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An allosteric PRC2 inhibitor targeting the H3K27me3 binding pocket of EED
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Gonzalez-Sandoval, Adriana, Towbin, Benjamin D., Kalck, Veronique, Cabianca, Daphne S., Gaidatzis, Dimos, Hauer, Michael H., Geng, Liqing, Wang, Li, Yang, Teddy, Wang, Xinghao, Zhao, Kehao, Gasser, Susan M.
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Published in Proceedings of the National Academy of Sciences - PNAS (26.12.2012)
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Histone Methylation by PRC2 Is Inhibited by Active Chromatin Marks
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Multiplexable high-temperature stable and low-loss intrinsic Fabry-Perot in-fiber sensors through nanograting engineering
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Published in Nature communications (16.10.2015)
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High-Throughput-Methyl-Reading (HTMR) assay: a solution based on nucleotide methyl-binding proteins enables large-scale screening for DNA/RNA methyltransferases and demethylases
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Structure-Guided Design of EED Binders Allosterically Inhibiting the Epigenetic Polycomb Repressive Complex 2 (PRC2) Methyltransferase
Lingel, Andreas, Sendzik, Martin, Huang, Ying, Shultz, Michael D, Cantwell, John, Dillon, Michael P, Fu, Xingnian, Fuller, John, Gabriel, Tobias, Gu, Justin, Jiang, Xiangqing, Li, Ling, Liang, Fang, McKenna, Maureen, Qi, Wei, Rao, Weijun, Sheng, Xijun, Shu, Wei, Sutton, James, Taft, Benjamin, Wang, Long, Zeng, Jue, Zhang, Hailong, Zhang, Maya, Zhao, Kehao, Lindvall, Mika, Bussiere, Dirksen E
Published in Journal of medicinal chemistry (12.01.2017)
Published in Journal of medicinal chemistry (12.01.2017)
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Discovery and Molecular Basis of a Diverse Set of Polycomb Repressive Complex 2 Inhibitors Recognition by EED
Li, Ling, Zhang, Hailong, Zhang, Man, Zhao, Mengxi, Feng, Lijian, Luo, Xiao, Gao, Zhenting, Huang, Ying, Ardayfio, Ophelia, Zhang, Ji-Hu, Lin, Ying, Fan, Hong, Mi, Yuan, Li, Guobin, Liu, Lei, Feng, Leying, Luo, Fangjun, Teng, Lin, Qi, Wei, Ottl, Johannes, Lingel, Andreas, Bussiere, Dirksen E, Yu, Zhengtian, Atadja, Peter, Lu, Chris, Li, En, Gu, Justin, Zhao, Kehao
Published in PloS one (10.01.2017)
Published in PloS one (10.01.2017)
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Simulation Analysis of Mode Hopping Impacts on OFDR Sensing Performance
Wang, Qirui, Lalam, Nageswara, Zhao, Kehao, Zhong, Shuda, Zhang, Guangyin, Wright, Ruishu, Chen, Kevin P.
Published in Photonics (20.06.2024)
Published in Photonics (20.06.2024)
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NSD2 Is Recruited through Its PHD Domain to Oncogenic Gene Loci to Drive Multiple Myeloma
ZHENG HUANG, HAIPING WU, GU, Justin, MAN ZHANG, YANG, Teddy, KEHAO ZHAO, YANYAN YU, JINGQUAN DAI, WEI YI, SHAOLIAN ZHOU, QIAN LI, JING WU, SHANNON CHUAI, JUN LIU, XU WU, CHAN, Homan, LU, Chris, ATADJA, Peter, EN LI, YAN WANG, MIN HU, FIONA XU, FENG YAN, ENGLUND, Nathan, ZHAOFU WANG, HAILONG ZHANG, MING FANG, YOUZHEN WANG
Published in Cancer research (Chicago, Ill.) (15.10.2013)
Published in Cancer research (Chicago, Ill.) (15.10.2013)
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Split luciferase-based biosensors for characterizing EED binders
Li, Ling, Feng, Lijian, Shi, Minlong, Zeng, Jue, Chen, Zijun, Zhong, Li, Huang, Li, Guo, Weihui, Huang, Ying, Qi, Wei, Lu, Chris, Li, En, Zhao, Kehao, Gu, Justin
Published in Analytical biochemistry (01.04.2017)
Published in Analytical biochemistry (01.04.2017)
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Structural Basis for Nicotinamide Cleavage and ADP-Ribose Transfer by NAD+-Dependent Sir2 Histone/Protein Deacetylases
Zhao, Kehao, Harshaw, Robyn, Chai, Xiaomei, Marmorstein, Ronen, Petsko, Gregory A.
Published in Proceedings of the National Academy of Sciences - PNAS (08.06.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (08.06.2004)
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Structure and Substrate Binding Properties of cobB, a Sir2 Homolog Protein Deacetylase from Escherichia coli
Zhao, Kehao, Chai, Xiaomei, Marmorstein, Ronen
Published in Journal of molecular biology (26.03.2004)
Published in Journal of molecular biology (26.03.2004)
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Structural Basis for Nicotinamide Inhibition and Base Exchange in Sir2 Enzymes
Sanders, Brandi D., Zhao, Kehao, Slama, James T., Marmorstein, Ronen
Published in Molecular cell (09.02.2007)
Published in Molecular cell (09.02.2007)
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Discovery of Small-Molecule Antagonists of the H3K9me3 Binding to UHRF1 Tandem Tudor Domain
Senisterra, Guillermo, Zhu, Hugh Y., Luo, Xiao, Zhang, Hailong, Xun, Guoliang, Lu, Chunliang, Xiao, Wen, Hajian, Taraneh, Loppnau, Peter, Chau, Irene, Li, Fengling, Allali-Hassani, Abdellah, Atadja, Peter, Oyang, Counde, Li, En, Brown, Peter J., Arrowsmith, Cheryl H., Zhao, Kehao, Yu, Zhengtian, Vedadi, Masoud
Published in SLAS discovery (01.10.2018)
Published in SLAS discovery (01.10.2018)
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