Refined crystal structures of Escherichia coli and chicken liver dihydrofolate reductase containing bound trimethoprim
Matthews, D A, Bolin, J T, Burridge, J M, Filman, D J, Volz, K W, Kaufman, B T, Beddell, C R, Champness, J N, Stammers, D K, Kraut, J
Published in The Journal of biological chemistry (10.01.1985)
Published in The Journal of biological chemistry (10.01.1985)
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Crystal structure of avian dihydrofolate reductase containing phenyltriazine and NADPH
Volz, K W, Matthews, D A, Alden, R A, Freer, S T, Hansch, C, Kaufman, B T, Kraut, J
Published in The Journal of biological chemistry (10.03.1982)
Published in The Journal of biological chemistry (10.03.1982)
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Effects on dihydrofolate reductase of methotrexate metabolites and intracellular folates formed following methotrexate exposure of human breast cancer cells
Drake, J C, Allegra, C J, Baram, J, Kaufman, B T, Chabner, B A
Published in Biochemical pharmacology (15.07.1987)
Published in Biochemical pharmacology (15.07.1987)
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Activation of bovine and chicken liver dihydrofolate reductases and its relationship to a specific cysteine residue in their NH2-terminal amino acid sequences
Kaufman, B T, Kumar, A A, Blankenship, D T, Freisheim, J H
Published in The Journal of biological chemistry (25.07.1980)
Published in The Journal of biological chemistry (25.07.1980)
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Inhibition of chicken liver dihydrofolate reductase by 5-(substituted benzyl)-2,4-diaminopyrimidines. A quantitative structure-activity relationship and graphics analysis
SELASSIE, C. D, FANG, Z.-X, LI, R.-L, HANSCH, C, KLEIN, T, LANGRIDGE, R, KAUFMAN, B. T
Published in Journal of medicinal chemistry (01.05.1986)
Published in Journal of medicinal chemistry (01.05.1986)
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Crystal structure of chicken liver dihydrofolate reductase complexed with NADP+ and biopterin
McTigue, Michele A, Davies, Jay F, Kaufman, Bernard T, Kraut, Joseph
Published in Biochemistry (Easton) (18.08.1992)
Published in Biochemistry (Easton) (18.08.1992)
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Why NADP?
Kaufman, Bernard T.
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (01.08.1993)
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (01.08.1993)
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On the structure selectivity problem in drug design. A comparative study of benzylpyrimidine inhibition of vertebrate and bacterial dihydrofolate reductase via molecular graphics and quantitative structure-activity relationships
Selassie, Cynthia Dias, Fang, Zhaoxia, Li, Renli, Hansch, Corwin, Debnath, Gargi, Klein, Teri, Langridge, Robert, Kaufman, Bernard T
Published in Journal of medicinal chemistry (01.08.1989)
Published in Journal of medicinal chemistry (01.08.1989)
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Chromatographic separation of the diastereoisomers of dl, L-5, 10-methylenetetrahydrofolate
KAUFMAN, B T, DONALDSON, K O, KERESZTESY, J C
Published in The Journal of biological chemistry (01.04.1963)
Published in The Journal of biological chemistry (01.04.1963)
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Crystallography, quantitative structure-activity relationships, (QSAR) and molecular graphics in a comparative analysis of the inhibition of dihydrofolate reductase from chicken liver and Lactobacillus casei by 4,6-diamino-1,2-dihydro-2,2-dimethyl-1-(substituted-phenyl)-s-triazines
Hansch, Corwin, Hathaway, Bruce A, Guo, Zongru, Selassie, Cynthia Dias, Dietrich, Stephen W, Blaney, Jeffrey M, Langridge, Robert, Volz, Karl W, Kaufman, Bernard T
Published in Journal of medicinal chemistry (01.02.1984)
Published in Journal of medicinal chemistry (01.02.1984)
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