Atropisomeric 4‑Phenyl‑4H‑1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Synthesis and Evaluation of Novel Phenylethanolamine Derivatives containing Acetanilides as Potent and Selective β3-Adrenergic Receptor Agonists
Maruyama, Tatsuya, Onda, Kenichi, Hayakawa, Masahiko, Suzuki, Takayuki, Kimizuka, Tetsuya, Matsui, Tetsuo, Takasu, Toshiyuki, Nagase, Itsuro, Hamada, Noritaka, Ohta, Mitsuaki
Published in Chemical & Pharmaceutical Bulletin (01.04.2010)
Published in Chemical & Pharmaceutical Bulletin (01.04.2010)
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Synthesis and evaluation of novel phenylethanolamine derivatives containing acetanilides as potent and selective beta3-adrenergic receptor agonists
Maruyama, Tatsuya, Onda, Kenichi, Hayakawa, Masahiko, Suzuki, Takayuki, Kimizuka, Tetsuya, Matsui, Tetsuo, Takasu, Toshiyuki, Nagase, Itsuro, Hamada, Noritaka, Ohta, Mitsuaki
Published in Chemical & pharmaceutical bulletin (2010)
Published in Chemical & pharmaceutical bulletin (2010)
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An efficient preparative route to 7-ethyl-1H-furo[2,3-g]indazole
Shimada, Maeno, K, Kimizuka, T, Goto, S, Takahashi, T, Nakamura, A, Miyafuji, A, Tsukamoto, S, Sakamoto, S
Published in Heterocycles (01.01.2004)
Published in Heterocycles (01.01.2004)
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Atropisomeric 4-Phenyl-4 H -1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4 H -1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4H-1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Practical and efficient synthesis of the (R)-atropisomer of a 4-phenyl 1,2,4-triazole derivative as a selective GlyT1 inhibitor
Sugane, Takashi, Hamada, Noritaka, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Tetrahedron: asymmetry (15.12.2012)
Published in Tetrahedron: asymmetry (15.12.2012)
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Synthesis and biological evaluation of (4H-1,2,4-triazol-4-yl)isoquinoline derivatives as selective glycine transporter 1 inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Morita, Takuma, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (01.01.2012)
Published in Bioorganic & medicinal chemistry (01.01.2012)
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Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol-1-yl)ethylamine derivatives as 5-HT2C receptor agonists
Shimada, Itsuro, Maeno, Kyoichi, Kazuta, Ken-ichi, Kubota, Hideki, Kimizuka, Tetsuya, Kimura, Yasuharu, Hatanaka, Ken-ichi, Naitou, Yuki, Wanibuchi, Fumikazu, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Synthesis and Evaluation of Novel Phenylethanolamine Derivatives containing Acetanilides as Potent and Selective beta 3-Adrenergic Receptor Agonists
Maruyama, Tatsuya, Onda, Kenichi, Hayakawa, Masahiko, Suzuki, Takayuki, Kimizuka, Tetsuya, Matsui, Tetsuo, Takasu, Toshiyuki, Nagase, Itsuro, Hamada, Noritaka, Ohta, Mitsuaki
Published in Chemical & pharmaceutical bulletin (01.04.2010)
Published in Chemical & pharmaceutical bulletin (01.04.2010)
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Synthesis and Evaluation of Novel Phenylethanolamine Derivatives containing Acetanilides as Potent and Selective [beta]3-Adrenergic Receptor Agonists
Maruyama, Tatsuya, Onda, Kenichi, Hayakawa, Masahiko, Suzuki, Takayuki, Kimizuka, Tetsuya, Matsui, Tetsuo, Takasu, Toshiyuki, Nagase, Itsuro, Hamada, Noritaka, Ohta, Mitsuaki
