Total Synthesis and Absolute Stereochemistry of Polygalolides A and B
Nakamura, Seiichi, Sugano, Yukihito, Kikuchi, Fumiaki, Hashimoto, Shunichi
Published in Angewandte Chemie (International ed.) (06.10.2006)
Published in Angewandte Chemie (International ed.) (06.10.2006)
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Journal Article
Total Syntheses of (+)-Polygalolide A and (+)-Polygalolide B: Elucidation of the Absolute Stereochemistry and Biogenetic Implications
Sugano, Yukihito, Kikuchi, Fumiaki, Toita, Akinori, Nakamura, Seiichi, Hashimoto, Shunichi
Published in Chemistry : a European journal (27.07.2012)
Published in Chemistry : a European journal (27.07.2012)
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Journal Article
Stereoselective synthesis of a C1–C6 fragment of pinnatoxin A via a 1,4-addition/alkylation sequence
Nakamura, Seiichi, Kikuchi, Fumiaki, Hashimoto, Shunichi
Published in Tetrahedron: asymmetry (16.05.2008)
Published in Tetrahedron: asymmetry (16.05.2008)
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Journal Article
Photoredox-based late-stage functionalization in SAR study for in vivo potent glucosylceramide synthase inhibitor
Wang, Junsi, Reynolds, Matthew, Ibáñez, Ignacio, Sasaki, Yusuke, Tanaka, Yuta, Kikuchi, Fumiaki, Ohashi, Tomohiro, Sato, Sho, Miyabayashi, Mariko, Fujii, Takahiro, Tanaka, Yuta
Published in Bioorganic & medicinal chemistry letters (01.12.2022)
Published in Bioorganic & medicinal chemistry letters (01.12.2022)
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Journal Article
Total Synthesis and Absolute Stereochemistry of Polygalolides A and B
Nakamura, Seiichi, Sugano, Yukihito, Kikuchi, Fumiaki, Hashimoto, Shunichi
Published in Angewandte Chemie (06.10.2006)
Published in Angewandte Chemie (06.10.2006)
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Journal Article
Design, Synthesis, and Biological Evaluation of a Novel Series of 4‑Guanidinobenzoate Derivatives as Enteropeptidase Inhibitors with Low Systemic Exposure for the Treatment of Obesity
Ikeda, Zenichi, Kakegawa, Keiko, Kikuchi, Fumiaki, Itono, Sachiko, Oki, Hideyuki, Yashiro, Hiroaki, Hiyoshi, Hideyuki, Tsuchimori, Kazue, Hamagami, Kenichi, Watanabe, Masanori, Sasaki, Masako, Ishihara, Youko, Tohyama, Kimio, Kitazaki, Tomoyuki, Maekawa, Tsuyoshi, Sasaki, Minoru
Published in Journal of medicinal chemistry (23.06.2022)
Published in Journal of medicinal chemistry (23.06.2022)
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Journal Article
Discovery of Brain-Penetrant Glucosylceramide Synthase Inhibitors with a Novel Pharmacophore
Tanaka, Yuta, Seto, Masaki, Kakegawa, Keiko, Takami, Kazuaki, Kikuchi, Fumiaki, Yamamoto, Takeshi, Nakamura, Minoru, Daini, Masaki, Murakami, Masataka, Ohashi, Tomohiro, Kasahara, Takahito, Wang, Junsi, Ikeda, Zenichi, Wada, Yasufumi, Puenner, Florian, Fujii, Takahiro, Inazuka, Masakazu, Sato, Sho, Suzaki, Tomohiko, Oak, Jeong-Ho, Takai, Yuichi, Kohara, Hiroshi, Kimoto, Kouya, Oki, Hideyuki, Mikami, Satoshi, Sasaki, Minoru, Tanaka, Yuta
Published in Journal of medicinal chemistry (10.03.2022)
Published in Journal of medicinal chemistry (10.03.2022)
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Journal Article
Discovery of a novel series of medium-sized cyclic enteropeptidase inhibitors
