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Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors

by Boby, Melissa L, Ferla, Matteo, Filep, Mihajlo, Koekemoer, Lizbé, Lee, Alpha A, London, Nir, Alonzi, Dominic S, Balcomb, Blake H, Bar-David, Elad, Ben-Shmuel, Amir, Bilenko, Vitaliy A, Boulet, Pascale, Calmiano, Mark, Carney, Daniel W, Chang, Edcon, Coffland, Joseph E, Cohen, Galit, Cole, Jason C, Cox, Lisa, De Jonghe, Steven, Donckers, Kim, Duberstein, Shirly, Dudgeon, Tim, Dunnett, Louise E, Eastman, Peter, Fate, Gwen, Ferrins, Lori, Foster, Richard, Foster, Holly, Fraisse, Laurent, Gabizon, Ronen, Gawriljuk, Victor O, Giroud, Charline, Godoy, Andre S, Gorichko, Marian, Griffen, Ed J, Henry, Michael, Huang, Qiu Yu Judy, Hurley, Matthew F D, Israely, Tomer, John, Tobias, Kenny, Peter W, Kovar, Boris, Laghnimi-Hahn, Sophie, Logvinenko, Ivan G, Macdonald, Hannah Bruce, Marples, Peter G, McCorkindale, Willam, Melamed, Sharon, Mikolajek, Halina, Minh, David, Moustakas, Demetri, Mowbray, Charles E, Neyts, Johan, Nguyen, Luong, Oliva, Glaucius, Pai, Ruby, Pan, Jin, Paran, Nir, Perry, Benjamin, Pingle, Maneesh, Politi, Boaz, Puni, Reut, Rangel, Victor L, Rees, Paul, Reid, Lauren, Rodriguez-Guerra, Jaime, Rosales, Romel, Rufa, Dominic A, Salah, Eidarus, Scheen, Jenke, Schiffer, Celia A, Schofield, Christopher J, Shi, Jiye, Shurrush, Khriesto, Singh, Sukrit, Sjö, Peter, Skyner, Rachael, Smalley, Adam, Smeets, Bart, Spencer, John, Strain-Damerell, Claire, Tamir, Hadas, Thompson, Warren, Thompson, Andrew, Tomlinson, Charles W E, Tsurupa, Igor S, van Rij, Ronald P, Vangeel, Laura, Vaschetto, Mariana, Voelz, Vincent, Volkamer, Andrea, Wild, Conor Francis, Wittmann, Matthew, Yahalom-Ronen, Yfat, Zaidmann, Daniel, Zhang, Ivy, Zidane, Hadeer, Zitzmann, Nicole, Zvornicanin, Sarah N
Published in Science (American Association for the Advancement of Science) (10.11.2023)

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Journal Article

Open Science Discovery of Potent Non-Covalent SARS-CoV-2 Main Protease Inhibitors

by Aimon, Anthony, Bar-David, Elad, Barr, Haim, Bilenko, Vitaliy A, Bowman, Gregory R, Brwewitz, Lennart, Sarma Bvnbs, Carbery, Anna, Carney, Daniel, Cattermole, Emma, Chang, Edcon, Cohen, Galit, Cole, Jason, Croll, Tristan Ian, Cvitkovic, Milan, Dias, Alex, Donckers, Kim, Dotson, David L, Duberstein, Shirly, Dunnett, Louise, Fairhead, Mike, Ferla, Matteo, Fernandes, Rafaela S, Ferrins, Lori, Foster, Richard, Fraisse, Laurent, Giroud, Charline, Glass, William G, Glen, Robert, Godoy, Andre S, Gorichko, Marian, Gorrie-Stone, Tyler, Hahn, Sophie, Heer, Jag, Henry, Michael, Israely, Tomer, Jajack, Andrew, Jochmans, Dirk, Tobias, John, Kang, Lulu, Kantsadi, Anastassia L, Kenny, Peter W, Kiappes, J L, La, Van, Lefker, Bruce A, London, Nir, Lukacik, Petra, Macdonald, Hannah Bruce, Maclean, Elizabeth M, Mccorkindale, Willam, Melamed, Sharon, Melnykov, Kostiantyn P, Miesen, Pascal, Mikolajek, Halina, Minh, David, Jose Brandao Neto, Neyts, Johan, Oliva, Glaucius, Pai, Ruby, Pan, Jin, Paran, Nir, Perry, Benjamin, Pingle, Maneesh, Powell, Ailsa, Pulido, Ivan, Rangel, Victor L, Reddi, Rambabu N, Reid, St Patrick, Rodriguez-Guerra, Jaime, Rosales, Romel, Rufa, Dominic A, Saar, Kadi, Kumar Singh Saikatendu, Eidarus Salah, Shafeev, Mikhail, Shaqra, Ala M, Sittner, Assa, Sjo, Peter, Skyner, Rachael, Smalley, Adam, Solmesky, Leonardo J, Spencer, John, Swamy, Vishwanath, Thompson, Warren, Thompson, Andrew, Tomlinson, Charlie, Tsurupa, Igor S, Tumber, Anthony, Vaschetto, Mariana, Vitner, Einat B, Voelz, Vincent, Frank Von Delft, Walsh, Martin, Weatherall, Charlie, Wild, Conor Francis, Witt, Karolina D, Wright, Nathan, Zaidmann, Daniel, Zitzmann, Nicole, Zvornicanin, Sarah N
Published in bioRxiv (02.03.2023)

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