In Vitro Activity of E1210, a Novel Antifungal, against Clinically Important Yeasts and Molds
MIYAZAKI, Mamiko, HORII, Takaaki, ABE, Shinya, YOSHIMATSU, Kentaro, ASADA, Makoto, HATA, Katsura, WATANABE, Nao-Aki, NAKAMOTO, Kazutaka, TANAKA, Keigo, SHIROTORI, Syuji, MURAI, Norio, INOUE, Satoshi, MATSUKURA, Masayuki
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
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Lyn Kinase Suppresses the Transcriptional Activity of IRF5 in the TLR-MyD88 Pathway to Restrain the Development of Autoimmunity
Ban, Tatsuma, Sato, Go R., Nishiyama, Akira, Akiyama, Ai, Takasuna, Marie, Umehara, Marina, Suzuki, Shinsuke, Ichino, Motohide, Matsunaga, Satoko, Kimura, Ayuko, Kimura, Yayoi, Yanai, Hideyuki, Miyashita, Sadakazu, Kuromitsu, Junro, Tsukahara, Kappei, Yoshimatsu, Kentaro, Endo, Itaru, Yamamoto, Tadashi, Hirano, Hisashi, Ryo, Akihide, Taniguchi, Tadatsugu, Tamura, Tomohiko
Published in Immunity (Cambridge, Mass.) (16.08.2016)
Published in Immunity (Cambridge, Mass.) (16.08.2016)
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Efficacy of Oral E1210, a New Broad-Spectrum Antifungal with a Novel Mechanism of Action, in Murine Models of Candidiasis, Aspergillosis, and Fusariosis
Hata, Katsura, Horii, Takaaki, Miyazaki, Mamiko, Watanabe, Nao-aki, Okubo, Miyuki, Sonoda, Jiro, Nakamoto, Kazutaka, Tanaka, Keigo, Shirotori, Syuji, Murai, Norio, Inoue, Satoshi, Matsukura, Masayuki, Abe, Shinya, Yoshimatsu, Kentaro, Asada, Makoto
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
Published in Antimicrobial Agents and Chemotherapy (01.10.2011)
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Genetic and chemical inhibition of IRF5 suppresses pre-existing mouse lupus-like disease
Ban, Tatsuma, Kikuchi, Masako, Sato, Go R., Manabe, Akio, Tagata, Noriko, Harita, Kayo, Nishiyama, Akira, Nishimura, Kenichi, Yoshimi, Ryusuke, Kirino, Yohei, Yanai, Hideyuki, Matsumoto, Yoshiko, Suzuki, Shuichi, Hihara, Hiroe, Ito, Masashi, Tsukahara, Kappei, Yoshimatsu, Kentaro, Yamamoto, Tadashi, Taniguchi, Tadatsugu, Nakajima, Hideaki, Ito, Shuichi, Tamura, Tomohiko
Published in Nature communications (19.07.2021)
Published in Nature communications (19.07.2021)
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M-COPA, a Golgi Disruptor, Inhibits Cell Surface Expression of MET Protein and Exhibits Antitumor Activity against MET-Addicted Gastric Cancers
Ohashi, Yoshimi, Okamura, Mutsumi, Hirosawa, Asaka, Tamaki, Naomi, Akatsuka, Akinobu, Wu, Kuo-Ming, Choi, Hyeong-Wook, Yoshimatsu, Kentaro, Shiina, Isamu, Yamori, Takao, Dan, Shingo
Published in Cancer research (Chicago, Ill.) (01.07.2016)
Published in Cancer research (Chicago, Ill.) (01.07.2016)
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Targeting the Golgi apparatus to overcome acquired resistance of non-small cell lung cancer cells to EGFR tyrosine kinase inhibitors
Ohashi, Yoshimi, Okamura, Mutsumi, Katayama, Ryohei, Fang, Siyang, Tsutsui, Saki, Akatsuka, Akinobu, Shan, Mingde, Choi, Hyeong-Wook, Fujita, Naoya, Yoshimatsu, Kentaro, Shiina, Isamu, Yamori, Takao, Dan, Shingo
Published in Oncotarget (05.01.2018)
Published in Oncotarget (05.01.2018)
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Stem Cell Factor/c-kit Signaling Promotes the Survival, Migration, and Capillary Tube Formation of Human Umbilical Vein Endothelial Cells
Matsui, Junji, Wakabayashi, Toshiaki, Asada, Makoto, Yoshimatsu, Kentaro, Okada, Masayuki
Published in The Journal of biological chemistry (30.04.2004)
Published in The Journal of biological chemistry (30.04.2004)
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Synthesis and evaluation of novel antifungal agents-quinoline and pyridine amide derivatives
Nakamoto, Kazutaka, Tsukada, Itaru, Tanaka, Keigo, Matsukura, Masayuki, Haneda, Toru, Inoue, Satoshi, Murai, Norio, Abe, Shinya, Ueda, Norihiro, Miyazaki, Mamiko, Watanabe, Naoaki, Asada, Makoto, Yoshimatsu, Kentaro, Hata, Katsura
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Discovery of Novel Antitumor Sulfonamides Targeting G1 Phase of the Cell Cycle
Owa, Takashi, Yoshino, Hiroshi, Okauchi, Tatsuo, Yoshimatsu, Kentaro, Ozawa, Yoichi, Sugi, Naoko Hata, Nagasu, Takeshi, Koyanagi, Nozomu, Kitoh, Kyosuke
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Pladienolides, New Substances from Culture of Streptomyces platensis Mer-11107: III. In Vitro and In Vivo Antitumor Activities
