Novel inhibitors of VEGF receptors-1 and -2 based on azole-5-carboxamide templates
Kiselyov, Alexander S., Milligan, Daniel, Ouyang, Xiaohu
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and II
Duncton, Matthew A.J., Piatnitski, Evgueni L., Katoch-Rouse, Reeti, Smith, Leon M., Kiselyov, Alexander S., Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Virtual and biomolecular screening converge on a selective agonist for GPR30
Oprea, Tudor I, Prossnitz, Eric R, Bologa, Cristian G, Revankar, Chetana M, Young, Susan M, Edwards, Bruce S, Arterburn, Jeffrey B, Kiselyov, Alexander S, Parker, Matthew A, Tkachenko, Sergey E, Savchuck, Nikolay P, Sklar, Larry A
Published in Nature chemical biology (01.04.2006)
Published in Nature chemical biology (01.04.2006)
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Quantitative 3D reconstruction of viral vector distribution in rodent and ovine brain following local delivery
Poceviciute, Roberta, Mitchell, Kenneth, Nikolakopoulou, Angeliki Maria, Cho, Suehyun K., Ma, Xiaobo, Chen, Phillip, Figueroa, Samantha, Sarmiento, Ethan J., Singh, Aryan, Hartstein, Oren, Loudon, William G., Cros, Florent, Kiselyov, Alexander S.
Published in Neuroimage. Reports (01.12.2024)
Published in Neuroimage. Reports (01.12.2024)
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Journal Article
3,4-Disubstituted isothiazoles: Novel potent inhibitors of VEGF receptors 1 and 2
Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
The o-Amino-Trifluoromethyl Functionality as a Novel Synthon for 4-Fluoroquinolines
Strekowski, Lucjan, Kiselyov, Alexander S, Hojjat, Maryam
Published in Journal of organic chemistry (01.10.1994)
Published in Journal of organic chemistry (01.10.1994)
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Journal Article
Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines
Ouyang, Xiaohu, Piatnitski, Evgueni L., Pattaropong, Vatee, Chen, Xiaoling, He, Hai-Ying, Kiselyov, Alexander S., Velankar, Avdhoot, Kawakami, Joel, Labelle, Marc, Smith, Leon, Lohman, Julia, Lee, Sui Ping, Malikzay, Asra, Fleming, James, Gerlak, Jason, Wang, Ying, Rosler, Robin L., Zhou, Kai, Mitelman, Stan, Camara, Margarita, Surguladze, David, Doody, Jacqueline F., Tuma, M. Carolina
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Journal Article
Arylphthalazines as potent, and orally bioavailable inhibitors of VEGFR-2
Duncton, Matthew A.J., Piatnitski Chekler, Eugene L., Katoch-Rouse, Reeti, Sherman, Dan, Wong, Wai C., Smith, Leon M., Kawakami, Joel K., Kiselyov, Alexander S., Milligan, Daniel L., Balagtas, Chris, Hadari, Yaron R., Wang, Ying, Patel, Sheetal N., Rolster, Robin L., Tonra, James R., Surguladze, David, Mitelman, Stan, Kussie, Paul, Bohlen, Peter, Doody, Jacqueline F.
Published in Bioorganic & medicinal chemistry (15.01.2009)
Published in Bioorganic & medicinal chemistry (15.01.2009)
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Journal Article
Discovery of Dual VEGFR-2 and Tubulin Inhibitors with in Vivo Efficacy
Chekler, Eugene L. Piatnitski, Kiselyov, Alexander S, Ouyang, Xiaohu, Chen, Xiaoling, Pattaropong, Vatee, Wang, Ying, Tuma, M. Carolina, Doody, Jacqueline F
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
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Journal Article
Design and chemical synthesis of [1,2,4]triazol[1,5- c]pyrimidin-5-yl amines, a novel class of VEGFR-2 kinase inhibitors
Kiselyov, Alexander S., Piatnitski Chekler, Eugene L., Chernisheva, Natalia B., Salamandra, Lev K., Semenov, Victor V.
Published in Tetrahedron letters (01.07.2009)
Published in Tetrahedron letters (01.07.2009)
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Journal Article
1-[4-(1 H-Benzoimidazol-2-yl)-phenyl]-3-[4-(1 H-benzoimidazol-2-yl)-phenyl]-urea derivatives as small molecule heparanase inhibitors
Pan, Weitao, Miao, Hua-Quan, Xu, Yong-Jiang, Navarro, Elizabeth C., Tonra, James R., Corcoran, Erik, Lahiji, Armin, Kussie, Paul, Kiselyov, Alexander S., Wong, Wai C., Liu, Hu
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
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Journal Article
Hetaryl imidazoles: A novel dual inhibitors of VEGF receptors I and II
Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V.
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
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Journal Article
Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors
Ouyang, Xiaohu, Chen, Xiaoling, Piatnitski, Evgueni L., Kiselyov, Alexander S., He, Hai-Ying, Mao, Yunyu, Pattaropong, Vatee, Yu, Yang, Kim, Ki H., Kincaid, John, Smith, Leon, Wong, Wai C., Lee, Sui Ping, Milligan, Daniel L., Malikzay, Asra, Fleming, James, Gerlak, Jason, Deevi, Dhanvanthri, Doody, Jacqueline F., Chiang, Hui-Hsien, Patel, Sheetal N., Wang, Ying, Rolser, Robin L., Kussie, Paul, Labelle, Marc, Tuma, M. Carolina
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
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Journal Article
4-(Azolylphenyl)-phthalazin-1-amines: Novel Inhibitors of VEGF Receptors I and II
Kiselyov, Alexander S., Semenov, Victor V., Milligan, Daniel
Published in Chemical biology & drug design (01.12.2006)
Published in Chemical biology & drug design (01.12.2006)
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Journal Article
Arylphthalazines: Identification of a new phthalazine chemotype as inhibitors of VEGFR kinase
Piatnitski, Evgueni L., Duncton, Matthew A.J., Kiselyov, Alexander S., Katoch-Rouse, Reeti, Sherman, Dan, Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
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