Fatty acid amide hydrolase inhibitors--progress and potential
Khanna, Ish K, Alexander, Christopher W
Published in CNS & neurological disorders drug targets (01.08.2011)
Published in CNS & neurological disorders drug targets (01.08.2011)
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Journal Article
Buprenorphine - an attractive opioid with underutilized potential in treatment of chronic pain
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Journal Article
Book Review
1,2-Diarylimidazoles as Potent, Cyclooxygenase-2 Selective, and Orally Active Antiinflammatory Agents
Khanna, Ish K, Weier, Richard M, Yu, Yi, Xu, Xiang D, Koszyk, Francis J, Collins, Paul W, Koboldt, Carol M, Veenhuizen, Amy W, Perkins, William E, Casler, Jacquelen J, Masferrer, Jaime L, Zhang, Yan Y, Gregory, Susan A, Seibert, Karen, Isakson, Peter C
Published in Journal of medicinal chemistry (23.05.1997)
Published in Journal of medicinal chemistry (23.05.1997)
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Journal Article
1,2-Diarylpyrroles as Potent and Selective Inhibitors of Cyclooxygenase-2
Khanna, Ish K, Weier, Richard M, Yu, Yi, Collins, Paul W, Miyashiro, Julie M, Koboldt, Carol M, Veenhuizen, Amy W, Currie, Jerry L, Seibert, Karen, Isakson, Peter C
Published in Journal of medicinal chemistry (23.05.1997)
Published in Journal of medicinal chemistry (23.05.1997)
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Convergent, parallel synthesis of a series of β-substituted 1,2,4-oxadiazole butanoic acids as potent and selective αvβ3 receptor antagonists
BOYS, Mark L, SCHRETZMAN, Lori A, STENMARK, Heather G, HONGWEI WU, SPANGLER, Dale P, CLARE, Michael, DESAI, Bipin N, KHANNA, Ish K, NGUYEN, Maria N, DUFFIN, Tiffany, WAYNE ENGLEMAN, V, FINN, Mary Beth, CHANDRAKUMAR, Nizal S, FREEMAN, Sandra K, HANNEKE, Melanie L, KEENE, Jeffery L, KLOVER, Jon A, NICKOLS, G. Allen, NICKOLS, Maureen A, STEININGER, Christina N, WESTLIN, Marisa, WESTLIN, William, YU, Yi X, TOLLEFSON, Michael B, YAPING WANG, DALTON, Christopher R, NORRING, Sarah A, MOHLER, Scott B, DOWNS, Victoria L, PENNING, Thomas D, RUSSELL, Mark A, WENDT, John A, CHEN, Barbara B
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Discovery of + (2 -{4 -[2 -(5,6,7,8 -tetrahydro -1,8 -naphthyridin -2-yl )ethoxy ]phenyl} -cyclopropyl )acetic acid as potent and selective αvβ3 inhibitor : Design, synthesis, and optimization
NAGARAJAN, Srinivasan R, LU, Hwang-Fun, KEENE, Jeffery L, DUFFIN, Tiffany, ENGLEMAN, V. Wayne, FINN, Mary B, FREEMAN, Sandra K, KLOVER, Jon A, NICKOLS, G. Alan, NICKOLS, Maureen A, SHANNON, Kristen E, STEININGER, Christina A, GASIECKI, Alan F, WESTLIN, William F, WESTLIN, Marisa M, WILLIAMS, Melanie L, KHANNA, Ish K, PARIKH, Mihir D, DESAI, Bipinchandra N, ROGERS, Thomas E, CLARE, Michael, CHEN, Barbara B, RUSSELL, Mark A
Published in Bioorganic & medicinal chemistry (15.05.2007)
Published in Bioorganic & medicinal chemistry (15.05.2007)
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Journal Article
Facile, Regioselective Syntheses of N-Alkylated 2,3-Diaminopyridines and Imidazo[4,5-b]pyridines
Khanna, Ish K, Weier, Richard M, Lentz, Kirk T, Swenton, Lydia, Lankin, David C
Published in Journal of organic chemistry (01.02.1995)
Published in Journal of organic chemistry (01.02.1995)
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Journal Article
Selective Cyclooxygenase-2 Inhibitors: Heteroaryl Modified 1,2-Diarylimidazoles Are Potent, Orally Active Antiinflammatory Agents
Khanna, Ish K, Yu, Yi, Huff, Renee M, Weier, Richard M, Xu, Xiangdong, Koszyk, Francis J, Collins, Paul W, Cogburn, J. Nita, Isakson, Peter C, Koboldt, Carol M, Masferrer, Jaime L, Perkins, William E, Seibert, Karen, Veenhuizen, Amy W, Yuan, Jinhua, Yang, Dai-Chang, Zhang, Yan Y
Published in Journal of medicinal chemistry (10.08.2000)
Published in Journal of medicinal chemistry (10.08.2000)
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Journal Article
SUBSTITUTED PYRAZOLYL BENZENE SULFONEAMIDES FOR THE TREATMENT OF INFLAMMATION
ROGIER, DONALD J. JR, TALLEY, JOHN J, MIYASHIRO, JULIE M, KHANNA, ISH K, YU, STELLA S, ROGERS, ROLAND S, BERTENSHAW, STEPHEN R, GRANETS, MATTHEW J, COLLINS, PAUL W, DOCTER, STEPHEN H, CARTER, JEFFERY S, PENNING, THOMAS D, MALECHA, JAMES W
Year of Publication 01.11.1999
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Year of Publication 01.11.1999
Patent
Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective alphavbeta3 inhibitor: design, synthesis, and optimization
Nagarajan, Srinivasan R, Lu, Hwang-Fun, Gasiecki, Alan F, Khanna, Ish K, Parikh, Mihir D, Desai, Bipinchandra N, Rogers, Thomas E, Clare, Michael, Chen, Barbara B, Russell, Mark A, Keene, Jeffery L, Duffin, Tiffany, Engleman, V Wayne, Finn, Mary B, Freeman, Sandra K, Klover, Jon A, Nickols, G Alan, Nickols, Maureen A, Shannon, Kristen E, Steininger, Christina A, Westlin, William F, Westlin, Marisa M, Williams, Melanie L
Published in Bioorganic & medicinal chemistry (15.05.2007)
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Published in Bioorganic & medicinal chemistry (15.05.2007)
Journal Article
Discovery of +(2-{4-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethoxy]phenyl}-cyclopropyl)acetic acid as potent and selective α vβ 3 inhibitor: Design, synthesis, and optimization
Nagarajan, Srinivasan R., Lu, Hwang-Fun, Gasiecki, Alan F., Khanna, Ish K., Parikh, Mihir D., Desai, Bipinchandra N., Rogers, Thomas E., Clare, Michael, Chen, Barbara B., Russell, Mark A., Keene, Jeffery L., Duffin, Tiffany, Engleman, V. Wayne, Finn, Mary B., Freeman, Sandra K., Klover, Jon A., Nickols, G. Alan, Nickols, Maureen A., Shannon, Kristen E., Steininger, Christina A., Westlin, William F., Westlin, Marisa M., Williams, Melanie L.
Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
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Journal Article
Convergent, parallel synthesis of a series of beta-substituted 1,2,4-oxadiazole butanoic acids as potent and selective alpha(v)beta3 receptor antagonists
Boys, Mark L, Schretzman, Lori A, Chandrakumar, Nizal S, Tollefson, Michael B, Mohler, Scott B, Downs, Victoria L, Penning, Thomas D, Russell, Mark A, Wendt, John A, Chen, Barbara B, Stenmark, Heather G, Wu, Hongwei, Spangler, Dale P, Clare, Michael, Desai, Bipin N, Khanna, Ish K, Nguyen, Maria N, Duffin, Tiffany, Engleman, V Wayne, Finn, Mary Beth, Freeman, Sandra K, Hanneke, Melanie L, Keene, Jeffery L, Klover, Jon A, Nickols, G Allen, Nickols, Maureen A, Steininger, Christina N, Westlin, Marisa, Westlin, William, Yu, Yi X, Wang, Yaping, Dalton, Christopher R, Norring, Sarah A
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Journal Article
Convergent, parallel synthesis of a series of beta -substituted 1,2,4- oxadiazole butanoic acids as potent and selective alpha sub(v) beta sub(3) receptor antagonists
Boys, Mark L, Schretzman, Lori A, Chandrakumar, Nizal S, Tollefson, Michael B, Mohler, Scott B, Downs, Victoria L, Penning, Thomas D, Russell, Mark A, Wendt, John A, Chen, Barbara B, Stenmark, Heather G, Wu, Hongwei, Spangler, Dale P, Clare, Michael, Desai, Bipin N, Khanna, Ish K, Nguyen, Maria N, Duffin, Tiffany, Engleman, VWayne, Finn, Mary Beth, Freeman, Sandra K, Hanneke, Melanie L, Keene, Jeffery L, Klover, Jon A, Nickols, GAllen, Nickols, Maureen A, Steininger, Christina N, Westlin, Marisa, Westlin, William, Yu, Yi X, Wang, Yaping, Dalton, Christopher R, Norring, Sarah A
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Journal Article
Convergent, parallel synthesis of a series of β-substituted 1,2,4-oxadiazole butanoic acids as potent and selective α vβ 3 receptor antagonists
Boys, Mark L., Schretzman, Lori A., Chandrakumar, Nizal S., Tollefson, Michael B., Mohler, Scott B., Downs, Victoria L., Penning, Thomas D., Russell, Mark A., Wendt, John A., Chen, Barbara B., Stenmark, Heather G., Wu, Hongwei, Spangler, Dale P., Clare, Michael, Desai, Bipin N., Khanna, Ish K., Nguyen, Maria N., Duffin, Tiffany, Engleman, V. Wayne, Finn, Mary Beth, Freeman, Sandra K., Hanneke, Melanie L., Keene, Jeffery L., Klover, Jon A., Nickols, G. Allen, Nickols, Maureen A., Steininger, Christina N., Westlin, Marisa, Westlin, William, Yu, Yi X., Wang, Yaping, Dalton, Christopher R., Norring, Sarah A.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Journal Article
The synthesis of 1,5-dideoxy-1,5-(alkyl)imino-2-C-methyl- d-glucitols
Khanna, Ish K., Weier, Richard M., Julien, Janet, Mueller, Richard A., Lankin, David C., Swenton, Lydia
Published in Tetrahedron letters (26.02.1996)
Published in Tetrahedron letters (26.02.1996)
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Journal Article
SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS
GRANETO, Matthew J, WEIER, Richard M, MALECHA, James W, NAGARAJAN, Srinivasan, KHANNA, Ish K, TALLEY, John J, CARTER, Jeffrey, BERTENSHAW, Stephen, XU, Xiangdong, ROGIER, Donald J, Jr, LI, Jinglin, BROWN, David L, PENNING, Thomas D
Year of Publication 10.10.2011
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Year of Publication 10.10.2011
Patent