Agonist-like SERM effects on ERα-mediated repression of MMP1 promoter activity predict in vivo effects on bone and uterus
Scafonas, Angela, Reszka, Alfred A., Kimmel, Donald B., Hou, Xiaoli Shirley, Su, Qin, Birzin, Elizabeth T., Kim, Seongkon, Chen, Helen Y., Tan, Qiang, Roher, Susan P., Dininno, Frank, Hammond, Milton L., Rodan, Gideon A., Towler, Dwight A., Schmidt, Azriel
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
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Journal Article
Side chain SAR of bicyclic b-lactamase inhibitors (BLIs). 1. Discovery of a class C BLI for combination with imipinem
Blizzard, Timothy A, Chen, Helen, Kim, Seongkon, Wu, Jane, Young, Katherine, Park, Young-Whan, Ogawa, Amy, Raghoobar, Susan, Painter, Ronald E, Hairston, Nichelle, Lee, Sang Ho, Misura, Andrew, Felcetto, Tom, Fitzgerald, Paula, Sharma, Nandini, Lu, Jun, Ha, Sookhee, Hickey, Emily, Hermes, Jeff, Hammond, Milton L
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Estrogen Receptor Ligands. 12. Synthesis of the Major Metabolites of an ERα-Selective, Dihydrobenzoxathiin Antagonist for Osteoporosis
Kim, Seongkon, Wu, Jane Y., Zhang, Zhoupeng, Tang, Wei, Doss, George A., Dean, Brian J., DiNinno, Frank, Hammond, Milton L.
Published in Organic letters (03.02.2005)
Published in Organic letters (03.02.2005)
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Journal Article
Estrogen receptor ligands. Part 13: Dihydrobenzoxathiin SERAMs with an optimized antagonist side chain
Blizzard, Timothy A., DiNinno, Frank, Chen, Helen Y., Kim, Seongkon, Wu, Jane Y., Chan, Wanda, Birzin, Elizabeth T., Yang, Yi Tien, Pai, Lee-Yuh, Hayes, Edward C., DaSilva, Carolyn A., Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
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Journal Article
Agonist-like SERM effects on ERalpha-mediated repression of MMP1 promoter activity predict in vivo effects on bone and uterus
Scafonas, Angela, Reszka, Alfred A, Kimmel, Donald B, Hou, Xiaoli Shirley, Su, Qin, Birzin, Elizabeth T, Kim, Seongkon, Chen, Helen Y, Tan, Qiang, Roher, Susan P, Dininno, Frank, Hammond, Milton L, Rodan, Gideon A, Towler, Dwight A, Schmidt, Azriel
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
Published in The Journal of steroid biochemistry and molecular biology (01.06.2008)
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Journal Article
Estrogen receptor ligands. Part 7: Dihydrobenzoxathiin SERAMs with bicyclic amine side chains
Blizzard, Timothy A, DiNinno, Frank, Morgan, Jerry D, Chen, Helen Y, Wu, Jane Y, Gude, Candido, Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T, Tien Yang, Yi, Pai, Lee-Yuh, Zhang, Zhoupeng, Hayes, Edward C, DaSilva, Carolyn A, Tang, Wei, Rohrer, Susan P, Schaeffer, James M, Hammond, Milton L
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Journal Article
Estrogen receptor ligands. Part 4: The SAR of the syn-dihydrobenzoxathiin SERAMs
Kim, Seongkon, Wu, Jane, Chen, Helen Y., Birzin, Elizabeth T., Chan, Wanda, Yang, Yi Tien, Colwell, Lawrence, Li, Susan, Dahllund, Johanna, DiNinno, Frank, Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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Journal Article
Estrogen receptor ligands. 12. Synthesis of the major metabolites of an ERalpha-selective, dihydrobenzoxathiin antagonist for osteoporosis
Kim, Seongkon, Wu, Jane Y, Zhang, Zhoupeng, Tang, Wei, Doss, George A, Dean, Brian J, Dininno, Frank, Hammond, Milton L
Published in Organic letters (03.02.2005)
