The first universal opioid ligand, (2S)-2-[(5R,6R,7R,14S)-N-cyclopropylmethyl-4,5-epoxy-6,14-ethano-3-hydroxy-6-methoxymorphinan-7-yl]-3,3-dimethylpentan-2-ol (BU08028): characterization of the in vitro profile and in vivo behavioral effects in mouse models of acute pain and cocaine-induced reward
Khroyan, Taline V, Polgar, Willma E, Cami-Kobeci, Gerta, Husbands, Stephen M, Zaveri, Nurulain T, Toll, Lawrence
Published in The Journal of pharmacology and experimental therapeutics (01.03.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2011)
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Genetics of nicotine dependence and pharmacotherapy
Lessov-Schlaggar, Christina N., Pergadia, Michele L., Khroyan, Taline V., Swan, Gary E.
Published in Biochemical pharmacology (01.01.2008)
Published in Biochemical pharmacology (01.01.2008)
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Hypocretin/orexin and nociceptin/orphanin FQ coordinately regulate analgesia in a mouse model of stress-induced analgesia
Xie, Xinmin, Wisor, Jonathan P, Hara, Junko, Crowder, Tara L, LeWinter, Robin, Khroyan, Taline V, Yamanaka, Akihiro, Diano, Sabrina, Horvath, Tamas L, Sakurai, Takeshi, Toll, Lawrence, Kilduff, Thomas S
Published in The Journal of clinical investigation (01.07.2008)
Published in The Journal of clinical investigation (01.07.2008)
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Journal Article
Synthesis, Biological Evaluation, and SAR Studies of 14β-phenylacetyl Substituted 17-cyclopropylmethyl-7, 8-dihydronoroxymorphinones Derivatives: Ligands With Mixed NOP and Opioid Receptor Profile
Kumar, Vinod, Polgar, Willma E, Cami-Kobeci, Gerta, Thomas, Mark P, Khroyan, Taline V, Toll, Lawrence, Husbands, Stephen M
Published in Frontiers in psychiatry (19.09.2018)
Published in Frontiers in psychiatry (19.09.2018)
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Journal Article
Cyclooxygenase inhibition targets neurons to prevent early behavioural decline in Alzheimer's disease model mice
Woodling, Nathaniel S, Colas, Damien, Wang, Qian, Minhas, Paras, Panchal, Maharshi, Liang, Xibin, Mhatre, Siddhita D, Brown, Holden, Ko, Novie, Zagol-Ikapitte, Irene, van der Hart, Marieke, Khroyan, Taline V, Chuluun, Bayarsaikhan, Priyam, Prachi G, Milne, Ginger L, Rassoulpour, Arash, Boutaud, Olivier, Manning-Boğ, Amy B, Heller, H Craig, Andreasson, Katrin I
Published in Brain (London, England : 1878) (01.07.2016)
Published in Brain (London, England : 1878) (01.07.2016)
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Peptides derived from the prohormone proNPQ/spexin are potent central modulators of cardiovascular and renal function and nociception
Toll, Lawrence, Khroyan, Taline V, Sonmez, Kemal, Ozawa, Akihiko, Lindberg, Iris, McLaughlin, Jay P, Eans, Shainnel O, Shahien, Amir A, Kapusta, Daniel R
Published in The FASEB journal (01.02.2012)
Published in The FASEB journal (01.02.2012)
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High affinity α3β4 nicotinic acetylcholine receptor ligands AT-1001 and AT-1012 attenuate cocaine-induced conditioned place preference and behavioral sensitization in mice
Khroyan, Taline V., Yasuda, Dennis, Toll, Lawrence, Polgar, Willma E., Zaveri, Nurulain T.
