The Screening Compound Collection: A Key Asset for Drug Discovery
Boss, Christoph, Hazemann, Julien, Kimmerlin, Thierry, von Korff, Modest, Lüthi, Urs, Peter, Oliver, Sander, Thomas, Siegrist, Romain
Published in Chimia (25.10.2017)
Published in Chimia (25.10.2017)
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Journal Article
Discovery and Optimization of Isoquinoline Ethyl Ureas as Antibacterial Agents
Panchaud, Philippe, Bruyère, Thierry, Blumstein, Anne-Catherine, Bur, Daniel, Chambovey, Alain, Ertel, Eric A, Gude, Markus, Hubschwerlen, Christian, Jacob, Loïc, Kimmerlin, Thierry, Pfeifer, Thomas, Prade, Lars, Seiler, Peter, Ritz, Daniel, Rueedi, Georg
Published in Journal of medicinal chemistry (11.05.2017)
Published in Journal of medicinal chemistry (11.05.2017)
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Journal Article
Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for de novo drug design and computational chemistry approaches
Hazemann, Julien, Kimmerlin, Thierry, Lange, Roland, Sweeney, Aengus Mac, Bourquin, Geoffroy, Ritz, Daniel, Czodrowski, Paul
Published in MedChemComm (19.06.2024)
Published in MedChemComm (19.06.2024)
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Journal Article
Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for drug design and computational chemistry approaches
Hazemann, Julien, Kimmerlin, Thierry, Lange, Roland, Sweeney, Aengus Mac, Bourquin, Geoffroy, Ritz, Daniel, Czodrowski, Paul
Published in RSC medicinal chemistry (19.06.2024)
Published in RSC medicinal chemistry (19.06.2024)
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Journal Article
CFTR 조절제로서의 마크로사이클
BOLLI MARTIN, SPRINGER JASPER, GATFIELD JOHN, COMMANDEUR MALGORZATA, WILLIAMS JODI T, KIMMERLIN THIERRY, WAGNER CLEMENS, WEGERT ANITA, BROTSCHI CHRISTINE, SIENDT HERVE
Year of Publication 19.12.2023
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Year of Publication 19.12.2023
Patent
How we drifted into peptide chemistry and where we have arrived at
Seebach, Dieter, Kimmerlin, Thierry, Šebesta, Radovan, Campo, Marino A., Beck, Albert K.
Published in Tetrahedron (23.08.2004)
Published in Tetrahedron (23.08.2004)
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Journal Article
Covalent Fluorescence Labeling of His-Tagged Proteins on the Surface of Living Cells
Hintersteiner, Martin, Weidemann, Thomas, Kimmerlin, Thierry, Filiz, Nimet, Buehler, Christof, Auer, Manfred
Published in Chembiochem : a European journal of chemical biology (16.06.2008)
Published in Chembiochem : a European journal of chemical biology (16.06.2008)
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Journal Article
INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
RENNEBERG DORTE, HUBLER FRANCIS, KIMMERLIN THIERRY, STAMM SIMON, HILPERT KURT
Year of Publication 17.08.2015
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Year of Publication 17.08.2015
Patent
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
RENNEBERG DORTE, HUBLER FRANCIS, KIMMERLIN THIERRY, STAMM SIMON, HILPERT KURT
Year of Publication 23.09.2014
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Year of Publication 23.09.2014
Patent
Investigation of the Interactions of β-Peptides with DNA Duplexes by Circular Dichroism Spectroscopy
Namoto, Kenji, Gardiner, James, Kimmerlin, Thierry, Seebach, Dieter
Published in Helvetica chimica acta (01.12.2006)
Published in Helvetica chimica acta (01.12.2006)
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Journal Article
CXCR7 RECEPTOR MODULATORS
FRETZ HEINZ, VALDENAIRE ANJA, POTHIER JULIEN, GUERRY PHILIPPE, LEHEMBRE FRANCOIS, KIMMERLIN THIERRY, SIENDT HERVE
Year of Publication 03.02.2016
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Year of Publication 03.02.2016
Patent
NOVEL ACRYLAMIDE DERIVATIVES AS ANTIMALARIAL AGENTS
CIANA CLAIRE LISE, AISSAOUI HAMED, SIEGRIST ROMAIN, KIMMERLIN THIERRY, BOSS CHRISTOPH
Year of Publication 25.11.2015
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Year of Publication 25.11.2015
Patent
1-[M-CARBOXAMIDO(HETERO)ARYL-METHYL]-HETEROCYCLYL-CARBOXAMIDE DERIVATIVES
GUDE MARKUS, FRETZ HEINZ, PFEIFER THOMAS, VALDENAIRE ANJA, GUERRY PHILIPPE, LEHEMBRE FRANCOIS, KIMMERLIN THIERRY
Year of Publication 05.03.2015
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Year of Publication 05.03.2015
Patent
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
RENNEBERG DORTE, MURPHY MARK, HUBLER FRANCIS, KIMMERLIN THIERRY, STAMM SIMON, HILPERT KURT
Year of Publication 07.05.2014
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Year of Publication 07.05.2014
Patent
Investigation of the Interactions of b-Peptides with DNA Duplexes by Circular Dichroism Spectroscopy
Namoto, Kenji, Gardiner, James, Kimmerlin, Thierry, Seebach, Dieter
Published in Helvetica chimica acta (01.12.2006)
Published in Helvetica chimica acta (01.12.2006)
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Journal Article