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Published in Expert opinion on therapeutic targets (01.07.2008)
Published in Expert opinion on therapeutic targets (01.07.2008)
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Identification of CXCR3 receptor agonists in combinatorial small-molecule libraries
Stroke, Ilana L., Cole, Andrew G., Simhadri, Srilatha, Brescia, Marc-Raleigh, Desai, Madhuri, Zhang, Joan J., Merritt, J. Robert, Appell, Kenneth C., Henderson, Ian, Webb, Maria L.
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Published in Biochemical and biophysical research communications (13.10.2006)
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Novel Pyrrolidine Ureas as C−C Chemokine Receptor 1 (CCR1) Antagonists
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Published in Journal of medicinal chemistry (12.03.2009)
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Novel pyrrolidine heterocycles as CCR1 antagonists
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Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Synthesis and initial evaluation of novel, non-peptidic antagonists of the alpha(v)-integrins alpha(v)beta(3) and alpha(v)beta(5)
Letourneau, Jeffrey J, Liu, Jinqi, Ohlmeyer, Michael H J, Riviello, Chris, Rong, Yajing, Li, Hong, Appell, Kenneth C, Bansal, Shalini, Jacob, Biji, Wong, Angela, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
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2-Benzimidazolyl-9-(chroman-4-yl)-purinone derivatives as JAK3 inhibitors
Cole, Andrew G., Bohnstedt, Adolph C., Paradkar, Vidyadhar, Kingsbury, Celia, Quintero, Jorge G., Park, Haengsoon, Lu, Yingchun, You, Ming, Neagu, Irina, Diller, David J., Letourneau, Jeffrey J., Shao, Yuefei, James, Ray A., Riviello, Christopher M., Ho, Koc-Kan, Lin, Tsung H., Wang, Bojing, Appell, Kenneth C., Sills, Matthew, Quadros, Elizabeth, Kimble, Earl F., Ohlmeyer, Michael H.J., Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
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Identification and initial evaluation of 4- N-aryl-[1,4]diazepane ureas as potent CXCR3 antagonists
Cole, Andrew G., Stroke, Ilana L., Brescia, Marc-Raleigh, Simhadri, Srilatha, Zhang, Joan J., Hussain, Zahid, Snider, Michael, Haskell, Christopher, Ribeiro, Sofia, Appell, Kenneth C., Henderson, Ian, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Identification and characterization of small-molecule inhibitors of Tie2 kinase
Liu, Jinqi, Lin, Tsung H., Cole, Andrew G., Wen, Rong, Zhao, Lian, Brescia, Marc-Raleigh, Jacob, Biji, Hussain, Zahid, Appell, Kenneth C., Henderson, Ian, Webb, Maria L.
Published in FEBS letters (05.03.2008)
Published in FEBS letters (05.03.2008)
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Synthesis and initial evaluation of novel, non-peptidic antagonists of the αv-integrins αvβ3 and αvβ5
LETOUMEAU, Jeffrey J, JINQI LIU, WEBB, Maria L, OHLMEYER, Michael H. J, RIVIELLO, Chris, YAJING RONG, HONG LI, APPELL, Kenneth C, BANSAL, Shalini, JACOB, Biji, WONG, Angela
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
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Journal Article
Synthesis and initial evaluation of novel, non-peptidic antagonists of the α v-integrins α vβ 3 and α vβ 5
Letourneau, Jeffrey J., Liu, Jinqi, Ohlmeyer, Michael H.J., Riviello, Chris, Rong, Yajing, Li, Hong, Appell, Kenneth C., Bansal, Shalini, Jacob, Biji, Wong, Angela, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
Published in Bioorganic & medicinal chemistry letters (15.01.2009)
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Synthesis of (3,4-dimethoxyphenoxy)alkylamino acetamides as orexin-2 receptor antagonists
Cole, Andrew G., Stroke, Ilana L., Qin, Lan-Ying, Hussain, Zahid, Simhadri, Srilatha, Brescia, Marc-Raleigh, Waksmunski, Frank S., Strohl, Barbara, Tellew, John E., Williams, John P., Saunders, John, Appell, Kenneth C., Henderson, Ian, Webb, Maria L.
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists
Cole, Andrew G., Metzger, Axel, Brescia, Marc-Raleigh, Qin, Lan-Ying, Appell, Kenneth C., Brain, Christopher T., Hallett, Allan, Ganju, Pam, Denholm, Alastair A., Wareing, James R., Ritchie, Timothy J., Drake, Gillian M., Bevan, Stuart J., MacGloinn, Aisling, McBryde, Andrew, Patel, Viral, Oakley, Paul J., Nunez, Ximena, Gstach, Hubert, Schneider, Peter, Baldwin, John J., Dolle, Roland E., McDonald, Edward, Henderson, Ian
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Synthesis and substance P receptor binding activity of androstano[3,2-b]pyrimido[1,2-a]benzimidazoles
Venepalli, Bhaskar R, Aimone, Lisa D, Appell, Kenneth C, Bell, Malcolm R, Dority, John A, Goswami, Ramanuj, Hall, Patricia L, Kumar, Virendra, Lawrence, Kristine B
Published in Journal of medicinal chemistry (01.01.1992)
Published in Journal of medicinal chemistry (01.01.1992)
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2-(Aminomethyl)-benzamide-based glycine transporter type-2 inhibitors
Ho, Koc-Kan, Appell, Kenneth C., Baldwin, John J., Bohnstedt, Adolph C., Dong, Guizhen, Guo, Tao, Horlick, Robert, Islam, Khondaker R., Kultgen, Steven G., Masterson, Christopher M., McDonald, Edward, McMillan, Kirk, Morphy, J.Richard, Rankovic, Zoran, Sundaram, Hardy, Webb, Maria
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
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Chemokine Receptor−Ligand Interactions Measured Using Time-Resolved Fluorescence
Inglese, James, Samama, Philippe, Patel, Sanjay, Burbaum, Jonathan, Stroke, Ilana L, Appell, Kenneth C
Published in Biochemistry (Easton) (24.02.1998)
Published in Biochemistry (Easton) (24.02.1998)
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A Novel High-Throughput Screening Format to Identify Inhibitors of Secreted Acid Sphingomyelinase
Mintzer, Robert J., Appell, Kenneth C., Cole, Andrew, Johns, Anthony, Pagila, Rene, Polokoff, Mark A., Tabas, Ira, Snider, R. Michael, Meurer-Ogden, Janet A.
Published in Journal of biomolecular screening (01.04.2005)
Published in Journal of biomolecular screening (01.04.2005)
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