Efficient, enantioselective synthesis of a β,β-disubstituted carboxylic acid by Ru-XylPhanePhos-catalyzed asymmetric hydrogenation
Grasa, Gabriela A., Zanotti-Gerosa, Antonio, Ghosh, Shyamali, Teleha, Christopher A., Kinney, William A., Maryanoff, Bruce E.
Published in Tetrahedron letters (01.09.2008)
Published in Tetrahedron letters (01.09.2008)
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Claisen rearrangement of 6-alkenyl-2-methylenetetrahydropyrans. A new approach to annulated 4-cyclooctenones and a stereospecific synthesis of precapnelladiene
Kinney, William A, Coghlan, Michael J, Paquette, Leo A
Published in Journal of the American Chemical Society (01.10.1984)
Published in Journal of the American Chemical Society (01.10.1984)
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Synthesis of an αvβ3 integrin antagonist intermediate via asymmetric hydrogenation of an α,β-unsaturated ester with BoPhoz-iridium and BoPhoz-rhodium catalysts
Zanotti-Gerosa, Antonio, Kinney, William A., Grasa, Gabriela A., Medlock, Jonathan, Seger, Andreas, Ghosh, Shyamali, Teleha, Christopher A., Maryanoff, Bruce E.
Published in Tetrahedron: asymmetry (01.05.2008)
Published in Tetrahedron: asymmetry (01.05.2008)
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Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alpha(V)beta(3)/alpha(V)beta(5) integrin antagonist. Enantioselective synthesis and stereochemical studies
Kinney, William A., Teleha, Christopher A., Thompson, Andrew S., Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C., McComsey, David F., Santulli, Rosemary J., Maryanoff, Bruce E.
Published in Journal of organic chemistry (21.03.2008)
Published in Journal of organic chemistry (21.03.2008)
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Journal Article
Synthesis of an alpha(v)beta(3) integrin antagonist intermediate via asymmetric hydrogenation of an alpha,beta-unsaturated ester with BoPhoz-iridium and BoPhoz-rhodium catalysts
Zanotti-Gerosa, Antonio, Kinney, William A., Grasa, Gabriela A., Medlock, Jonathan, Seger, Andreas, Ghosh, Shyamali, Teleha, Christopher A., Maryanoff, Bruce E.
Published in Tetrahedron: asymmetry (01.05.2008)
Published in Tetrahedron: asymmetry (01.05.2008)
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Journal Article
N-Phenyl-2-pyridinecarbothioamides as gastric mucosal protectants
Kinney, William A, Lee, Nancy E, Blank, Robert M, Demerson, Christopher A, Sarnella, Carol S, Scherer, Noreen T, Mir, G. Nabi, Borella, Luis E, DiJoseph, John F, Wells, Cheryl
Published in Journal of medicinal chemistry (01.01.1990)
Published in Journal of medicinal chemistry (01.01.1990)
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Squalamine inhibits angiogenesis and solid tumor growth in vivo and perturbs embryonic vasculature
SILLS, A. K, WILLIAMS, J. I, KINNEY, W. A, CHAO, T. L, DONOWITZ, M, LATERRA, J, ZASLOFF, M, BREM, H, TYLER, B. M, EPSTEIN, D. S, SIPOS, E. P, DAVIS, J. D, MCLANE, M. P, PITCHFORD, S, CHESHIRE, K, GANNON, F. H
Published in Cancer research (Chicago, Ill.) (01.07.1998)
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Published in Cancer research (Chicago, Ill.) (01.07.1998)
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FUNCTIONALIZED 1,3-BENZENE DIOLS AND THEIR METHOD OF USE FOR THE TREATMENT OF INFLAMMATION AND PAIN
MCDONNELL, Mark E, PETKANAS, Dean, BRENNEMAN, Douglas, KINNEY, William A
Year of Publication 25.04.2024
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Year of Publication 25.04.2024
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