Search Results - "KEVIN SHREDER" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors

Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors

by Li, Bei, Cociorva, Oana M., Nomanbhoy, Tyzoon, Weissig, Helge, Li, Qiang, Nakamura, Kai, Liyanage, Marek, Zhang, Melissa C., Shih, Ann Y., Aban, Arwin, Hu, Yi, Cajica, Julia, Pham, Lan, Kozarich, John W., Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (15.09.2013)

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Journal Article

Quinolone derivatives containing strained spirocycle as orally active glycogen synthase kinase 3β (GSK-3β) inhibitors for type 2 diabetics

Quinolone derivatives containing strained spirocycle as orally active glycogen synthase kinase 3β (GSK-3β) inhibitors for type 2 diabetics

by Seto, Shigeki, Yumoto, Kazuhiko, Okada, Kyoko, Asahina, Yoshikazu, Iwane, Aya, Iwago, Maki, Terasawa, Reiko, Shreder, Kevin R., Murakami, Koji, Kohno, Yasushi
Published in Bioorganic & medicinal chemistry (01.02.2012)

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High-Resolution Functional Proteomics by Active-Site Peptide Profiling

High-Resolution Functional Proteomics by Active-Site Peptide Profiling

by Okerberg, Eric S., Wu, Jiangyue, Zhang, Baohong, Samii, Babak, Blackford, Kelly, Winn, David T., Shreder, Kevin R., Burbaum, Jonathan J., Patricelli, Matthew P., Stubbe, JoAnne
Published in Proceedings of the National Academy of Sciences - PNAS (05.04.2005)

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Amides of 4-hydroxy-8-methanesulfonylamino-quinoline-2-carboxylic acid as zinc-dependent inhibitors of Lp-PLA(2)

Amides of 4-hydroxy-8-methanesulfonylamino-quinoline-2-carboxylic acid as zinc-dependent inhibitors of Lp-PLA(2)

by Hu, Yi, Lin, Emme C. K., Pham, Lan M., Cajica, Julia, Amantea, Christopher M., Okerberg, Eric, Brown, Heidi E., Fraser, Allister, Du, Lingling, Kohno, Yasushi, Ishiyama, Junichi, Kozarich, John W., Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (01.03.2013)

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Synthesis and structure–activity relationship of 4-quinolone-3-carboxylic acid based inhibitors of glycogen synthase kinase-3β

Synthesis and structure–activity relationship of 4-quinolone-3-carboxylic acid based inhibitors of glycogen synthase kinase-3β

by Cociorva, Oana M., Li, Bei, Nomanbhoy, Tyzoon, Li, Qiang, Nakamura, Ayako, Nakamura, Kai, Nomura, Masahiro, Okada, Kyoko, Seto, Shigeki, Yumoto, Kazuhiro, Liyanage, Marek, Zhang, Melissa C., Aban, Arwin, Leen, Brandon, Szardenings, Anna Katrin, Rosenblum, Jonathan S., Kozarich, John W., Kohno, Yasushi, Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (01.10.2011)

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Amides of xanthurenic acid as zinc-dependent inhibitors of Lp-PLA

Amides of xanthurenic acid as zinc-dependent inhibitors of Lp-PLA

by Lin, Emme C.K, Hu, Yi, Amantea, Christopher M, Pham, Lan M, Cajica, Julia, Okerberg, Eric, Brown, Heidi E, Fraser, Allister, Du, Lingling, Kohno, Yasushi, Ishiyama, Junichi, Kozarich, John W, Shreder, Kevin R
Published in Bioorganic & medicinal chemistry letters (15.01.2012)

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Synthesis and structure–activity relationship of (1-halo-2-naphthyl) carbamate-based inhibitors of KIAA1363 (NCEH1/AADACL1)

Synthesis and structure–activity relationship of (1-halo-2-naphthyl) carbamate-based inhibitors of KIAA1363 (NCEH1/AADACL1)

by Shreder, Kevin R., Lin, Emme C.K., Wu, Jiangyue, Cajica, Julia, Amantea, Christopher M., Hu, Yi, Okerberg, Eric, Brown, Heidi E., Pham, Lan M., Chung, De Michael, Fraser, Allister S., McGee, Ethel, Rosenblum, Jonathan S., Kozarich, John W.
Published in Bioorganic & medicinal chemistry letters (01.09.2012)

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6-Position optimization of tricyclic 4-quinolone-based inhibitors of glycogen synthase kinase-3β: Discovery of nitrile derivatives with picomolar potency

6-Position optimization of tricyclic 4-quinolone-based inhibitors of glycogen synthase kinase-3β: Discovery of nitrile derivatives with picomolar potency

by Li, Bei, Cociorva, Oana M., Nomanbhoy, Tyzoon, Li, Qiang, Nakamura, Kai, Nomura, Masahiro, Okada, Kyoko, Yumoto, Kazuhiro, Liyanage, Marek, Zhang, Melissa C., Aban, Arwin, Szardenings, Anna Katrin, Kozarich, John W., Kohno, Yasushi, Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (15.01.2012)

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Journal Article

Synthesis of AX7593, a Quinazoline-Derived Photoaffinity Probe for EGFR

Synthesis of AX7593, a Quinazoline-Derived Photoaffinity Probe for EGFR

by Shreder, Kevin R, Wong, Melissa S, Nomanbhoy, Tyzoon, Leventhal, Phillip S, Fuller, Stacy R
Published in Organic letters (14.10.2004)

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Synthesis and optimization of 2-pyridin-3-yl-benzo[ d][1,3]oxazin-4-one based inhibitors of human neutrophil elastase

