Search Results - "KAZUTA, Yuji" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of E2730, a novel selective uncompetitive GAT1 inhibitor, as a candidate for anti‐seizure medication

Discovery of E2730, a novel selective uncompetitive GAT1 inhibitor, as a candidate for anti‐seizure medication

by Fukushima, Kazuyuki, Higashiyama, Hiroyuki, Kazuta, Yuji, Hashimoto, Keisuke, Watanabe, Naoto, Furuya, Yoshiaki, Ito, Yoshimasa, Wu, Ting, Kosasa, Takashi, Talos, Delia M., Song, Yeri, Roberts, Nicholas S., Jensen, Frances E., Hanada, Takahisa, Ido, Katsutoshi
Published in Epilepsia open (01.09.2023)

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Journal Article

Cyclopropane-Based Conformational Restriction of Histamine. (1S,2S)-2-(2-Aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a Highly Selective Agonist for the Histamine H3 Receptor, Having a cis-Cyclopropane Structure

Cyclopropane-Based Conformational Restriction of Histamine. (1S,2S)-2-(2-Aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a Highly Selective Agonist for the Histamine H3 Receptor, Having a cis-Cyclopropane Structure

by Kazuta, Yuji, Hirano, Kazufumi, Natsume, Kentaro, Yamada, Shizuo, Kimura, Ryohei, Matsumoto, Shun-ichiro, Furuichi, Kiyoshi, Matsuda, Akira, Shuto, Satoshi
Published in Journal of medicinal chemistry (08.05.2003)

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Construction of a cis-Cyclopropane via Reductive Radical Decarboxylation. Enantioselective Synthesis of cis- and trans-1-Arylpiperazyl-2-phenylcyclopropanes Designed as Antidopaminergic Agents

Construction of a cis-Cyclopropane via Reductive Radical Decarboxylation. Enantioselective Synthesis of cis- and trans-1-Arylpiperazyl-2-phenylcyclopropanes Designed as Antidopaminergic Agents

by Yamaguchi, Kazuya, Kazuta, Yuji, Abe, Hiroshi, Matsuda, Akira, Shuto, Satoshi
Published in Journal of organic chemistry (28.11.2003)

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Synthesis of derivatives of (1 S,2 R)-1-phenyl-2-[( S)-1-aminopropyl] -N,N-diethylcyclopropanecarboxamide (PPDC) modified at the 1-aromatic moiety as novel NMDA receptor antagonists: the aromatic group is essential for the activity

Synthesis of derivatives of (1 S,2 R)-1-phenyl-2-[( S)-1-aminopropyl] -N,N-diethylcyclopropanecarboxamide (PPDC) modified at the 1-aromatic moiety as novel NMDA receptor antagonists: the aromatic group is essential for the activity

by Kazuta, Yuji, Tsujita, Ryuichi, Yamashita, Kanako, Uchino, Shigeo, Kohsaka, Shinichi, Matsuda, Akira, Shuto, Satoshi
Published in Bioorganic & medicinal chemistry (01.12.2002)

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THERAPEUTIC AGENT FOR EPILEPSY

THERAPEUTIC AGENT FOR EPILEPSY

by KAZUTA YUJI, HIGASHIYAMA HIROYUKI, WATANABE NAOTO, HASHIMOTO KEISUKE, FUKUSHIMA KAZUYUKI
Year of Publication 29.02.2024

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Patent

Conformational Analysis of the NMDA Receptor Antagonist (1S,2R)-1-Phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide (PPDC) Designed by a Novel Conformational Restriction Method Based on the Structural Feature of Cyclopropane Ring

Conformational Analysis of the NMDA Receptor Antagonist (1S,2R)-1-Phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide (PPDC) Designed by a Novel Conformational Restriction Method Based on the Structural Feature of Cyclopropane Ring

by Ono, Sizuka, Ogawa, Kiyoshi, Yamashita, Kanako, Yamamoto, Tamotsu, Kazuta, Yuji, Matsuda, Akira, Shuto, Satoshi
Published in Chemical & pharmaceutical bulletin (01.07.2002)

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Journal Article

Silinanyl Rhodamines and Silinanyl Fluoresceins for Super-Resolution Microscopy

Silinanyl Rhodamines and Silinanyl Fluoresceins for Super-Resolution Microscopy

by Hara, Daiki, Uno, Shin-nosuke, Motoki, Takafumi, Kazuta, Yuji, Norimine, Yoshihiko, Suganuma, Masatoshi, Fujiyama, Shingo, Shimaoka, Yuki, Yamashita, Kazuto, Okada, Masaya, Nishikawa, Youichi, Amino, Hiroyuki, Iwanaga, Shigeki
Published in The journal of physical chemistry. B (12.08.2021)

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Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists

Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists

by Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.11.2014)

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Journal Article

THERAPEUTIC AGENT FOR EPILEPSY

THERAPEUTIC AGENT FOR EPILEPSY

by HIGASHIYAMA Hiroyuki, WATANABE Naoto, FUKUSHIMA Kazuyuki, KAZUTA Yuji, HASHIMOTO Keisuke, FURUYA Yoshiaki
Year of Publication 02.06.2022

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Patent

Stereochemical Diversity-Oriented Conformational Restriction Strategy. Development of Potent Histamine H3 and/or H4 Receptor Antagonists with an Imidazolylcyclopropane Structure

Stereochemical Diversity-Oriented Conformational Restriction Strategy. Development of Potent Histamine H3 and/or H4 Receptor Antagonists with an Imidazolylcyclopropane Structure

by Watanabe, Mizuki, Kazuta, Yuji, Hayashi, Hideki, Yamada, Shizuo, Matsuda, Akira, Shuto, Satoshi
Published in Journal of medicinal chemistry (07.09.2006)