Kikuchi, Fumiaki, Ikeda, Zenichi, Kakegawa, Keiko, Nishikawa, Youichi, Sasaki, Shigekazu, Fukuda, Koichiro, Takami, Kazuaki, Banno, Yoshihiro, Nishikawa, Hitoaki, Taya, Naohiro, Nakahata, Takashi, Itono, Sachiko, Yashiro, Hiroaki, Tsuchimori, Kazue, Hiyoshi, Hideyuki, Sasaki, Masako, Tohyama, Kimio, Matsumiya, Kouta, Ishihara, Youko, Kawamoto, Tetsuji, Kamaura, Masahiro, Watanabe, Masanori, Kitazaki, Tomoyuki, Maekawa, Tsuyoshi, Sasaki, Minoru
Published in Bioorganic & medicinal chemistry (01.10.2023)
Published in Bioorganic & medicinal chemistry (01.10.2023)
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Journal Article
Total Synthesis of Pinnatoxin A
Nakamura, Seiichi, Kikuchi, Fumiaki, Hashimoto, Shunichi
Published in Angewandte Chemie (International ed.) (01.09.2008)
Published in Angewandte Chemie (International ed.) (01.09.2008)
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Journal Article
Total Syntheses of (+)-PolygalolideA and (+)-PolygalolideB: Elucidation of the Absolute Stereochemistry and Biogenetic Implications
Sugano, Yukihito, Kikuchi, Fumiaki, Toita, Akinori, Nakamura, Seiichi, Hashimoto, Shunichi
Published in Chemistry : a European journal (27.07.2012)
Published in Chemistry : a European journal (27.07.2012)
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Journal Article
FUSED HETEROCYCLIC COMPOUND
IKEDA ZENICHI, SASAKI MINORU, NISHIKAWA YOICHI, KIKUCHI FUMIAKI, KAKEGAWA KEIKO
Year of Publication 06.10.2016
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Year of Publication 06.10.2016
Patent
FUSED HETEROCYCLIC COMPOUND
IKEDA, Zenichi, KIKUCHI, Fumiaki, SASAKI, Minoru, NISHIKAWA, Yoichi, KAKEGAWA, Keiko
Year of Publication 06.10.2016
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Year of Publication 06.10.2016
Patent
HETEROCYCLIC COMPOUND
IKEDA ZENICHI, SASAKI MINORU, NISHIKAWA YOICHI, KIKUCHI FUMIAKI, KAKEGAWA KEIKO
Year of Publication 28.09.2016
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Year of Publication 28.09.2016
Patent
NUCLEIC ACID COMPLEX
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Year of Publication 25.03.2021
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Year of Publication 25.03.2021
Patent
HETEROCYCLIC COMPOUND
IKEDA, Zenichi, TAKAMI, Kazuaki, PUENNER, Florian, SASAKI, Minoru, YAMAMOTO, Takeshi, NAKAMURA, Minoru, DAINI, Masaki, KIKUCHI, Fumiaki, SETO, Masaki, MURAKAMI, Masataka, MIKAMI, Satoshi, KASAHARA, Takahito, KAKEGAWA, Keiko, OHASHI, Tomohiro, TANAKA, Yuta
Year of Publication 04.02.2021
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Year of Publication 04.02.2021
Patent
HETEROCYCLIC COMPOUND
IKEDA, Zenichi, TAKAMI, Kazuaki, PUENNER, Florian, SASAKI, Minoru, YAMAMOTO, Takeshi, NAKAMURA, Minoru, DAINI, Masaki, KIKUCHI, Fumiaki, WADA, Yasufumi, SETO, Masaki, MURAKAMI, Masataka, MIKAMI, Satoshi, KASAHARA, Takahito, WANG, Junsi, KAKEGAWA, Keiko, OHASHI, Tomohiro, TANAKA, Yuta
Year of Publication 04.02.2021
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Year of Publication 04.02.2021
Patent
HETEROCYCLIC COMPOUND AND USE THEREOF
KUBO, Osamu, TAKASHIMA, Sachie, PUENNER, Florian, YAMAGUCHI, Fumie, NAKAMURA, Minoru, DAINI, Masaki, KAMATA, Makoto, KIKUCHI, Fumiaki, MIKAMI, Satoshi, MURAKAMI, Masataka, OGURO, Yuya, KASAHARA, Takahito, TOITA, Akinori, YUKAWA, Takafumi, MORIMOTO, Shinji, IKEDA, Shuhei
Year of Publication 30.07.2020
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Year of Publication 30.07.2020
Patent