärtner, Achim, Hoffmann, Eike, Niewoehner, Jens, Patsch, Christoph, Baumann, Karlheinz, Loetscher, Hansruedi, Kitas, Eric, Freskgård, Per-Ola
Published in EBioMedicine (01.10.2017)
Published in EBioMedicine (01.10.2017)
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Journal Article
Substituted 2-oxo-azepane derivatives are potent, orally active γ-secretase inhibitors
Kitas, Eric A., Galley, Guido, Jakob-Roetne, Roland, Flohr, Alexander, Wostl, Wolfgang, Mauser, Harald, Alker, André M., Czech, Christian, Ozmen, Laurence, David-Pierson, Pascale, Reinhardt, Dieter, Jacobsen, Helmut
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
Endothelin-Converting Enzyme-1 Inhibition and Growth of Human Glioblastoma Cells
Berger, Yann, Dehmlow, Henrietta, Blum-Kaelin, Denise, Kitas, Eric A, Löffler, Bernd-Michael, Aebi, Johannes D, Juillerat-Jeanneret, Lucienne
Published in Journal of medicinal chemistry (27.01.2005)
Published in Journal of medicinal chemistry (27.01.2005)
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Journal Article
SEAP expression in transiently transfected mammalian cells grown in serum-free suspension culture
SCHLAEGER, Ernst-Jürgen, KITAS, Eric A, DORN, Arnulf
Published in Cytotechnology (Dordrecht) (01.05.2003)
Published in Cytotechnology (Dordrecht) (01.05.2003)
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Journal Article
riDOM, a cell penetrating peptide. Interaction with phospholipid bilayers
Québatte, Gabriela, Kitas, Eric, Seelig, Joachim
Published in Biochimica et biophysica acta (01.03.2014)
Published in Biochimica et biophysica acta (01.03.2014)
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Journal Article
riDOM, a Cell-Penetrating Peptide. Interaction with DNA and Heparan Sulfate
Québatte, Gabriela, Kitas, Eric, Seelig, Joachim
Published in The journal of physical chemistry. B (19.09.2013)
Published in The journal of physical chemistry. B (19.09.2013)
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Journal Article
Substrate specificities of catalytic fragments of protein tyrosine phosphatases (HPTPβ, LAR, and CD45) toward phosphotyrosylpeptide substrates and thiophosphotyrosylated peptides as inhibitors
Cho, Hyeongjin, Krishnaraj, Ravichandran, Walsh, Christopher T., Itoh, Michyasu, Saito, Haruo, Kitas, Eric, Bannwarth, Willi
Published in Protein science (01.06.1993)
Published in Protein science (01.06.1993)
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Journal Article
암의 치료를 위한 면역요법
ZIGLER MAYA, KITAS ERIC, BAJIC DAVOR, BROKA DERRICK, POMBO VILLAR ESTEBAN, SCHADE BABETTE
Year of Publication 13.06.2023
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Year of Publication 13.06.2023
Patent
Cargo Delivery into the Brain by in vivo identified Transport Peptides
Urich, Eduard, Schmucki, Roland, Ruderisch, Nadine, Kitas, Eric, Certa, Ulrich, Jacobsen, Helmut, Schweitzer, Christophe, Bergadano, Alessandra, Ebeling, Martin, Loetscher, Hansruedi, Freskgård, Per-Ola
Published in Scientific reports (28.09.2015)
Published in Scientific reports (28.09.2015)
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Journal Article
1170 EGFR-Ta:RNA: multimodal mechanism of action potentiates immune checkpoint inhibitor activity
Schade, Babette, Broka, Derrick, De Feyter, Caroline, Klein, Shoshana, Shir, Alexei, Levitzki, Alexander, Bajic, Davor, Lucia D’Amico, Colecchia, David, Kitas, Eric, Jarzebinska, Anita, Pombo-Villar, Esteban, Zigler, Maya
Published in Journal for immunotherapy of cancer (01.11.2022)
Published in Journal for immunotherapy of cancer (01.11.2022)
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Journal Article
Protease-triggered siRNA delivery vehicles
Rozema, David B, Blokhin, Andrei V, Wakefield, Darren H, Benson, Jonathan D, Carlson, Jeffrey C, Klein, Jason J, Almeida, Lauren J, Nicholas, Anthony L, Hamilton, Holly L, Chu, Qili, Hegge, Julia O, Wong, So C, Trubetskoy, Vladimir S, Hagen, Collin M, Kitas, Eric, Wolff, Jon A, Lewis, David L
Published in Journal of controlled release (10.07.2015)
Published in Journal of controlled release (10.07.2015)
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Journal Article
암의 치료를 위한 면역요법
COLECCHIA DAVID, ZIGLER MAYA, KITAS ERIC, JARZEBINSKA ANITA, LEVITZKI ALEXANDER, BAJIC DAVOR, BROKA DERRICK, POMBO VILLAR ESTEBAN, SHIR ALEXEI, D'AMICO LUCIA
Year of Publication 06.12.2021
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Year of Publication 06.12.2021
Patent
Purification and characterization of active recombinant human napsin A
Schauer‐Vukasinovic, Vesna, Bur, Daniel, Kitas, Eric, Schlatter, Daniel, Rossé, Gerard, Lahm, Hans‐Werner, Giller, Thomas
Published in European journal of biochemistry (01.05.2000)
Published in European journal of biochemistry (01.05.2000)
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Journal Article
Allosteric FBPase inhibitors gain 10(5) times in potency when simultaneously binding two neighboring AMP sites
Hebeisen, Paul, Kuhn, Bernd, Kohler, Philipp, Gubler, Marcel, Huber, Walter, Kitas, Eric, Schott, Brigitte, Benz, Jörg, Joseph, Catherine, Ruf, Armin
Published in Bioorganic & medicinal chemistry letters (15.08.2008)
Published in Bioorganic & medicinal chemistry letters (15.08.2008)
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Journal Article