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Journal Article

Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H-3 and/or H-4 receptor antagonists with an imidazolylcyclopropane structure

Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H-3 and/or H-4 receptor antagonists with an imidazolylcyclopropane structure

by Watanabe, Mizuki, Kazuta, Yuji, Hayashi, Hideki, Yamada, Shizuo, Matsuda, Akira, Shuto, Satoshi
Published in Journal of medicinal chemistry (07.09.2006)

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Journal Article

THERAPEUTIC AND/OR PREVENTIVE AGENT COMPRISING 1-INDANSULFAMIDE DERIVATIVE FOR PAIN

THERAPEUTIC AND/OR PREVENTIVE AGENT COMPRISING 1-INDANSULFAMIDE DERIVATIVE FOR PAIN

by KAZUTA YUJI, HIGASHIYAMA HIROYUKI, HASHIMOTO KEISUKE
Year of Publication 09.09.2016

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Patent

Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists” [Bioorg. Med. Chem. 22 (2014) 6071–6088]

Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists” [Bioorg. Med. Chem. 22 (2014) 6071–6088]

by Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.07.2015)

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Journal Article

FLUORESCENT DYE AND USE THEREOF

FLUORESCENT DYE AND USE THEREOF

by NORIMINE YOSHIHIKO, KAZUTA YUJI, FUJIYAMA SHINGO, HARA DAIKI, IWANAGA SHIGEKI, NISHIKAWA YOICHI, AMINO HIROYUKI, YAMASHITA KAZUTO, MOTOKI TAKASHI, SUGANUMA MASATOSHI, OKADA MASAYA
Year of Publication 30.08.2021

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Patent

THERAPEUTIC AND/OR PREVENTIVE AGENT COMPRISING 1-INDANSULFAMIDE DERIVATIVE FOR PAIN

THERAPEUTIC AND/OR PREVENTIVE AGENT COMPRISING 1-INDANSULFAMIDE DERIVATIVE FOR PAIN

by KAZUTA YUJI, HIGASHIYAMA HIROYUKI, HASHIMOTO KEISUKE
Year of Publication 25.06.2015

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Patent

Synthesis of (1S,2R)-1-phenyl-2-[(S)-1-aminoalkyl]-N,N-diethylcyclopropanecarboxamides as novel NMDA receptor antagonists having a unique NMDA receptor subtype selectivity

Synthesis of (1S,2R)-1-phenyl-2-[(S)-1-aminoalkyl]-N,N-diethylcyclopropanecarboxamides as novel NMDA receptor antagonists having a unique NMDA receptor subtype selectivity

by Kazuta, Y, Tsujita, R, Uchino, S, Kamiyama, N, Mochizuki, D, Yamashita, K, Ohmori, Y, Yamashita, A, Yamamoto, T, Kohsaka, S, Matsuda, A, Shuto, S
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (26.04.2002)

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Journal Article

Synthesis of 1-arylpiperazyl-2-phenylcyclopropanes designed as antidopaminergic agents: Cyclopropane-based conformationally restricted analogs of haloperidol

Synthesis of 1-arylpiperazyl-2-phenylcyclopropanes designed as antidopaminergic agents: Cyclopropane-based conformationally restricted analogs of haloperidol

by Yamaguchi, Kazuya, Kazuta, Yuji, Hirano, Kazufumi, Yamada, Shizuo, Matsuda, Akira, Shuto, Satoshi
Published in Bioorganic & medicinal chemistry (01.10.2008)

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Development of Versatile cis- and trans-Dicarbon-Substituted Chiral Cyclopropane Units: Synthesis of (1S,2R)- and (1R,2R)-2-Aminomethyl-1-(1H-imidazol-4-yl)cyclopropanes and Their Enantiomers as Conformationally Restricted Analogues of Histamine

Development of Versatile cis- and trans-Dicarbon-Substituted Chiral Cyclopropane Units: Synthesis of (1S,2R)- and (1R,2R)-2-Aminomethyl-1-(1H-imidazol-4-yl)cyclopropanes and Their Enantiomers as Conformationally Restricted Analogues of Histamine

by Kazuta, Yuji, Matsuda, Akira, Shuto, Satoshi
Published in Journal of organic chemistry (08.03.2002)

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Journal Article

Cyclopropane-based conformational restriction of histamine. (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a highly selective agonist for the histamine H-3 receptor, having a cis-cyclopropane structure

Cyclopropane-based conformational restriction of histamine. (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a highly selective agonist for the histamine H-3 receptor, having a cis-cyclopropane structure

by Kazuta, Y, Hirano, K, Natsume, K, Yamada, S, Kimura, R, Matsumoto, SI, Furuichi, K, Matsuda, A, Shuto, S
Published in Journal of medicinal chemistry (08.05.2003)

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A Systematic Study of the Hydride Reduction of Cyclopropyl Ketones with Structurally Simplified Substrates. Highly Stereoselective Reductions of Trans-Substituted Cyclopropyl Ketones via the Bisected s-Cis Conformation

A Systematic Study of the Hydride Reduction of Cyclopropyl Ketones with Structurally Simplified Substrates. Highly Stereoselective Reductions of Trans-Substituted Cyclopropyl Ketones via the Bisected s-Cis Conformation

by Kazuta, Yuji, Abe, Hiroshi, Yamamoto, Tamotsu, Matsuda, Akira, Shuto, Satoshi
Published in Journal of organic chemistry (02.05.2003)

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