Design, Synthesis, and Structure–Activity Relationships Study of N-Pyrimidyl/Pyridyl-2-thiazolamine Analogues as Novel Positive Allosteric Modulators of M3 Muscarinic Acetylcholine Receptor
Tanaka, Hiroaki, Akaiwa, Michinori, Negoro, Kenji, Kawaminami, Eiji, Mihara, Hisashi, Fuji, Hideyoshi, Okimoto, Risa, Ino, Katsutoshi, Ishizu, Kenichiro, Takahashi, Taisuke
Published in Chemical & pharmaceutical bulletin (01.04.2021)
Published in Chemical & pharmaceutical bulletin (01.04.2021)
Get full text
Journal Article
Design, Synthesis, and Structure-Activity Relationships Study of N-Pyrimidyl/Pyridyl-2-thiazolamine Analogues as Novel Positive Allosteric Modulators of M3 Muscarinic Acetylcholine Receptor
Hiroaki Tanaka, Michinori Akaiwa, Kenji Negoro, Eiji Kawaminami, Hisashi Mihara, Hideyoshi Fuji, Risa Okimoto, Katsutoshi Ino, Kenichiro Ishizu, Taisuke Takahashi
Published in Chemical and Pharmaceutical Bulletin (01.04.2021)
Get full text
Published in Chemical and Pharmaceutical Bulletin (01.04.2021)
Journal Article
Design, Synthesis, and Structure-Activity Relationships Study of N-Pyrimidyl/Pyridyl-2-thiazolamine Analogues as Novel Positive Allosteric Modulators of M-3 Muscarinic Acetylcholine Receptor
Tanaka, Hiroaki, Akaiwa, Michinori, Negoro, Kenji, Kawaminami, Eiji, Mihara, Hisashi, Fuji, Hideyoshi, Okimoto, Risa, Ino, Katsutoshi, Ishizu, Kenichiro, Takahashi, Taisuke
Published in Chemical & pharmaceutical bulletin (01.04.2021)
Published in Chemical & pharmaceutical bulletin (01.04.2021)
Get full text
Journal Article
Effect of ASP6432, a Novel Type 1 Lysophosphatidic Acid Receptor Antagonist, on Urethral Function and Prostate Cell Proliferation
Sakamoto, Kazuyuki, Noguchi, Yukiko, Ueshima, Koji, Yamakuni, Hisashi, Ohtake, Akiyoshi, Sato, Shuichi, Ishizu, Kenichiro, Hosogai, Naomi, Kawaminami, Eiji, Takeda, Masahiro, Masuda, Noriyuki
Published in The Journal of pharmacology and experimental therapeutics (01.08.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2018)
Get full text
Journal Article
Novel Malonamide Derivatives as αvβ3 Antagonists. Syntheses and Evaluation of 3-(3-Indolin-1-yl-3-oxopropanoyl)aminopropanoic Acids on Vitronectin Interaction with αvβ3
NAGASHIMA, Shinya, AKAMATSU, Seijiro, KAWAMINAMI, Eiji, KAWAZOE, Souichirou, OGAMI, Tetsuro, MATSUMOTO, Yuzo, OKADA, Minoru, SUZUKI, Ken-Ichi, TSUKAMOTO, Shin-Ichi
Published in Chemical & pharmaceutical bulletin (2001)
Published in Chemical & pharmaceutical bulletin (2001)
Get full text
Journal Article
HETEROCYCLIC COMPOUND FOR INDUCING DEGRADATION OF G12V MUTANT KRAS PROTEIN
IMAIZUMI, Tomoyoshi, KAWAMINAMI, Eiji, MORIKAWA, Takahiro, KURAMOTO, Kazuyuki, IMADA, Sunao, KOGANEMARU, Yohei, OKUMURA, Mitsuaki, HAMAGUCHI, Hisao, YOSHINARI, Tomohiro, NISHIZONO, Yoshihiro
Year of Publication 15.02.2024
Get full text
Year of Publication 15.02.2024
Patent
HETEROCYCLIC COMPOUND FOR INDUCING DEGRADATION OF MUTANT KRAS PROTEIN
FUJIWARA, Yuta, MORIKAWA, Takahiro, KURAMOTO, Kazuyuki, IMADA, Sunao, HAMAGUCHI, Hisao, NISHIZONO, Yoshihiro, ISHIOKA, Hiroki, IMAIZUMI, Tomoyoshi, KAWAMINAMI, Eiji, HONJO, Eriko, KOGANEMARU, Yohei, OKUMURA, Mitsuaki, YOSHINARI, Tomohiro
Year of Publication 08.02.2024
Get full text
Year of Publication 08.02.2024
Patent
HETEROCYCLIC COMPOUND THAT ACTS ON G12D MUTANT KRAS PROTEIN
MORIKAWA, Takahiro, KURAMOTO, Kazuyuki, WATANABE, Hideyuki, HAMAGUCHI, Hisao, ISHIOKA, Hiroki, KAWAMINAMI, Eiji, KAWAGUCHI, Kenichi, IMAIZUMI, Tomoyoshi, INAMURA, Kohei, INAMI, Hiroshi, TAKAHASHI, Fumie, KAMIKUBO, Takashi, NAGASHIMA, Takeyuki, YOSHINARI, Tomohiro
