Potential SARS-CoV-2 RdRp inhibitors of cytidine derivatives: Molecular docking, molecular dynamic simulations, ADMET, and POM analyses for the identification of pharmacophore sites
M A Kawsar, Sarkar, Hosen, Mohammed A, Ahmad, Sajjad, El Bakri, Youness, Laaroussi, Hamid, Ben Hadda, Taibi, Almalki, Faisal A, Ozeki, Yasuhiro, Goumri-Said, Souraya
Published in PloS one (28.11.2022)
Published in PloS one (28.11.2022)
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Marine-Derived Compounds as Potential Inhibitors of Hsp90 for Anticancer and Antimicrobial Drug Development: A Comprehensive In Silico Study
Ouassaf, Mebarka, Bourougaa, Lotfi, Al-Mijalli, Samiah Hamad, Abdallah, Emad M, Bhat, Ajmal R, A Kawsar, Sarkar M
Published in Molecules (Basel, Switzerland) (01.12.2023)
Published in Molecules (Basel, Switzerland) (01.12.2023)
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Efficient Antibacterial/Antifungal Activities: Synthesis, Molecular Docking, Molecular Dynamics, Pharmacokinetic, and Binding Free Energy of Galactopyranoside Derivatives
Ahmmed, Faez, Islam, Anis Ul, Mukhrish, Yousef E, Bakri, Youness El, Ahmad, Sajjad, Ozeki, Yasuhiro, Kawsar, Sarkar M A
Published in Molecules (Basel, Switzerland) (26.12.2022)
Published in Molecules (Basel, Switzerland) (26.12.2022)
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Establishing the Role of Iridoids as Potential Kirsten Rat Sarcoma Viral Oncogene Homolog G12C Inhibitors Using Molecular Docking; Molecular Docking Simulation; Molecular Mechanics Poisson-Boltzmann Surface Area; Frontier Molecular Orbital Theory; Molecular Electrostatic Potential; and Absorption, Distribution, Metabolism, Excretion, and Toxicity Analysis
Alamri, Mubarak A, Alawam, Abdullah S, Alshahrani, Mohammed Merae, Kawsar, Sarkar M A, Prinsa, Saha, Supriyo
Published in Molecules (Basel, Switzerland) (28.06.2023)
Published in Molecules (Basel, Switzerland) (28.06.2023)
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Exploring Cinnamoyl-Substituted Mannopyranosides: Synthesis, Evaluation of Antimicrobial Properties, and Molecular Docking Studies Targeting H5N1 Influenza A Virus
Akter, Sabina, Alhatlani, Bader Y, Abdallah, Emad M, Saha, Supriyo, Ferdous, Jannatul, Hossain, Md Emdad, Ali, Ferdausi, Kawsar, Sarkar M A
Published in Molecules (Basel, Switzerland) (01.12.2023)
Published in Molecules (Basel, Switzerland) (01.12.2023)
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Layer‐by‐layer preparation of electromagnetic NH2‐SiO2/polypyrrole/Ni nanocomposites, characterization and their electrochemical properties
Ali, M Sagor, Rahman, M Mahabur, Minami, Hideto, Hossain, M Kawsar, Rahman, M Abdur, Gafur, M Abdul, Ahmad, Hasan
Published in Polymer international (01.04.2023)
Published in Polymer international (01.04.2023)
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Pharmacoinformatics and Breed-Based De Novo Hybridization Studies to Develop New Neuraminidase Inhibitors as Potential Anti-Influenza Agents
Lotfi, Bourougaa, Mebarka, Ouassaf, Alhatlani, Bader Y, Abdallah, Emad M, Kawsar, Sarkar M. A
Published in Molecules (Basel, Switzerland) (01.09.2023)
Published in Molecules (Basel, Switzerland) (01.09.2023)
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Diverse Localization Patterns of an R-Type Lectin in Marine Annelids
Kawsar, Sarkar M. Abe, Hasan, Imtiaj, Rajia, Sultana, Koide, Yasuhiro, Fujii, Yuki, Hayashi, Ryuhei, Yamada, Masao, Ozeki, Yasuhiro
Published in Molecules (Basel, Switzerland) (07.08.2021)
Published in Molecules (Basel, Switzerland) (07.08.2021)
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Methyl β-D-galactopyranoside esters as potential inhibitors for SARS-CoV-2 protease enzyme: synthesis, antimicrobial, PASS, molecular docking, molecular dynamics simulations and quantum computations
Amin, Md R., Yasmin, Farhana, Dey, Sujan, Mahmud, Shafi, Saleh, Md A., Emran, Talha B., Hasan, Imtiaj, Rajia, Sultana, Ogawa, Yukiko, Fujii, Yuki, Yamada, Masao, Ozeki, Yasuhiro, Kawsar, Sarkar M. A.
