Effects of Charge on Antibody Tissue Distribution and Pharmacokinetics
Boswell, C. Andrew, Tesar, Devin B., Mukhyala, Kiran, Theil, Frank-Peter, Fielder, Paul J., Khawli, Leslie A.
Published in Bioconjugate chemistry (15.12.2010)
Published in Bioconjugate chemistry (15.12.2010)
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Conjugation site modulates the in vivo stability and therapeutic activity of antibody-drug conjugates
Shen, Ben-Quan, Xu, Keyang, Liu, Luna, Raab, Helga, Bhakta, Sunil, Kenrick, Margaret, Parsons-Reponte, Kathryn L, Tien, Janet, Yu, Shang-Fan, Mai, Elaine, Li, Dongwei, Tibbitts, Jay, Baudys, Jakub, Saad, Ola M, Scales, Suzie J, McDonald, Paul J, Hass, Philip E, Eigenbrot, Charles, Nguyen, Trung, Solis, Willy A, Fuji, Reina N, Flagella, Kelly M, Patel, Darshana, Spencer, Susan D, Khawli, Leslie A, Ebens, Allen, Wong, Wai Lee, Vandlen, Richard, Kaur, Surinder, Sliwkowski, Mark X, Scheller, Richard H, Polakis, Paul, Junutula, Jagath R
Published in Nature biotechnology (01.02.2012)
Published in Nature biotechnology (01.02.2012)
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A Humanized Lym-1 CAR with Novel DAP10/DAP12 Signaling Domains Demonstrates Reduced Tonic Signaling and Increased Antitumor Activity in B-Cell Lymphoma Models
Zheng, Long, Ren, Luqing, Kouhi, Aida, Khawli, Leslie A, Hu, Peisheng, Kaslow, Harvey R, Epstein, Alan L
Published in Clinical cancer research (15.07.2020)
Published in Clinical cancer research (15.07.2020)
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Enhancing brain entry and therapeutic activity of chimeric antigen receptor T cells with intra-arterial NEO100 in a mouse model of CNS lymphoma
Wang, Weijun, He, Haiping, Zheng, Long, Zeng, Shan, Cho, Hee-Yeon, Kouhi, Aida, Khawli, Leslie A, Chen, Ligang, Stathopoulos, Apostolos, Schönthal, Axel H, Epstein, Alan L, Chen, Thomas C
Published in Journal of neurosurgery (01.06.2024)
Published in Journal of neurosurgery (01.06.2024)
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Physiochemical and Biochemical Factors Influencing the Pharmacokinetics of Antibody Therapeutics
Bumbaca, Daniela, Boswell, C. Andrew, Fielder, Paul J., Khawli, Leslie A.
Published in The AAPS journal (01.09.2012)
Published in The AAPS journal (01.09.2012)
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Charge variants in IgG1: Isolation, characterization, in vitro binding properties and pharmacokinetics in rats
Khawli, Leslie A., Goswami, Sirj, Hutchinson, Ryan, Kwong, Zephania W., Yang, Jihong, Wang, Xiangdan, Yao, Zhenling, Sreedhara, Alavattam, Cano, Tony, Tesar, Devin B., Nijem, Ihsan, Allison, David E., Wong, Pin Yee, Kao, Yung-Hsiang, Quan, Cynthia, Joshi, Amita, Harris, Reed J., Motchnik, Paul
Published in mAbs (01.11.2010)
Published in mAbs (01.11.2010)
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Evaluating the Use of Antibody Variable Region (Fv) Charge as a Risk Assessment Tool for Predicting Typical Cynomolgus Monkey Pharmacokinetics
Bumbaca Yadav, Daniela, Sharma, Vikas K., Boswell, Charles Andrew, Hotzel, Isidro, Tesar, Devin, Shang, Yonglei, Ying, Yong, Fischer, Saloumeh K., Grogan, Jane L., Chiang, Eugene Y., Urban, Konnie, Ulufatu, Sheila, Khawli, Leslie A., Prabhu, Saileta, Joseph, Sean, Kelley, Robert F.