Published in Biochemical pharmacology (15.10.2015)
Published in Biochemical pharmacology (15.10.2015)
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Journal Article
Differential effects of nociceptin/orphanin FQ (NOP) receptor agonists in acute versus chronic pain: studies with bifunctional NOP/μ receptor agonists in the sciatic nerve ligation chronic pain model in mice
Khroyan, Taline V, Polgar, Willma E, Orduna, Juan, Montenegro, Jose, Jiang, Faming, Zaveri, Nurulain T, Toll, Lawrence
Published in The Journal of pharmacology and experimental therapeutics (01.11.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2011)
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Journal Article
Nociceptin/orphanin FQ receptor activation attenuates antinociception induced by mixed nociceptin/orphanin FQ/mu-opioid receptor agonists
Khroyan, Taline V, Polgar, Willma E, Jiang, Faming, Zaveri, Nurulain T, Toll, Lawrence
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
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Journal Article
AT-1001: A High Affinity and Selective alpha 3 beta 4 Nicotinic Acetylcholine Receptor Antagonist Blocks Nicotine Self-Administration in Rats
Toll, Lawrence, Zaveri, Nurulain T, Polgar, Willma E, Jiang, Faming, Khroyan, Taline V, Zhou, Wei, Xie, Xinmin, Stauber, Gregory B, Costello, Matthew R, Leslie, Frances M
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2012)
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2012)
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Journal Article
AT- 1001: A High Affinity and Selective α3β4 Nicotinic Acetylcholine Receptor Antagonist Blocks Nicotine Self-Administration in Rats
TOLL, Lawrence, ZAVERI, Nurulain T, POLGAR, Willma E, FAMING JIANG, KHROYAN, Taline V, WEI ZHOU, XIE, Xinmin (simon), STAUBER, Gregory B, COSTELLO, Matthew R, LESLIE, Frances M
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2012)
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2012)
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Journal Article
Anti-nociceptive and anti-allodynic effects of a high affinity NOP hexapeptide [Ac-RY(3-Cl)YRWR-NH 2] (Syn 1020) in rodents
Khroyan, Taline V., Polgar, Willma E., Orduna, Juan, Zaveri, Naunihal T., Judd, Amrit K., Tuttle, David J., Sanchez, Agustin, Toll, Lawrence
Published in European journal of pharmacology (29.03.2007)
Published in European journal of pharmacology (29.03.2007)
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Journal Article
AT‐1001: a high‐affinity α3β4 nAChR ligand with novel nicotine‐suppressive pharmacology
Cippitelli, Andrea, Wu, Jinhua, Gaiolini, Kelly A, Mercatelli, Daniela, Schoch, Jennifer, Gorman, Michelle, Ramirez, Alejandra, Ciccocioppo, Roberto, Khroyan, Taline V, Yasuda, Dennis, Zaveri, Nurulain T, Pascual, Conrado, Xie, Xinmin (Simon), Toll, Lawrence
Published in British journal of pharmacology (01.04.2015)
Published in British journal of pharmacology (01.04.2015)
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Journal Article
Rodent models of nicotine reward: What do they tell us about tobacco abuse in humans?
O'Dell, Laura E., Khroyan, Taline V.
Published in Pharmacology, biochemistry and behavior (01.02.2009)
Published in Pharmacology, biochemistry and behavior (01.02.2009)
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Journal Article
AT-1001: a high-affinity alpha 3 beta 4 nAChR ligand with novel nicotine-suppressive pharmacology
Cippitelli, Andrea, Wu, Jinhua, Gaiolini, Kelly A, Mercatelli, Daniela, Schoch, Jennifer, Gorman, Michelle, Ramirez, Alejandra, Ciccocioppo, Roberto, Khroyan, Taline V, Yasuda, Dennis, Zaveri, Nurulain T, Pascual, Conrado, Xie, Xinmin, Toll, Lawrence
Published in British journal of pharmacology (01.04.2015)
Published in British journal of pharmacology (01.04.2015)
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Journal Article
Comparison of the antinociceptive and antirewarding profiles of novel bifunctional nociceptin receptor/mu-opioid receptor ligands: implications for therapeutic applications
Toll, Lawrence, Khroyan, Taline V, Polgar, Willma E, Jiang, Faming, Olsen, Cris, Zaveri, Nurulain T
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2009)
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Journal Article
In Vitro and In Vivo Profile of PPL-101 and PPL-103: Mixed Opioid Partial Agonist Analgesics with Low Abuse Potential
Khroyan, Taline V, Cippitelli, Andrea, Toll, Nicholas, Lawson, John A, Crossman, William, Polgar, Willma E, Toll, Lawrence
Published in Frontiers in psychiatry (12.04.2017)
Published in Frontiers in psychiatry (12.04.2017)
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Journal Article
Retrodialysis of N/OFQ into the nucleus accumbens shell blocks cocaine-induced increases in extracellular dopamine and locomotor activity
Vazquez-DeRose, Jacqueline, Stauber, Gregory, Khroyan, Taline V., Xie, Xinmin Simon, Zaveri, Nurulain T., Toll, Lawrence
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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