Generation of novel, potent urotensin-II receptor antagonists by alkylation–cyclization of isoindolinone C3-carbanions
Luci, Diane K., Lawson, Edward C., Ghosh, Shyamali, Kinney, William A., Smith, Charles E., Qi, Jenson, Wang, Yuanping, Minor, Lisa K., Maryanoff, Bruce E.
Published in Tetrahedron letters (02.09.2009)
Published in Tetrahedron letters (02.09.2009)
Get full text
Journal Article
Synthesis of Squalamine Utilizing a Readily Accessible Spermidine Equivalent
Zhang, Xuehai, Rao, Meenakshi N, Jones, Stephen R, Shao, Bin, Feibush, Penina, McGuigan, Melissa, Tzodikov, Nathan, Feibush, Binyamin, Sharkansky, Ilya, Snyder, Brad, Mallis, Larry M, Sarkahian, Ani, Wilder, Susan, Turse, Joshua E, Kinney, William A, Kjærsgaard, Hans Jørgen, Michalak, Ronald S
Published in Journal of organic chemistry (13.11.1998)
Published in Journal of organic chemistry (13.11.1998)
Get full text
Journal Article
Studies with an orally bioavailable alpha V integrin antagonist in animal models of ocular vasculopathy: retinal neovascularization in mice and retinal vascular permeability in diabetic rats
Santulli, Rosemary J, Kinney, William A, Ghosh, Shyamali, Decorte, Bart L, Liu, Li, Tuman, Robert W A, Zhou, Zhao, Huebert, Norman, Bursell, Sven E, Clermont, Alan C, Grant, Maria B, Shaw, Lynn C, Mousa, Shaker A, Galemmo, Jr, Robert A, Johnson, Dana L, Maryanoff, Bruce E, Damiano, Bruce P
Published in The Journal of pharmacology and experimental therapeutics (01.03.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2008)
Get full text
Journal Article
Practical Approaches to Remote Asymmetric Induction in Steroidal Side-Chains Utilizing Oxazaborolidine Reagents
Rao, Meenakshi N, McGuigan, Melissa A, Zhang, Xuehai, Shaked, Ze'ev, Kinney, William A, Bulliard, Michel, Laboue, Blandine, Lee, Nancy E
Published in Journal of organic chemistry (27.06.1997)
Published in Journal of organic chemistry (27.06.1997)
Get full text
Journal Article
Suzuki−Miyaura Approach to JNJ-26076713, an Orally Active Tetrahydroquinoline-Containing αVβ3/αVβ5 Integrin Antagonist. Enantioselective Synthesis and Stereochemical Studies
Kinney, William A, Teleha, Christopher A, Thompson, Andrew S, Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C, McComsey, David F, Santulli, Rosemary J, Maryanoff, Bruce E
Published in Journal of organic chemistry (21.03.2008)
Published in Journal of organic chemistry (21.03.2008)
Get full text
Journal Article
Structure-Function Analysis of Urotensin II and Its Use in the Construction of a Ligand-Receptor Working Model
Kinney, William A., Almond, Jr, Harold R., Qi, Jenson, Smith, Charles E., Santulli, Rosemary J., de Garavilla, Lawrence, Andrade-Gordon, Patricia, Cho, Daniel S., Everson, Anita M., Feinstein, Mark A., Leung, Perry A., Maryanoff, Bruce E.
Published in Angewandte Chemie (International ed.) (16.08.2002)
Published in Angewandte Chemie (International ed.) (16.08.2002)
Get full text
Journal Article
Knockdown siRNA targeting GPR55 reveals significant differences between the anti-inflammatory actions of KLS-13019 and cannabidiol
Brenneman, Douglas E, Kinney, William A, McDonnell, Mark E, Ippolito, Michael J, Ward, Sara Jane
Published in Research square (28.02.2024)
Published in Research square (28.02.2024)
Get more information
Journal Article
Aminosterols from the Dogfish Shark Squalus acanthias
Rao, Meenakshi N, Shinnar, Ann E, Noecker, Lincoln A, Chao, Tessa L, Feibush, Binyamin, Snyder, Brad, Sharkansky, Ilya, Sarkahian, Ani, Zhang, Xuehai, Jones, Stephen R, Kinney, William A, Zasloff, Michael
Published in Journal of natural products (Washington, D.C.) (01.05.2000)
Published in Journal of natural products (Washington, D.C.) (01.05.2000)
Get full text
Journal Article
Phenylpiperidine-benzoxazinones as urotensin-II receptor antagonists: Synthesis, SAR, and in vivo assessment
Luci, Diane K., Ghosh, Shyamali, Smith, Charles E., Qi, Jenson, Wang, Yuanping, Haertlein, Barbara, Parry, Tom J., Li, Jian, Almond, Harold R., Minor, Lisa K., Damiano, Bruce P., Kinney, William A., Maryanoff, Bruce E., Lawson, Edward C.
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
Get full text
Journal Article
The synthesis of spermine analogs of the shark aminosterol squalamine
Shu, Youheng, Jones, Stephen R, Kinney, William A, Selinsky, Barry S
Published in Steroids (01.03.2002)
Published in Steroids (01.03.2002)
Get full text
Journal Article