Year of Publication 25.01.2024
Get full text
Year of Publication 25.01.2024
Patent
Studies on Aromatase Inhibitors. I. Synthesis and Biological Evaluation of 4-Amino-4H-1, 2, 4-triazole Derivatives
OKADA, Minoru, YODEN, Toru, KAWAMINAMI, Eiji, SHIMADA, Yoshiaki, KUDOH, Masafumi, ISOMURA, Yasuo, SHIKAMA, Hisataka, FUJIKURA, Takashi
Published in Chemical & pharmaceutical bulletin (1996)
Published in Chemical & pharmaceutical bulletin (1996)
Get full text
Journal Article
G12D 변이 KRAS 단백의 분해를 유도하기 위한 퀴나졸린화합물
WATANABE HIDEYUKI, YOSHINARI TOMOHIRO, INAMURA KOHEI, HAMAGUCHI HISAO, NAGASHIMA TAKEYUKI, KAWAGUCHI KENICHI, KURAMOTO KAZUYUKI, MORIKAWA TAKAHIRO, ISHIOKA HIROKI, IMADA SUNAO, OKUMURA MITSUAKI, IMAIZUMI TOMOYOSHI, KAWAMINAMI EIJI
Year of Publication 17.10.2023
Get full text
Year of Publication 17.10.2023
Patent
4-아미노퀴나졸린 화합물
KURIWAKI IKUMI, HAMAGUCHI HISAO, NAGASHIMA TAKEYUKI, KAWAGUCHI KENICHI, KURAMOTO KAZUYUKI, SATO RYO, SEKI YOHEI, MORIKAWA TAKAHIRO, ISHIOKA HIROKI, FUKUDOME HIROKI, IMADA SUNAO, OKUMURA MITSUAKI, IMAIZUMI TOMOYOSHI, KAWAMINAMI EIJI
Year of Publication 17.10.2023
Get full text
Year of Publication 17.10.2023
Patent
HETEROCYCLIC COMPOUND FOR INDUCING DEGRADATION OF G12D MUTANT KRAS PROTEIN
ISHIOKA, Hiroki, KAWAGUCHI, Kenichi, KAWAMINAMI, Eiji, IMAIZUMI, Tomoyoshi, MORIKAWA, Takahiro, INAMURA, Kohei, KURAMOTO, Kazuyuki, TAKAHASHI, Fumie, WATANABE, Hideyuki, HAMAGUCHI, Hisao, NAGASHIMA, Takeyuki, YOSHINARI, Tomohiro
Year of Publication 14.09.2023
Get full text
Year of Publication 14.09.2023
Patent
4-AMINOQUINAZOLINE COMPOUNDS
MORIKAWA, Takahiro, KURAMOTO, Kazuyuki, IMADA, Sunao, HAMAGUCHI, Hisao, KURIWAKI, Ikumi, SATO, Ryo, ISHIOKA, Hiroki, FUKUDOME, Hiroki, KAWAGUCHI, Kenichi, IMAIZUMI, Tomoyoshi, KAWAMINAMI, Eiji, SEKI, Yohei, OKUMURA, Mitsuaki, NAGASHIMA, Takeyuki
Year of Publication 18.08.2022
Get full text
Year of Publication 18.08.2022
Patent
QUINAZOLINE COMPOUND FOR INDUCING DEGRADATION OF G12D-MUTATION KRAS PROTEIN
MORIKAWA, Takahiro, KURAMOTO, Kazuyuki, IMADA, Sunao, WATANABE, Hideyuki, HAMAGUCHI, Hisao, ISHIOKA, Hiroki, KAWAMINAMI, Eiji, KAWAGUCHI, Kenichi, IMAIZUMI, Tomoyoshi, INAMURA, Kohei, OKUMURA, Mitsuaki, NAGASHIMA, Takeyuki, YOSHINARI, Tomohiro
Year of Publication 18.08.2022
Get full text
Year of Publication 18.08.2022
Patent
Studies on Aromatase Inhibitors. III. Synthesis and Biological Evaluation of ((4-Bromobenzyl)(4-cyanophenyl)amino)azoles and Their Azine Analogs
OKADA, Minoru, YODEN, Toru, KAWAMINAMI, Eiji, SHIMADA, Yoshiaki, KUDOH, Masafumi, ISOMURA, Yasuo
Published in Chemical & pharmaceutical bulletin (1997)
Published in Chemical & pharmaceutical bulletin (1997)
Get full text
Journal Article
Studies on Aromatase Inhibitors IV. Synthesis and Biological Evaluation of N, N-Disubstituted-5-aminopyrimidine Derivatives
OKADA, Minoru, YODEN, Toru, KAWAMINAMI, Eiji, SHIMADA, Yosiaki, KUDOU, Masafumi, ISOMURA, Yasuo
Published in Chemical & pharmaceutical bulletin (1997)
Published in Chemical & pharmaceutical bulletin (1997)
Get full text
Journal Article
SUBSTITUTED AMIDE COMPOUND
SAKAMOTO KAZUYUKI, KANAYAMA TAKATOSHI, TAKAHASHI TATSUHISA, KAWAMINAMI EIJI
Year of Publication 05.09.2013
Get full text
Year of Publication 05.09.2013
Patent
SUBSTITUTED AMIDE COMPOUND
SAKAMOTO KAZUYUKI, KANAYAMA TAKATOSHI, TAKAHASHI TATSUHISA, KAWAMINAMI EIJI
Year of Publication 29.03.2012
Get full text
Year of Publication 29.03.2012
Patent