Design and synthesis of a highly selective, orally active and potent anaplastic lymphoma kinase inhibitor (CH5424802)
Kinoshita, Kazutomo, Asoh, Kohsuke, Furuichi, Noriyuki, Ito, Toshiya, Kawada, Hatsuo, Hara, Sousuke, Ohwada, Jun, Miyagi, Takuho, Kobayashi, Takamitsu, Takanashi, Kenji, Tsukaguchi, Toshiyuki, Sakamoto, Hiroshi, Tsukuda, Takuo, Oikawa, Nobuhiro
Published in Bioorganic & medicinal chemistry (01.02.2012)
Published in Bioorganic & medicinal chemistry (01.02.2012)
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Journal Article
Discovery of CH7057288 as an Orally Bioavailable, Selective, and Potent pan-TRK Inhibitor
Ito, Toshiya, Kinoshita, Kazutomo, Tomizawa, Masaki, Shinohara, Shojiro, Nishii, Hiroki, Matsushita, Masayuki, Hattori, Kazuo, Kohchi, Yasunori, Kohchi, Masami, Hayase, Tadakatsu, Watanabe, Fumio, Hasegawa, Kiyoshi, Tanaka, Hiroshi, Kuramoto, Shino, Takanashi, Kenji, Oikawa, Nobuhiro
Published in Journal of medicinal chemistry (22.09.2022)
Published in Journal of medicinal chemistry (22.09.2022)
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Development of a Scalable Manufacturing Process for Alectinib with a Concise Preparation of the Indole-Containing Tetracyclic Core
Oki, Tomohiro, Tsukazaki, Masao, Shiina, Junichi, Fukuda, Hiroshi, Yamawaki, Minoru, Kito, Yasushi, Ishizawa, Takenori, Kinoshita, Kazutomo, Hara, Sosuke, Furuichi, Noriyuki, Kawada, Hatsuo, Ito, Toshiya, Tanaka, Kota, Maruyama, Noriaki, Tamaru, Daisuke, Ichige, Takahiro, Koizumi, Masatoshi, Hosoya, Yosuke, Kimura, Masahiro, Yamaguchi, Mami, Sato, Shigeki, Miyazaki, Yuta, Toya, Azusa, Iwamura, Hiroshi, Maeda, Kenji
Published in Organic process research & development (22.10.2024)
Published in Organic process research & development (22.10.2024)
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Journal Article
9-Substituted 6,6-Dimethyl-11-oxo-6,11-dihydro-5H-benzo[b]carbazoles as Highly Selective and Potent Anaplastic Lymphoma Kinase Inhibitors
Kinoshita, Kazutomo, Kobayashi, Takamitsu, Asoh, Kohsuke, Furuichi, Noriyuki, Ito, Toshiya, Kawada, Hatsuo, Hara, Sousuke, Ohwada, Jun, Hattori, Kazuo, Miyagi, Takuho, Hong, Woo-Sang, Park, Min-Jeong, Takanashi, Kenji, Tsukaguchi, Toshiyuki, Sakamoto, Hiroshi, Tsukuda, Takuo, Oikawa, Nobuhiro
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Journal Article
Discovery of novel tetracyclic compounds as anaplastic lymphoma kinase inhibitors
Kinoshita, Kazutomo, Ono, Yoshiyuki, Emura, Takashi, Asoh, Kohsuke, Furuichi, Noriyuki, Ito, Toshiya, Kawada, Hatsuo, Tanaka, Shota, Morikami, Kenji, Tsukaguchi, Toshiyuki, Sakamoto, Hiroshi, Tsukuda, Takuo, Oikawa, Nobuhiro
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
COMPOUND LIBRARY
