Pharmacologic inhibition of STAT5 in acute myeloid leukemia
Wingelhofer, Bettina, Maurer, Barbara, Heyes, Elizabeth C., Cumaraswamy, Abbarna A., Berger-Becvar, Angelika, de Araujo, Elvin D., Orlova, Anna, Freund, Patricia, Ruge, Frank, Park, Jisung, Tin, Gary, Ahmar, Siawash, Lardeau, Charles-Hugues, Sadovnik, Irina, Bajusz, Dávid, Keserű, György Miklós, Grebien, Florian, Kubicek, Stefan, Valent, Peter, Gunning, Patrick T., Moriggl, Richard
Published in Leukemia (01.05.2018)
Published in Leukemia (01.05.2018)
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Designed Peptide Inhibitors of STEP Phosphatase–GluA2 AMPA Receptor Interaction Enhance the Cognitive Performance in Rats
Szedlacsek, Horea Stefan, Bajusz, Dávid, Badea, Rodica Aura, Pop, Andreea, Bică, Constantin Cătălin, Ravasz, Lilla, Mittli, Dániel, Mátyás, Dominik, Necula-Petrăreanu, Georgiana, Munteanu, Cristian V. A, Papp, Ildikó, Juhász, Gábor, Hritcu, Lucian, Keserű, György Miklós, Szedlacsek, Stefan Eugen
Published in Journal of medicinal chemistry (13.01.2022)
Published in Journal of medicinal chemistry (13.01.2022)
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Cysteine specific bioconjugation with benzyl isothiocyanates
Petri, László, Szijj, Péter A, Kelemen, Ádám, Imre, Tímea, Gömöry, Ágnes, Lee, Maximillian T. W, Heged s, Krisztina, Ábrányi-Balogh, Péter, Chudasama, Vijay, Keser, György Miklós
Published in RSC advances (16.04.2020)
Published in RSC advances (16.04.2020)
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A novel three-component reaction between isocyanides, alcohols or thiols and elemental sulfur: a mild, catalyst-free approach towards O -thiocarbamates and dithiocarbamates
Németh, András György, Keserű, György Miklós, Ábrányi-Balogh, Péter
Published in Beilstein journal of organic chemistry (10.07.2019)
Published in Beilstein journal of organic chemistry (10.07.2019)
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Effective synthesis, development and application of a highly fluorescent cyanine dye for antibody conjugation and microscopy imaging
Szepesi Kovács, Dénes, Kontra, Bence, Chiovini, Balázs, Müller, Dalma, Tóth, Estilla Zsófia, Ábrányi-Balogh, Péter, Wittner, Lucia, Várady, György, Turczel, Gábor, Farkas, Ödön, Owen, Michael C, Katona, Gergely, Gy rffy, Balázs, Keser, György Miklós, Mucsi, Zoltán, Rózsa, Balázs J, Kovács, Ervin
Published in Organic & biomolecular chemistry (15.11.2023)
Published in Organic & biomolecular chemistry (15.11.2023)
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Synthesis and characterization of new fluorescent boro-β-carboline dyes
Szepesi Kovács, Dénes, Hajdu, Imre, Mészáros, Gergely, Wittner, Lucia, Meszéna, Domokos, Tóth, Estilla Zsófia, Heged s, Zita, Ran elovi, Ivan, Tóvári, József, Szabó, Tímea, Szilágyi, Bence, Milen, Mátyás, Keser, György Miklós, Ábrányi-Balogh, Péter
Published in RSC advances (01.04.2021)
Published in RSC advances (01.04.2021)
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Synthesis and fluorescent properties of boroisoquinolines, a new family of fluorophores
Sóvári, Dénes, Kormos, Attila, Demeter, Orsolya, Dancsó, András, Keserű, György Miklós, Milen, Mátyás, Ábrányi-Balogh, Péter
Published in RSC advances (01.01.2018)
Published in RSC advances (01.01.2018)
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Bromo-Cyclobutenaminones as New Covalent UDP-N-Acetylglucosamine Enolpyruvyl Transferase (MurA) Inhibitors
Hamilton, David J., Ábrányi-Balogh, Péter, Keeley, Aaron, Petri, László, Hrast, Martina, Imre, Tímea, Wijtmans, Maikel, Gobec, Stanislav, Esch, Iwan J. P. de, Keserű, György Miklós
Published in Pharmaceuticals (Basel, Switzerland) (03.11.2020)
Published in Pharmaceuticals (Basel, Switzerland) (03.11.2020)
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Synthesis and Application of Two-Photon Active Fluorescent Rhodol Dyes for Antibody Conjugation and In Vitro Cell Imaging
Szepesi Kovács, Dénes, Chiovini, Balázs, Müller, Dalma, Tóth, Estilla Zsófia, Fülöp, Anna, Ábrányi-Balogh, Péter, Wittner, Lucia, Várady, György, Farkas, Ödön, Turczel, Gábor, Katona, Gergely, Győrffy, Balázs, Keserű, György Miklós, Mucsi, Zoltán, Rózsa, Balázs J., Kovács, Ervin
Published in ACS omega (27.06.2023)
Published in ACS omega (27.06.2023)
