A general alkyl-alkyl cross-coupling enabled by redox-active esters and alkylzinc reagents
Qin, Tian, Cornella, Josep, Li, Chao, Malins, Lara R., Edwards, Jacob T., Kawamura, Shuhei, Maxwell, Brad D., Eastgate, Martin D., Baran, Phil S.
Published in Science (American Association for the Advancement of Science) (13.05.2016)
Published in Science (American Association for the Advancement of Science) (13.05.2016)
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Journal Article
Practical Ni-Catalyzed Aryl–Alkyl Cross-Coupling of Secondary Redox-Active Esters
Cornella, Josep, Edwards, Jacob T, Qin, Tian, Kawamura, Shuhei, Wang, Jie, Pan, Chung-Mao, Gianatassio, Ryan, Schmidt, Michael, Eastgate, Martin D, Baran, Phil S
Published in Journal of the American Chemical Society (24.02.2016)
Published in Journal of the American Chemical Society (24.02.2016)
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Journal Article
Influence of a plasma-treated nutrient solution containing 2,4-dichlorobenzoic acid on the growth of cucumber in a hydroponic system
Takahashi, Katsuyuki, Kawamura, Shuhei, Takada, Ryosuke, Takaki, Koichi, Satta, Naoya, Fujio, Takuya
Published in Journal of applied physics (14.04.2021)
Published in Journal of applied physics (14.04.2021)
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Journal Article
Structurally Novel Highly Potent Proteasome Inhibitors Created by the Structure-Based Hybridization of Nonpeptidic Belactosin Derivatives and Peptide Boronates
Kawamura, Shuhei, Unno, Yuka, Asai, Akira, Arisawa, Mitsuhiro, Shuto, Satoshi
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Journal Article
Potent Proteasome Inhibitors Derived from the Unnatural cis-Cyclopropane Isomer of Belactosin A: Synthesis, Biological Activity, and Mode of Action
Kawamura, Shuhei, Unno, Yuka, List, Anja, Mizuno, Akirai, Tanaka, Motohiro, Sasaki, Takuma, Arisawa, Mitsuhiro, Asai, Akira, Groll, Michael, Shuto, Satoshi
Published in Journal of medicinal chemistry (09.05.2013)
Published in Journal of medicinal chemistry (09.05.2013)
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Journal Article
Modeling and System Integration for a Thin Pneumatic Rubber 3-DOF Actuator
Kawamura, Shuhei, Sudani, Mizuki, Deng, Mingcong, Noge, Yuichi, Wakimoto, Shuichi
Published in Actuators (01.06.2019)
Published in Actuators (01.06.2019)
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Journal Article
Investigation of the Noncovalent Binding Mode of Covalent Proteasome Inhibitors around the Transition State by Combined Use of Cyclopropylic Strain-Based Conformational Restriction and Computational Modeling
Kawamura, Shuhei, Unno, Yuka, Tanaka, Motohiro, Sasaki, Takuma, Yamano, Akihito, Hirokawa, Takatsugu, Kameda, Tomoshi, Asai, Akira, Arisawa, Mitsuhiro, Shuto, Satoshi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Journal Article
Cyclopropane-based conformational restriction of GABA by a stereochemical diversity-oriented strategy: Identification of an efficient lead for potent inhibitors of GABA transports
Nakada, Kazuaki, Yoshikawa, Mamie, Ide, Soichiro, Suemasa, Akihiro, Kawamura, Shuhei, Kobayashi, Takaaki, Masuda, Eiji, Ito, Yoshihiko, Hayakawa, Wataru, Katayama, Takahiro, Yamada, Shizuo, Arisawa, Mitsuhiro, Minami, Masabumi, Shuto, Satoshi
Published in Bioorganic & medicinal chemistry (01.09.2013)
Published in Bioorganic & medicinal chemistry (01.09.2013)
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Journal Article
Simple Sulfinate Synthesis Enables CH Trifluoromethylcyclopropanation
Gianatassio, Ryan, Kawamura, Shuhei, Eprile, Cecil L, Foo, Klement, Ge, Jason, Burns, Aaron C., Collins, Michael R., Baran, Phil S.