HAYASE, Tadakatsu, NISHIMOTO, Masahiro, SAITO, Masato, KINOSHITA, Kazutomo, TSUCHIYA, Satoshi, NOMURA, Kenichi, EMURA, Takashi, KAMAKURA, Daiki, IIKURA, Hitoshi, ITO, Taisuke, OGAWA, Hiroko, ORI, Kazutomo, MURATA, Yoshihisa
Year of Publication 14.07.2022
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Year of Publication 14.07.2022
Patent
9-Substituted 6,6-Dimethyl-11-oxo-6,11-dihydro-5 H -benzo[ b ]carbazoles as Highly Selective and Potent Anaplastic Lymphoma Kinase Inhibitors
Kinoshita, Kazutomo, Kobayashi, Takamitsu, Asoh, Kohsuke, Furuichi, Noriyuki, Ito, Toshiya, Kawada, Hatsuo, Hara, Sousuke, Ohwada, Jun, Hattori, Kazuo, Miyagi, Takuho, Hong, Woo-Sang, Park, Min-Jeong, Takanashi, Kenji, Tsukaguchi, Toshiyuki, Sakamoto, Hiroshi, Tsukuda, Takuo, Oikawa, Nobuhiro
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Journal Article
Abstract 3593: Generation of a potent and selective inhibitor of ALK, CH5424802, showing superior oral bioavailability, PK profile and in vivo efficacy
Oikawa, Nobuhiro, Kinoshita, Kazutomo, Asoh, Kohsuke, Furuichi, Noriyuki, Itoh, Toshiya, Kawada, Hatsuo, Hara, Sosuke, Miyagi, Takuho, Ohwada, Jun, Taniguchi, Saori, Hattori, Kazuo, Tsukuda, Takuo, Takanashi, Kenji, Sakamoto, Hiroshi, Tsukaguchi, Toshiyuki, Ishii, Nobuya, Aoki, Yuko, Shimma, Nobuo
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Design and evaluation of new antipsoriatic antedrug candidates having 16-en-22-oxa-vitamin D3 structures
SHIMIZU, Kazuki, KAWASE, Akira, YAMAGUCHI, Koji, MORITA, Keiichi, SEKIGUCHI, Nobuo, YAMAMOTO, Tessai, MATSUSHITA, Tomochika, SHIMAOKA, Shin, SUGITA, Atsuko, MORIKAWA, Kazumi, HANEISHI, Tsuyoshi, KATO, Yasuharu, KINOSHITA, Kazutomo, OHMORI, Masayuki, FURUTA, Yoshiyuki, EMURA, Takashi, KATO, Nobuaki, MITSUI, Tetsuya
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
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Journal Article
Design and evaluation of new antipsoriatic antedrug candidates having 16-en-22-oxa-vitamin D 3 structures
Shimizu, Kazuki, Kawase, Akira, Haneishi, Tsuyoshi, Kato, Yasuharu, Kinoshita, Kazutomo, Ohmori, Masayuki, Furuta, Yoshiyuki, Emura, Takashi, Kato, Nobuaki, Mitsui, Tetsuya, Yamaguchi, Koji, Morita, Keiichi, Sekiguchi, Nobuo, Yamamoto, Tessai, Matsushita, Tomochika, Shimaoka, Shin, Sugita, Atsuko, Morikawa, Kazumi
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
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TETRACYCLIC COMPOUND
SAKAMOTO HIROSHI, ONO YOSHIYUKI, EMURA TAKASHI, HONG WOOSANG, FURUICHI NORIYUKI, PARK MINJEONG, KATO YASUHARU, KAWADA HATSUO, KINOSHITA KAZUTOMO, ISHII NOBUYA, ITO TOSHIYA, ASOH KOHSUKE, MORIKAMI KENJI, OIKAWA NOBUHIRO
Year of Publication 16.12.2010
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Year of Publication 16.12.2010
Patent
TETRACYCLIC COMPOUND