MIZUI, YOSHIHARU, SAKAI, TAKASHI, IWATA, MASAO, UENAKA, TOSHIMITSU, OKAMOTO, KIYOSHI, SHIMIZU, HAJIME, YAMORI, TAKAO, YOSHIMATSU, KENTARO, ASADA, MAKOTO
Published in Journal of antibiotics (01.03.2004)
Published in Journal of antibiotics (01.03.2004)
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Report of the international conference on regulatory endeavors towards the sound development of human cell therapy products
Hayakawa, Takao, Aoi, Takashi, Bravery, Christopher, Hoogendoorn, Karin, Knezevic, Ivana, Koga, Junichi, Maeda, Daisuke, Matsuyama, Akifumi, McBlane, James, Morio, Tomohiro, Petricciani, John, Rao, Mahendra, Ridgway, Anthony, Sato, Daisaku, Sato, Yoji, Stacey, Glyn, Sakamoto, Norihisa, Trouvin, Jean-Hugues, Umezawa, Akihiro, Yamato, Masayuki, Yano, Kazuo, Yokote, Hiroyuki, Yoshimatsu, Kentaro, Zorzi-Morre, Pierrette
Published in Biologicals (01.09.2015)
Published in Biologicals (01.09.2015)
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Conference Proceeding
Medicinal genetics approach towards identifying the molecular target of a novel inhibitor of fungal cell wall assembly
Tsukahara, Kappei, Hata, Katsura, Nakamoto, Kazutaka, Sagane, Koji, Watanabe, Nao‐aki, Kuromitsu, Junro, Kai, Junko, Tsuchiya, Mamiko, Ohba, Fuminori, Jigami, Yoshifumi, Yoshimatsu, Kentaro, Nagasu, Takeshi
Published in Molecular microbiology (01.05.2003)
Published in Molecular microbiology (01.05.2003)
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Profiling Novel Sulfonamide Antitumor Agents with Cell-based Phenotypic Screens and Array-based Gene Expression Analysis
Yokoi, Akira, Kuromitsu, Junro, Kawai, Takatoshi, Nagasu, Takeshi, Sugi, Naoko Hata, Yoshimatsu, Kentaro, Yoshino, Hiroshi, Owa, Takashi
Published in Molecular cancer therapeutics (01.02.2002)
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Published in Molecular cancer therapeutics (01.02.2002)
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Synthesis and Evaluation of Novel Pyrimido-Acridone, -Phenoxadine, and -Carbazole as Topoisomerase II Inhibitors
Kamata, Junichi, Okada, Toshimi, Kotake, Yoshihiko, Niijima, Jun, Nakamura, Katsuji, Uenaka, Toshimitsu, Yamaguchi, Atsumi, Tsukahara, Kappei, Nagasu, Takeshi, Koyanagi, Nozomu, Kitoh, Kyosuke, Yoshimatsu, Kentaro, Yoshino, Hiroshi, Sugumi, Hiroyuki
Published in Chemical & Pharmaceutical Bulletin (01.09.2004)
Published in Chemical & Pharmaceutical Bulletin (01.09.2004)
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α6β1 integrin induces proteasome-mediated cleavage of erbB2 in breast cancer cells
SHIMIZU, Hajime, SEIKI, Takashi, ASADA, Makoto, YOSHIMATSU, Kentaro, KOYAMA, Noriyuki
Published in Oncogene (13.02.2003)
Published in Oncogene (13.02.2003)
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A focused compound library of novel N-(7-indolyl)benzenesulfonamides for the discovery of potent cell cycle inhibitors
OWA, T, OKAUCHI, T, YOSHIMATSU, K, SUGI, N. H, OZAWA, Y, NAGASU, T, KOYANAGI, N, OKABE, T, KITOH, K, YOSHINO, H
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
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A novel carbazole topoisomerase II poison, ER‐37328: potent tumoricidal activity against human solid tumors in vitro and in vivo
Nakamura, Katsuji, Uenaka, Toshimitsu, Nagasu, Takeshi, Sugumi, Hiroyuki, Yamaguchi, Atsumi, Kotake, Yoshihiko, Okada, Toshimi, Kamata, Junichi, Niijima, Jun, Taniguchi, Tomoyoshi, Koyanagi, Nozomu, Yoshino, Hiroshi, Kitoh, Kyosuke, Yoshimatsu, Kentaro
Published in Cancer science (01.01.2003)
Published in Cancer science (01.01.2003)
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Antitumor Activity of ER-37328, a Novel Carbazole Topoisomerase II Inhibitor
Nakamura, Katsuji, Sugumi, Hiroyuki, Yamaguchi, Atsumi, Uenaka, Toshimitsu, Kotake, Yoshihiko, Okada, Toshimi, Kamata, Junichi, Niijima, Jun, Nagasu, Takeshi, Koyanagi, Nozomu, Yoshino, Hiroshi, Kitoh, Kyosuke, Yoshimatsu, Kentaro
Published in Molecular cancer therapeutics (01.01.2002)
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Published in Molecular cancer therapeutics (01.01.2002)
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An Angiogenesis Inhibitor E7820 Shows Broad-Spectrum Tumor Growth Inhibition in a Xenograft Model
Semba, Taro, Funahashi, Yasuhiro, Ono, Naoto, Yamamoto, Yuji, Sugi, Naoko Hata, Asada, Makoto, Yoshimatsu, Kentaro, Wakabayashi, Toshiaki
Published in Clinical cancer research (15.02.2004)
Published in Clinical cancer research (15.02.2004)
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