Published in Angewandte Chemie (08.09.2014)
Published in Angewandte Chemie (08.09.2014)
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Journal Article
Synthesis and pharmacological evaluation of nucleoside prodrugs designed to target siderophore biosynthesis in Mycobacterium tuberculosis
Dawadi, Surendra, Kawamura, Shuhei, Rubenstein, Anja, Remmel, Rory, Aldrich, Courtney C.
Published in Bioorganic & medicinal chemistry (15.03.2016)
Published in Bioorganic & medicinal chemistry (15.03.2016)
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Journal Article
Design and synthesis of unprecedented 9- and 10-membered cyclonucleosides with PRMT5 inhibitory activity
Kawamura, Shuhei, Palte, Rachel L., Kim, Hai-Young, Saurí, Josep, Sondey, Christopher, Mansueto, My S., Altman, Michael D., Machacek, Michelle R.
Published in Bioorganic & medicinal chemistry (15.07.2022)
Published in Bioorganic & medicinal chemistry (15.07.2022)
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Journal Article
Ligand–Phospholipid Conjugation: A Versatile Strategy for Developing Long-Acting Ligands That Bind to Membrane Proteins by Restricting the Subcellular Localization of the Ligand
Kawamura, Shuhei, Ito, Yoshihiko, Hirokawa, Takatsugu, Hikiyama, Eriko, Yamada, Shizuo, Shuto, Satoshi
Published in Journal of medicinal chemistry (10.05.2018)
Published in Journal of medicinal chemistry (10.05.2018)
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Journal Article
Development of a new class of proteasome inhibitors with an epoxyketone warhead: Rational hybridization of non-peptidic belactosin derivatives and peptide epoxyketones
Kawamura, Shuhei, Unno, Yuka, Asai, Akira, Arisawa, Mitsuhiro, Shuto, Satoshi
Published in Bioorganic & medicinal chemistry (15.06.2014)
Published in Bioorganic & medicinal chemistry (15.06.2014)
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Journal Article
Rational hopping of a peptidic scaffold into non-peptidic scaffolds: structurally novel potent proteasome inhibitors derived from a natural product, belactosin A
Kawamura, Shuhei, Unno, Yuka, Hirokawa, Takatsugu, Asai, Akira, Arisawa, Mitsuhiro, Shuto, Satoshi
Published in Chemical communications (Cambridge, England) (07.03.2014)
Published in Chemical communications (Cambridge, England) (07.03.2014)
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Journal Article
The Discovery of Two Novel Classes of 5,5-Bicyclic Nucleoside-Derived PRMT5 Inhibitors for the Treatment of Cancer
Quiroz, Ryan V, Reutershan, Michael H, Schneider, Sebastian E, Sloman, David, Lacey, Brian M, Swalm, Brooke M, Yeung, Charles S, Gibeau, Craig, Spellman, Daniel S, Rankic, Danica A, Chen, Dapeng, Witter, David, Linn, Doug, Munsell, Erik, Feng, Guo, Xu, Haiyan, Hughes, Jonathan M. E, Lim, Jongwon, Saurí, Josep, Geddes, Kristin, Wan, Murray, Mansueto, My Sam, Follmer, Nicole E, Fier, Patrick S, Siliphaivanh, Phieng, Daublain, Pierre, Palte, Rachel L, Hayes, Robert P, Lee, Sandra, Kawamura, Shuhei, Silverman, Steven, Sanyal, Sulagna, Henderson, Timothy J, Ye, Yingchun, Gao, Yuanwei, Nicholson, Benjamin, Machacek, Michelle R
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Journal Article
Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5)
Palte, Rachel L, Schneider, Sebastian E, Altman, Michael D, Hayes, Robert P, Kawamura, Shuhei, Lacey, Brian M, Mansueto, My Sam, Reutershan, Michael, Siliphaivanh, Phieng, Sondey, Christopher, Xu, Haiyan, Xu, Zangwei, Ye, Yingchun, Machacek, Michelle R
Published in ACS medicinal chemistry letters (10.09.2020)
Published in ACS medicinal chemistry letters (10.09.2020)
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Journal Article