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Published in Organic letters (03.02.2005)
Journal Article
Antagonist-Induced, Activation Function-2-Independent Estrogen Receptor α Phosphorylation
Lipfert, Lorraine, Fisher, John E, Wei, Nan, Scafonas, Angela, Su, Qin, Yudkovitz, Joel, Chen, Fang, Warrier, Sudha, Birzin, Elizabeth T, Kim, Seongkon, Chen, Helen Y, Tan, Qiang, Schmidt, Azriel, Dininno, Frank, Rohrer, Susan P, Hammond, Milton L, Rodan, Gideon A, Freedman, Leonard P, Reszka, Alfred A
Published in Molecular endocrinology (Baltimore, Md.) (01.03.2006)
Published in Molecular endocrinology (Baltimore, Md.) (01.03.2006)
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Journal Article
Biomimetic Total Syntheses of (+)-Cephalostatin 7, (+)-Cephalostatin 12, and (+)-Ritterazine K
Jeong, Jae Uk, Sutton, Scott C, Kim, Seongkon, Fuchs, P. L
Published in Journal of the American Chemical Society (01.10.1995)
Published in Journal of the American Chemical Society (01.10.1995)
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Journal Article
Estrogen receptor ligands. Part 8: Dihydrobenzoxathiin SERAMs with heteroatom-substituted side chains
Blizzard, Timothy A, DiNinno, Frank, Morgan, Jerry D, Wu, Jane Y, Chen, Helen Y, Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T, Yang, Yi Tien, Pai, Lee-Yuh, Zhang, Zhoupeng, Hayes, Edward C, DaSilva, Carolyn A, Tang, Wei, Rohrer, Susan P, Schaeffer, James M, Hammond, Milton L
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Journal Article
Estrogen receptor ligands. Part 15: Synthesis of benzothiopyran-based selective estrogen receptor alpha modulators (SERAM)
Kim, S, DiNinno, F, Birzin, ET, Chan, W, Yang, YT, Hammond, ML
Published in Heterocycles (01.01.2006)
Published in Heterocycles (01.01.2006)
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Journal Article
Estrogen receptor ligands. II. Discovery of benzoxathiins as potent, selective estrogen receptor a modulators
KIM, Seongkon, WU, Jane Y, DAHLLUND, Johanna, THORSELL, Ann-Gerd, DININNO, Frank, ROHRER, Susan P, SCHAEFFER, James M, HAMMOND, Milton L, BIRZIN, Elizabeth T, FRISCH, Katalin, CHAN, Wanda, PAI, Lee-Yuh, YI TIEN YANG, MOSLEY, Ralph T, FITZGERALD, Paula M. D, SHARMA, Nandini
Published in Journal of medicinal chemistry (2004)
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Published in Journal of medicinal chemistry (2004)
Journal Article
Synthesis of the North 1 Unit of the Cephalostatin Family from Hecogenin Acetate 1
Kim, Seongkon, Sutton, Scott C., Guo, Chuangxing, LaCour, Thomas G., Fuchs, P. L.
Published in Journal of the American Chemical Society (01.03.1999)
Published in Journal of the American Chemical Society (01.03.1999)
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Journal Article
Synthesis of the North 1 Unit of the Cephalostatin Family from Hecogenin Acetate1
Kim, Seongkon, Sutton, Scott C, Guo, Chuangxing, LaCour, Thomas G, Fuchs, P. L
Published in Journal of the American Chemical Society (17.03.1999)
Published in Journal of the American Chemical Society (17.03.1999)
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Journal Article
BETA-LACTAMASE INHIBITORS
RIVERA, NELO, MORTKO, CHRISTOPHER, J, CHEN, HELEN, GUDE, CANDIDO, HERMES, JEFFREY, D, MANGION, IAN, SHEVLIN, MICHAEL, WU, JANE Y, IMBRIGLIO, JASON, E, RUCK, REBECCA, T, KIM, SEONGKON, HA, SOOKHEE, BLIZZARD, TIMOTHY, A
Year of Publication 15.06.2017
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Year of Publication 15.06.2017
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