SAKAMOTO HIROSHI, ONO YOSHIYUKI, EMURA TAKASHI, PARK, MIN JEONG, FURUICHI NORIYUKI, KATO YASUHARU, KAWADA HATSUO, KINOSHITA KAZUTOMO, ISHII NOBUYA, ITO TOSHIYA, ASOH KOHSUKE, MORIKAMI KENJI, OIKAWA NOBUHIRO, HONG, WOO SANG
Year of Publication 12.04.2012
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Year of Publication 12.04.2012
Patent
Design and evaluation of new antipsoriatic antedrug candidates having 16-en- 22-oxa-vitamin D sub(3) structures
Shimizu, Kazuki, Kawase, Akira, Haneishi, Tsuyoshi, Kato, Yasuharu, Kinoshita, Kazutomo, Ohmori, Masayuki, Furuta, Yoshiyuki, Emura, Takashi, Kato, Nobuaki, Mitsui, Tetsuya, Yamaguchi, Koji, Morita, Keiichi, Sekiguchi, Nobuo, Yamamoto, Tessai, Matsushita, Tomochika, Shimaoka, Shin, Sugita, Atsuko, Morikawa, Kazumi
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
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Journal Article
METHOD FOR PRODUCING VITAMIN D DERIVATIVE UTILIZING PHOTOREACTION
KATO, YASUHARU, KITOH, YASUSHI, KOBAYASHI, MIO, KAWASE, AKIRA, HANEISHI, TSUYOSHI, MARUYAMA, NORIAKI, KINOSHITA, KAZUTOMO, IKEDA, TAKUMA
Year of Publication 07.06.2007
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Year of Publication 07.06.2007
Patent
METHOD OF ASSAYING ACTIVITY OF BINDING TO VITAMIN D3 RECEPTOR USING FLUORESCENCE POLARIZATION
ITO, SUSUMU, KAWASE, AKIRA, ABE, SATOSHI, KINOSHITA, KAZUTOMO, KOBAYASHI, TAKAMITSU
Year of Publication 28.08.2003
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Year of Publication 28.08.2003
Patent
VITAMIN D DERIVATIVES
KAWASE, AKIRA, SHIMIZU, KAZUKI, KINOSHITA, KAZUTOMO, SHIMIZU, HITOSHI, EMURA, TAKASHI
Year of Publication 25.10.2001
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Year of Publication 25.10.2001
Patent
COMPOUND LIBRARY
HAYASE, Tadakatsu, NISHIMOTO, Masahiro, SAITO, Masato, KINOSHITA, Kazutomo, TSUCHIYA, Satoshi, NOMURA, Kenichi, EMURA, Takashi, KAMAKURA, Daiki, IIKURA, Hitoshi, ITO, Taisuke, OGAWA, Hiroko, ORI, Kazutomo, MURATA, Yoshihisa
Year of Publication 15.11.2023
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Year of Publication 15.11.2023
Patent
TETRACYCLIC COMPOUND
ONO, Yoshiyuki, ISHII, Nobuya, MORIKAMI, Kenji, KAWADA, Hatsuo, KATO, Yasuharu, KINOSHITA, Kazutomo, ITO, Toshiya, OIKAWA, Nobuhiro, PARK, MinJeong, FURUICHI, Noriyuki, EMURA, Takashi, SAKAMOTO, Hiroshi, ASOH, Kohsuke, HONG, WooSang
Year of Publication 11.05.2023
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Year of Publication 11.05.2023
Patent
TETRACYCLIC COMPOUND
ONO, Yoshiyuki, ISHII, Nobuya, MORIKAMI, Kenji, KAWADA, Hatsuo, KATO, Yasuharu, KINOSHITA, Kazutomo, ITO, Toshiya, OIKAWA, Nobuhiro, PARK, MinJeong, FURUICHI, Noriyuki, EMURA, Takashi, SAKAMOTO, Hiroshi, ASOH, Kohsuke, HONG, WooSang
Year of Publication 29.09.2022
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Year of Publication 29.09.2022
Patent