Published in The Journal of biological chemistry (11.12.2015)
Published in The Journal of biological chemistry (11.12.2015)
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Impact of Drug Conjugation on Pharmacokinetics and Tissue Distribution of Anti-STEAP1 Antibody–Drug Conjugates in Rats
Boswell, C. Andrew, Mundo, Eduardo E, Zhang, Crystal, Bumbaca, Daniela, Valle, Nicole R, Kozak, Katherine R, Fourie, Aimee, Chuh, Josefa, Koppada, Neelima, Saad, Ola, Gill, Herman, Shen, Ben-Quan, Rubinfeld, Bonnee, Tibbitts, Jay, Kaur, Surinder, Theil, Frank-Peter, Fielder, Paul J, Khawli, Leslie A, Lin, Kedan
Published in Bioconjugate chemistry (19.10.2011)
Published in Bioconjugate chemistry (19.10.2011)
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A novel in vitro method to model the fate of subcutaneously administered biopharmaceuticals and associated formulation components
Kinnunen, Hanne M., Sharma, Vikas, Contreras-Rojas, Luis Rodrigo, Yu, Yafei, Alleman, Chlöe, Sreedhara, Alavattam, Fischer, Stefan, Khawli, Leslie, Yohe, Stefan T., Bumbaca, Daniela, Patapoff, Thomas W., Daugherty, Ann L., Mrsny, Randall J.
Published in Journal of controlled release (28.09.2015)
Published in Journal of controlled release (28.09.2015)
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Spatio-temporal biodistribution of 89Zr-oxine labeled huLym-1-A-BB3z-CAR T-cells by PET imaging in a preclinical tumor model
Sta Maria, Naomi S., Khawli, Leslie A., Pachipulusu, Vyshnavi, Lin, Sharon W., Zheng, Long, Cohrs, Daniel, Liu, Xiaodan, Hu, Peisheng, Epstein, Alan L., Jacobs, Russell E.
Published in Scientific reports (23.07.2021)
Published in Scientific reports (23.07.2021)
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Unraveling the Effect of Immunogenicity on the PK/PD, Efficacy, and Safety of Therapeutic Proteins
Theil, Frank-Peter, Epstein, Alan L., Frutoz, Kimberley, Jaw, Stacey, Manoli, Hugh, Smith, Alison, Khawli, Leslie A.
Published in Journal of Immunology Research (01.01.2016)
Published in Journal of Immunology Research (01.01.2016)
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Lym-1 Chimeric Antigen Receptor T Cells Exhibit Potent Anti-Tumor Effects against B-Cell Lymphoma
Zheng, Long, Hu, Peisheng, Wolfe, Brandon, Gonsalves, Caryn, Ren, Luqing, Khawli, Leslie A, Kaslow, Harvey R, Epstein, Alan L
Published in International journal of molecular sciences (20.12.2017)
Published in International journal of molecular sciences (20.12.2017)
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Compartmental Tissue Distribution of Antibody Therapeutics: Experimental Approaches and Interpretations
Boswell, C. Andrew, Bumbaca, Daniela, Fielder, Paul J., Khawli, Leslie A.
Published in The AAPS journal (01.09.2012)
Published in The AAPS journal (01.09.2012)
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Biodistribution and efficacy of an anti-TENB2 antibody-drug conjugate in a patient-derived model of prostate cancer
Boswell, C. Andrew, Yadav, Daniela Bumbaca, Mundo, Eduardo E., Yu, Shang-Fan, Lacap, Jennifer Arca, Fourie-O’Donohue, Aimee, Kozak, Katherine R., Ferl, Gregory Z., Zhang, Crystal, Ho, Jason, Ulufatu, Sheila, Khawli, Leslie A., Lin, Kedan
Published in Oncotarget (22.10.2019)
Published in Oncotarget (22.10.2019)
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