Published in Glycoconjugate journal (01.04.2022)
Published in Glycoconjugate journal (01.04.2022)
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Design, Synthesis, In Silico and POM Studies for the Identification of the Pharmacophore Sites of Benzylidene Derivatives
Hosen, Mohammad I, Mukhrish, Yousef E, Jawhari, Ahmed Hussain, Celik, Ismail, Erol, Meryem, Abdallah, Emad M, Al-Ghorbani, Mohammed, Baashen, Mohammed, Almalki, Faisal A, Laaroussi, Hamid, Hadda, Taibi Ben, Kawsar, Sarkar M A
Published in Molecules (Basel, Switzerland) (13.03.2023)
Published in Molecules (Basel, Switzerland) (13.03.2023)
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Systematic challenges and opportunities in insect monitoring: a Global South perspective
Sánchez Herrera, Melissa, Forero, Dimitri, Calor, Adolfo Ricardo, Romero, Gustavo Q, Riyaz, Muzafar, Callisto, Marcos, de Oliveira Roque, Fabio, Elme-Tumpay, Araseli, Khan, M Kawsar, Justino de Faria, Ana Paula, Pires, Mateus Marques, Silva de Azevêdo, Carlos Augusto, Juen, Leandro, Zakka, Usman, Samaila, Akeweta Emmanuel, Hussaini, Suwaiba, Kemabonta, Kehinde, Guillermo-Ferreira, Rhainer, Ríos-Touma, Blanca, Maharaj, Gyanpriya
Published in Philosophical transactions of the Royal Society of London. Series B. Biological sciences (24.06.2024)
Published in Philosophical transactions of the Royal Society of London. Series B. Biological sciences (24.06.2024)
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Multifunctional Cell Regulation Activities of the Mussel Lectin SeviL: Induction of Macrophage Polarization toward the M1 Functional Phenotype
Fujii, Yuki, Kamata, Kenichi, Gerdol, Marco, Hasan, Imtiaj, Rajia, Sultana, Kawsar, Sarkar M A, Padma, Somrita, Chatterjee, Bishnu Pada, Ohkawa, Mayuka, Ishiwata, Ryuya, Yoshimoto, Suzuna, Yamada, Masao, Matsuzaki, Namiho, Yamamoto, Keita, Niimi, Yuka, Miyanishi, Nobumitsu, Konno, Masamitsu, Pallavicini, Alberto, Kawasaki, Tatsuya, Ogawa, Yukiko, Ozeki, Yasuhiro, Fujita, Hideaki
Published in Marine drugs (01.06.2024)
Published in Marine drugs (01.06.2024)
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Impact of mesoporous SiO2 support for Ni/polypyrrole nanocomposite particles on their capacitive performance
M Sagor Ali, Rahman, M Mahabur, M Kawsar Hossain, Minami, Hideto, Rahman, M Mahbubor, Hoque, S Manjura, Alam, M Ashraful, Ahmad, Hasan
Published in New journal of chemistry (2022)
Published in New journal of chemistry (2022)
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Recent Progress in Synthesis, POM Analyses and SAR of Coumarin-Hybrids as Potential Anti-HIV Agents—A Mini Review
Suleiman, Mustapha, Almalki, Faisal A, Ben Hadda, Taibi, Kawsar, Sarkar M. A, Chander, Subhash, Murugesan, Sankaranarayanan, Bhat, Ajmal R, Bogoyavlenskiy, Andrey, Jamalis, Joazaizulfazli
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2023)
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Efficient Synthesis, Structural Characterization, Antibacterial Assessment, ADME-Tox Analysis, Molecular Docking and Molecular Dynamics Simulations of New Functionalized Isoxazoles
Arzine, Aziz, Hadni, Hanine, Boujdi, Khalid, Chebbac, Khalid, Barghady, Najoua, Rhazi, Yassine, Chalkha, Mohammed, Nakkabi, Asmae, Chkirate, Karim, Mague, Joel T, Kawsar, Sarkar M A, Al Houari, Ghali, M Alanazi, Mohammed, El Yazidi, Mohamed
Published in Molecules (Basel, Switzerland) (17.07.2024)
Published in Molecules (Basel, Switzerland) (17.07.2024)
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Uridine Derivatives: Synthesis, Biological Evaluation, and In Silico Studies as Antimicrobial and Anticancer Agents
Munia, Nasrin S, Alanazi, Mohammed M, El Bakri, Youness, Alanazi, Ashwag S, Mukhrish, Yousef E, Hasan, Imtiaj, Kawsar, Sarkar M A
Published in Medicina (Kaunas, Lithuania) (01.06.2023)
Published in Medicina (Kaunas, Lithuania) (01.06.2023)
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Galactoside-Based Molecule Enhanced Antimicrobial Activity through Acyl Moiety Incorporation: Synthesis and In Silico Exploration for Therapeutic Target
Ahmmed, Faez, Al-Mijalli, Samiah Hamad, Abdallah, Emad M, Eissa, Ibrahim H, Ali, Ferdausi, Bhat, Ajmal R, Jamalis, Joazaizulfazli, Ben Hadda, Taibi, Kawsar, Sarkar M A
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.07.2023)
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New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors
Messore, Antonella, Malune, Paolo, Patacchini, Elisa, Madia, Valentina Noemi, Ialongo, Davide, Arpacioglu, Merve, Albano, Aurora, Ruggieri, Giuseppe, Saccoliti, Francesco, Scipione, Luigi, Tramontano, Enzo, Canton, Serena, Corona, Angela, Scognamiglio, Sante, Paulis, Annalaura, Suleiman, Mustapha, Al-Maqtari, Helmi Mohammed, Abid, Fatma Mohamed A, Kawsar, Sarkar M A, Sankaranarayanan, Murugesan, Di Santo, Roberto, Esposito, Francesca, Costi, Roberta
Published in Pharmaceuticals (Basel, Switzerland) (01.05.2024)
Published in Pharmaceuticals (Basel, Switzerland) (01.05.2024)
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