Synthesis and optimization of 2-pyridin-3-yl-benzo[ d][1,3]oxazin-4-one based inhibitors of human neutrophil elastase

by Shreder, Kevin R., Cajica, Julia, Du, Lingling, Fraser, Allister, Hu, Yi, Kohno, Yasushi, Lin, Emme C.K., Liu, Steve J., Okerberg, Eric, Pham, Lan, Wu, Jiangyue, Kozarich, John W.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)

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Amides of xanthurenic acid as zinc-dependent inhibitors of Lp-PLA2

Amides of xanthurenic acid as zinc-dependent inhibitors of Lp-PLA2

by Lin, Emme C.K., Hu, Yi, Amantea, Christopher M., Pham, Lan M., Cajica, Julia, Okerberg, Eric, Brown, Heidi E., Fraser, Allister, Du, Lingling, Kohno, Yasushi, Ishiyama, Junichi, Kozarich, John W., Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (15.01.2012)

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Journal Article

Protonated Sapphyrins. Highly Effective Phosphate Receptors

Protonated Sapphyrins. Highly Effective Phosphate Receptors

by Král, Vladimír, Furuta, Hiroyuki, Shreder, Kevin, Lynch, Vincent, Sessler, Jonathan L
Published in Journal of the American Chemical Society (21.02.1996)

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Design and Synthesis of AX7574: A Microcystin-Derived, Fluorescent Probe for Serine/Threonine Phosphatases

Design and Synthesis of AX7574: A Microcystin-Derived, Fluorescent Probe for Serine/Threonine Phosphatases

by Shreder, Kevin R, Liu, Yongsheng, Nomanhboy, Tyzoon, Fuller, Stacy R, Wong, Melissa S, Gai, Wen Zhi, Wu, Jiangyue, Leventhal, Phillip S, Lill, Jennie R, Corral, Sergio
Published in Bioconjugate chemistry (01.07.2004)

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Journal Article

Design and synthesis of AX4697, a bisindolylmaleimide exo-affinity probe that labels protein kinase C alpha and beta

Design and synthesis of AX4697, a bisindolylmaleimide exo-affinity probe that labels protein kinase C alpha and beta

by Liu, Yongsheng, Wu, Jiangyue, Weissig, Helge, Betancort, Juan M., Gai, Wen Zhi, Leventhal, Phillip S., Patricelli, Matthew P., Samii, Babak, Szardenings, Anna K., Shreder, Kevin R., Kozarich, John W.
Published in Bioorganic & medicinal chemistry (15.11.2008)

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Synthesis and structure–activity relationship of N-alkyl Gly-boro-Pro inhibitors of DPP4, FAP, and DPP7

Synthesis and structure–activity relationship of N-alkyl Gly-boro-Pro inhibitors of DPP4, FAP, and DPP7

by Hu, Yi, Ma, Lifu, Wu, Min, Wong, Melissa S., Li, Bei, Corral, Sergio, Yu, Zhizhou, Nomanbhoy, Tyzoon, Alemayehu, Senaiet, Fuller, Stacy R., Rosenblum, Jonathan S., Rozenkrants, Natasha, Minimo, Lauro C., Ripka, William C., Szardenings, Anna K., Kozarich, John W., Shreder, Kevin R.
Published in Bioorganic & medicinal chemistry letters (01.10.2005)

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Quenching of Biotinylated Aequorin Bioluminescence by Dye-Labeled Avidin Conjugates: Application to Homogeneous Bioluminescence Resonance Energy Transfer Assays

Quenching of Biotinylated Aequorin Bioluminescence by Dye-Labeled Avidin Conjugates: Application to Homogeneous Bioluminescence Resonance Energy Transfer Assays

by Adamczyk, Maciej, Moore, Jeffrey A, Shreder, Kevin
Published in Organic letters (14.06.2001)

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Journal Article

Synthesis of a constrained enkephalin analog to illustrate a novel route to the piperazinone ring structure

Synthesis of a constrained enkephalin analog to illustrate a novel route to the piperazinone ring structure

by Shreder, Kevin, Zhang, Li, Goodman, Murray
Published in Tetrahedron letters (01.01.1998)

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Journal Article

Boro-norleucine as a P1 residue for the design of selective and potent DPP7 inhibitors

Boro-norleucine as a P1 residue for the design of selective and potent DPP7 inhibitors

by Shreder, Kevin R., Wong, Melissa S., Corral, Sergio, Yu, Zhizhou, Winn, David T., Wu, Min, Hu, Yi, Nomanbhoy, Tyzoon, Alemayehu, Senaiet, Fuller, Stacy R., Rosenblum, Jonathan S., Kozarich, John W.
Published in Bioorganic & medicinal chemistry letters (01.10.2005)

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Region-Selective Labeling of Antibodies as Determined by Electrospray Ionization-Mass Spectrometry (ESI-MS)

Region-Selective Labeling of Antibodies as Determined by Electrospray Ionization-Mass Spectrometry (ESI-MS)

by Adamczyk, Maciej, Gebler, John, Shreder, Kevin, Wu, Jiang
Published in Bioconjugate chemistry (01.07.2000)

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Journal Article

Wortmannin, a Widely Used Phosphoinositide 3-Kinase Inhibitor, also Potently Inhibits Mammalian Polo-like Kinase

Wortmannin, a Widely Used Phosphoinositide 3-Kinase Inhibitor, also Potently Inhibits Mammalian Polo-like Kinase

by Liu, Yongsheng, Shreder, Kevin R., Gai, Wenzhi, Corral, Sergio, Ferris, Douglas K., Rosenblum, Jonathan S.
Published in Chemistry & biology (2005)

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