Published in Chemical & pharmaceutical bulletin (01.04.2010)
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Published in Chemical & pharmaceutical bulletin (01.04.2010)
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Synthesis and structure-activity relationships of a series of substituted 2-(1H-furo[2,3-g]indazol -1 -yl)ethylamine derivatives as 5-HT2Creceptor agonists
SHIMADA, Itsuro, MAENO, Kyoichi, TSUKAMOTO, Shin-Ichi, KAZUTA, Ken-Ichi, KUBOTA, Hideki, KIMIZUKA, Tetsuya, KIMURA, Yasuharu, HATANAKA, Ken-Ichi, NAITOU, Yuki, WANIBUCHI, Fumikazu, SAKAMOTO, Shuichi
Published in Bioorganic & medicinal chemistry (2008)
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Published in Bioorganic & medicinal chemistry (2008)
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Synthesis and structure–activity relationships of a series of substituted 2-(1 H-furo[2,3- g]indazol-1-yl)ethylamine derivatives as 5-HT 2C receptor agonists
Shimada, Itsuro, Maeno, Kyoichi, Kazuta, Ken-ichi, Kubota, Hideki, Kimizuka, Tetsuya, Kimura, Yasuharu, Hatanaka, Ken-ichi, Naitou, Yuki, Wanibuchi, Fumikazu, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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SODIUM CHANNEL INHIBITOR
TOMIYAMA, HIROSHI, WATANABE, TOSHIHIRO, TOKUZAKI, KAZUO, SONEGAWA, MOTOHARU, HONDO, TAKESHI, KIMIZUKA, TETSUYA, IWAI, YOSHINORI, KIKUCHI, KAZUMI, NAGAKURA, YUKINORI, OKU, MAKOTO
Year of Publication 05.02.2004
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Year of Publication 05.02.2004
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2-ACYLAMINOTHIAZOLE DERIVATIVE OR ITS SALT
SUZUKI, KEN-ICHI, KOSHIO, HIROYUKI, SUGASAWA, KEIZO, KOGA, YUJI, WATANUKI, SUSUMU, NAGATA, HIROSHI, KIMIZUKA, TETSUYA, ABE, MASAKI
Year of Publication 15.08.2002
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Year of Publication 15.08.2002
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AMIDE DERIVATIVES OR SALTS THEREOF
MARUYAMA, TATSUYA, ONDA, KENICHI, HAYAKAWA, MASAHIKO, SUZUKI, TAKAYUKI, MORITOMO, HIROYUKI, KIMIZUKA, TETSUYA, MATSUI, TETSUO
Year of Publication 29.04.1999
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Year of Publication 29.04.1999
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TRICYCLIC PYRROLE OR PYRAZOLE DERIVATIVES
KAZUTA, KEN-ICHI, WANIBUCHI, FUMIKAZU, MAENO, KYOICHI, SHIMADA, ITSURO, KIMIZUKA, TETSUYA, SAKAMOTO, SHUICHI, KUBOTA, HIDEKI
Year of Publication 17.12.1998
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Year of Publication 17.12.1998
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TRIAZOLE DERIVATIVES
KOHARA, ATSUYUKI, MIYATA, JUNJI, TOBE, TAKAHIKO, ARLT, MICHAEL, HAMAGUCHI, WATARU, SHIMADA, ITSURO, MAENO, KYOICHI, KIMIZUKA, TETSUYA, MORITA, TAKUMA, GREINER, HARTMUT, SUGANE, TAKASHI, SUZUKI, TAKESHI
Year of Publication 22.11.2001
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Year of Publication 22.11.2001
Patent
ChemInform Abstract: Synthesis and Evaluation of Novel Phenylethanolamine Derivatives Containing Acetanilides as Potent and Selective β3-Adrenergic Receptor Agonists
Maruyama, Tatsuya, Onda, Kenichi, Hayakawa, Masahiko, Suzuki, Takayuki, Kimizuka, Tetsuya, Matsui, Tetsuo, Takasu, Toshiyuki, Nagase, Itsuro, Hamada, Noritaka, Ohta, Mitsuaki
Published in ChemInform (31.08.2010)
Published in ChemInform (31.08.2010)
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