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Antioxidant activity-guided phytochemical investigation of Artemisia gmelinii Webb. ex Stechm.: Isolation and spectroscopic challenges of 3,5- O-dicaffeoyl (epi?) quinic acid and its ethyl ester
Könczöl, Árpád, Béni, Zoltán, Sipos, Márta Meszlényi, Rill, Attila, Háda, Viktor, Hohmann, Judit, Máthé, Imre, Szántay, Csaba, Keserű, György Miklós, Balogh, György Tibor
Published in Journal of pharmaceutical and biomedical analysis (05.02.2012)
Published in Journal of pharmaceutical and biomedical analysis (05.02.2012)
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Electrophilic warheads in covalent drug discovery: an overview
Péczka, Nikolett, Orgován, Zoltán, Ábrányi-Balogh, Péter, Keserű, György Miklós
Published in Expert opinion on drug discovery (03.04.2022)
Published in Expert opinion on drug discovery (03.04.2022)
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Comparative reactivity analysis of small-molecule thiol surrogates
Petri, László, Ábrányi-Balogh, Péter, Varga, Petra Regina, Imre, Tímea, Keserű, György Miklós
Published in Bioorganic & medicinal chemistry (01.04.2020)
Published in Bioorganic & medicinal chemistry (01.04.2020)
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Allosteric regulation and crystallographic fragment screening of SARS-CoV-2 NSP15 endoribonuclease
Godoy, Andre Schutzer, Nakamura, Aline Minalli, Douangamath, Alice, Song, Yun, Noske, Gabriela Dias, Gawriljuk, Victor Oliveira, Fernandes, Rafaela Sachetto, Pereira, Humberto D Muniz, Oliveira, Ketllyn Irene Zagato, Fearon, Daren, Dias, Alexandre, Krojer, Tobias, Fairhead, Michael, Powell, Alisa, Dunnet, Louise, Brandao-Neto, Jose, Skyner, Rachael, Chalk, Rod, Bajusz, Dávid, Bege, Miklós, Borbás, Anikó, Keserű, György Miklós, von Delft, Frank, Oliva, Glaucius
Published in Nucleic acids research (09.06.2023)
Published in Nucleic acids research (09.06.2023)
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Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile
Ágai-Csongor, Éva, Nógrádi, Katalin, Galambos, János, Vágó, István, Bielik, Attila, Magdó, Ildikó, Ignácz-Szendrei, Györgyi, Keserű, György Miklós, Greiner, István, Laszlovszky, István, Béla Kiss, Éva Schmidt, Judit Laszy, Katalin Sághy, Gyertyán, István, Zájer-Balázs, Mária, Gémesi, Larisza, Domány, György
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Emerging therapeutic targets in myeloproliferative neoplasms and peripheral T-cell leukemia and lymphomas
Orlova, Anna, Wingelhofer, Bettina, Neubauer, Heidi A., Maurer, Barbara, Berger-Becvar, Angelika, Keserű, György Miklós, Gunning, Patrick T., Valent, Peter, Moriggl, Richard
Published in Expert opinion on therapeutic targets (02.01.2018)
Published in Expert opinion on therapeutic targets (02.01.2018)
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Fingerprint-Based Machine Learning Approach to Identify Potent and Selective 5-HT2BR Ligands
Rataj, Krzysztof, Kelemen, Ádám, Brea, José, Loza, María, Bojarski, Andrzej, Keserű, György
Published in Molecules (Basel, Switzerland) (10.05.2018)
Published in Molecules (Basel, Switzerland) (10.05.2018)
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The first synthesis of furo[2,3-c]pyridazin-4(1H)-one derivatives
Kelemen, Adam Andor, Szabo, Balazs Peter, Kovacs, Peter, Kesertu, Gyoergy Miklos
Published in Tetrahedron letters (06.01.2016)
Published in Tetrahedron letters (06.01.2016)
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Positive allosteric modulators for mGluR2 receptors: a medicinal chemistry perspective
Szabó, György, Keserű, György Miklós
Published in Current topics in medicinal chemistry (01.01.2014)
Published in Current topics in medicinal chemistry (01.01.2014)
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Natural Apocarotenoids and Their Synthetic Glycopeptide Conjugates Inhibit SARS-CoV-2 Replication
Bereczki, Ilona, Papp, Henrietta, Kuczmog, Anett, Madai, Mónika, Nagy, Veronika, Agócs, Attila, Batta, Gyula, Milánkovits, Márton, Ostorházi, Eszter, Mitrović, Ana, Kos, Janko, Zsigmond, Áron, Hajdú, István, Lőrincz, Zsolt, Bajusz, Dávid, Keserű, György Miklós, Hodek, Jan, Weber, Jan, Jakab, Ferenc, Herczegh, Pál, Borbás, Anikó
Published in Pharmaceuticals (Basel, Switzerland) (30.10.2021)
Published in Pharmaceuticals (Basel, Switzerland) (30.10.2021)
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