In Vitro Bioactivation of Dihydrobenzoxathiin Selective Estrogen Receptor Modulators by Cytochrome P450 3A4 in Human Liver Microsomes: Formation of Reactive Iminium and Quinone Type Metabolites
Zhang, Zhoupeng, Chen, Qing, Li, Ying, Doss, George A, Dean, Brian J, Ngui, Jason S, Silva Elipe, Maria, Kim, Seongkon, Wu, Jane Y, DiNinno, Frank, Hammond, Milton L, Stearns, Ralph A, Evans, David C, Baillie, Thomas A, Tang, Wei
Published in Chemical research in toxicology (01.04.2005)
Published in Chemical research in toxicology (01.04.2005)
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Synthesis and properties of several isomers of the cardioactive steroid ouabain
Hong, Bor-Cherng, Kim, Seongkon, Kim, Tae-Seong, Corey, E.J.
Published in Tetrahedron letters (17.04.2006)
Published in Tetrahedron letters (17.04.2006)
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Estrogen receptor ligands. Part 3: The SAR of dihydrobenzoxathiin SERMs
Chen, Helen Y., Kim, Seongkon, Wu, Jane Y., Birzin, Elizabeth T., Chan, Wanda, Yang, Yi Tien, Dahllund, Johanna, DiNinno, Frank, Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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Discovery of MK-7655, a β-lactamase inhibitor for combination with Primaxin
Blizzard, Timothy A., Chen, Helen, Kim, Seongkon, Wu, Jane, Bodner, Rena, Gude, Candido, Imbriglio, Jason, Young, Katherine, Park, Young-Whan, Ogawa, Aimie, Raghoobar, Susan, Hairston, Nichelle, Painter, Ronald E., Wisniewski, Doug, Scapin, Giovanna, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hermes, Jeff, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
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Abstract 2653: Integrative analysis of proteomic alterations in human PBMC’s treated by HPK1 inhibitor FB849 reveals enriched pathways from various immune cells leading to potential novel biomarker discovery
Lim, Seungmook, Jin, Sooryeonhwa, Park, A Yeong, Kim, Hyekyoung, Kim, Seongkon, Kim, Jamie Jae Eun, Lee, Jinhwa
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract 2651: A selective HPK1 inhibitor FB849 reprograms intratumoral immune cells and elicits strong anti-cancer immunity
Kim, Hyekyoung, Lim, Seungmook, Park, A Yeong, Lee, Jinhwa, Kim, Jamie Jae Eun, Jeon, Seung Hyuck, Lee, Yong Joon, Shin, Eui-Cheol, Kim, Seongkon
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Fraud and financial crime detection model using malware forensics
Kim, Ae Chan, Kim, Seongkon, Park, Won Hyung, Lee, Dong Hoon
Published in Multimedia tools and applications (2014)
Published in Multimedia tools and applications (2014)
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Side chain SAR of bicyclic β-lactamase inhibitors (BLIs). 2. N-Alkylated and open chain analogs of MK-8712
Chen, Helen, Blizzard, Timothy A., Kim, Seongkon, Wu, Jane, Young, Katherine, Park, Young-Whan, Ogawa, Aimie M., Raghoobar, Susan, Painter, Ronald E., Wisniewski, Doug, Hairston, Nichelle, Fitzgerald, Paula, Sharma, Nandini, Scapin, Giovanna, Lu, Jun, Hermes, Jeff, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
Published in Bioorganic & medicinal chemistry letters (15.07.2011)
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Side chain SAR of bicyclic β-lactamase inhibitors (BLIs). 1. Discovery of a class C BLI for combination with imipinem
Blizzard, Timothy A., Chen, Helen, Kim, Seongkon, Wu, Jane, Young, Katherine, Park, Young-Whan, Ogawa, Amy, Raghoobar, Susan, Painter, Ronald E., Hairston, Nichelle, Lee, Sang Ho, Misura, Andrew, Felcetto, Tom, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hickey, Emily, Hermes, Jeff, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Discovery of MK-7655, a beta -lactamase inhibitor for combination with Primaxin registered
Blizzard, Timothy, Chen, Helen, Kim, Seongkon, Wu, Jane, Bodner, Rena, Gude, Candido, Imbriglio, Jason, Young, Katherine, Park, Young-Whan, Ogawa, Aimie, Raghoobar, Susan, Hairston, Nichelle, Painter, Ronald, Wisniewski, Doug, Scapin, Giovanna, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hermes, Jeff, Hammond, Milton
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
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Estrogen Receptor Ligands. II. Discovery of Benzoxathiins as Potent, Selective Estrogen Receptor α Modulators
Kim, Seongkon, Wu, Jane Y, Birzin, Elizabeth T, Frisch, Katalin, Chan, Wanda, Pai, Lee-Yuh, Yang, Yi Tien, Mosley, Ralph T, Fitzgerald, Paula M. D, Sharma, Nandini, Dahllund, Johanna, Thorsell, Ann-Gerd, DiNinno, Frank, Rohrer, Susan P, Schaeffer, James M, Hammond, Milton L
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers
Blizzard, Timothy A., DiNinno, Frank, Morgan, Jerry D., Chen, Helen Y., Wu, Jane Y., Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T., Yang, Yi Tien, Pai, Lee-Yuh, Fitzgerald, Paula M.D., Sharma, Nandini, Li, Ying, Zhang, Zhoupeng, Hayes, Edward C., DaSilva, Carolyn A., Tang, Wei, Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
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Side chain SAR of bicyclic [beta]-lactamase inhibitors (BLIs). 1. Discovery of a class C BLI for combination with imipinem
Blizzard, Timothy A., Chen, Helen, Kim, Seongkon, Wu, Jane, Young, Katherine, Park, Young-Whan, Ogawa, Amy, Raghoobar, Susan, Painter, Ronald E., Hairston, Nichelle, Lee, Sang Ho, Misura, Andrew, Felcetto, Tom, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hickey, Emily, Hermes, Jeff, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (17.09.2010)
Published in Bioorganic & medicinal chemistry letters (17.09.2010)
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