Next-generation XPO1 inhibitor shows improved efficacy and in vivo tolerability in hematological malignancies
Hing, Z A, Fung, H Y J, Ranganathan, P, Mitchell, S, El-Gamal, D, Woyach, J A, Williams, K, Goettl, V M, Smith, J, Yu, X, Meng, X, Sun, Q, Cagatay, T, Lehman, A M, Lucas, D M, Baloglu, E, Shacham, S, Kauffman, M G, Byrd, J C, Chook, Y M, Garzon, R, Lapalombella, R
Published in Leukemia (01.12.2016)
Published in Leukemia (01.12.2016)
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XPO1 (CRM1) inhibition represses STAT3 activation to drive a survivin-dependent oncogenic switch in triple-negative breast cancer
Cheng, Yan, Holloway, Michael P, Nguyen, Kevin, McCauley, Dilara, Landesman, Yosef, Kauffman, Michael G, Shacham, Sharon, Altura, Rachel A
Published in Molecular cancer therapeutics (01.03.2014)
Published in Molecular cancer therapeutics (01.03.2014)
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Preclinical and clinical efficacy of XPO1/CRM1 inhibition by the karyopherin inhibitor KPT-330 in Ph+ leukemias
Walker, Christopher J., Oaks, Joshua J., Santhanam, Ramasamy, Neviani, Paolo, Harb, Jason G., Ferenchak, Gregory, Ellis, Justin J., Landesman, Yosef, Eisfeld, Ann-Kathrin, Gabrail, Nash Y., Smith, Carrie L., Caligiuri, Michael A., Hokland, Peter, Roy, Denis Claude, Reid, Alistair, Milojkovic, Dragana, Goldman, John M., Apperley, Jane, Garzon, Ramiro, Marcucci, Guido, Shacham, Sharon, Kauffman, Michael G., Perrotti, Danilo
Published in Blood (24.10.2013)
Published in Blood (24.10.2013)
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Oral eltanexor treatment of patients with higher-risk myelodysplastic syndrome refractory to hypomethylating agents
Lee, Sangmin, Mohan, Sanjay, Knupp, Jessica, Chamoun, Kamal, de Jonge, Adrienne, Yang, Fan, Baloglu, Erkan, Shah, Jatin, Kauffman, Michael G, Shacham, Sharon, Bhatnagar, Bhavana
Published in Journal of hematology and oncology (03.08.2022)
Published in Journal of hematology and oncology (03.08.2022)
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Oral Selinexor–Dexamethasone for Triple-Class Refractory Multiple Myeloma
Chari, Ajai, Vogl, Dan T, Gavriatopoulou, Maria, Nooka, Ajay K, Yee, Andrew J, Huff, Carol A, Moreau, Philippe, Dingli, David, Cole, Craig, Lonial, Sagar, Dimopoulos, Meletios, Stewart, A. Keith, Richter, Joshua, Vij, Ravi, Tuchman, Sascha, Raab, Marc S, Weisel, Katja C, Delforge, Michel, Cornell, Robert F, Kaminetzky, David, Hoffman, James E, Costa, Luciano J, Parker, Terri L, Levy, Moshe, Schreder, Martin, Meuleman, Nathalie, Frenzel, Laurent, Mohty, Mohamad, Choquet, Sylvain, Schiller, Gary, Comenzo, Raymond L, Engelhardt, Monika, Illmer, Thomas, Vlummens, Philip, Doyen, Chantal, Facon, Thierry, Karlin, Lionel, Perrot, Aurore, Podar, Klaus, Kauffman, Michael G, Shacham, Sharon, Li, Lingling, Tang, Shijie, Picklesimer, Carla, Saint-Martin, Jean-Richard, Crochiere, Marsha, Chang, Hua, Parekh, Samir, Landesman, Yosef, Shah, Jatin, Richardson, Paul G, Jagannath, Sundar
Published in The New England journal of medicine (22.08.2019)
Published in The New England journal of medicine (22.08.2019)
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Selinexor‐based regimens in patients with multiple myeloma after prior anti‐B‐cell maturation antigen treatment
Baljevic, Muhamed, Gasparetto, Cristina, Schiller, Gary J., Tuchman, Sascha A., Callander, Natalie S., Lentzsch, Suzanne, Monge, Jorge, Kotb, Rami, Bahlis, Nizar J., White, Darrell, Chen, Christine I., Sutherland, Heather J., Madan, Sumit, LeBlanc, Richard, Sebag, Michael, Venner, Christopher P., Bensinger, William I., Biran, Noa, DeCastro, Andrew, Van Domelen, Dane R., Zhang, Chris, Shah, Jatin J., Shacham, Sharon, Kauffman, Michael G., Bentur, Ohad S., Lipe, Brea
Published in EJHaem (01.11.2022)
Published in EJHaem (01.11.2022)
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High-resolution stratigraphy of the Cenomanian–Turonian boundary interval at Pueblo (USA) and wadi Bahloul (Tunisia): stable isotope and bio-events correlation
Caron, Michèle, Dall’Agnolo, Stephan, Accarie, Hugues, Barrera, Enriqueta, Kauffman, Erle G., Amédro, Francis, Robaszynski, Francis
Published in Geobios (01.03.2006)
Published in Geobios (01.03.2006)
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A 0.9-V DAC-Calibration-Free Continuous-Time Incremental Delta-Sigma Modulator Achieving 97-dB SFDR at 2 MS/s in 28-nm CMOS
Mokhtar, Mohamed A., Abdelaal, Ahmed, Sporer, Markus, Becker, Joachim, Kauffman, John G., Ortmanns, Maurits
Published in IEEE journal of solid-state circuits (01.11.2022)
Published in IEEE journal of solid-state circuits (01.11.2022)
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Survival among patients with relapsed/refractory diffuse large B cell lymphoma treated with single-agent selinexor in the SADAL study
Maerevoet, Marie, Zijlstra, Josee M, Follows, George, Casasnovas, Rene-Olivier, Vermaat, J. S. P, Kalakonda, Nagesh, Goy, Andre, Choquet, Sylvain, Van Den Neste, Eric, Hill, Brian, Thieblemont, Catherine, Cavallo, Federica, De la Cruz, Fatima, Kuruvilla, John, Hamad, Nada, Jaeger, Ulrich, Caimi, Paolo, Gurion, Ronit, Warzocha, Krzysztof, Bakhshi, Sameer, Sancho, Juan-Manuel, Schuster, Michael, Egyed, Miklos, Offner, Fritz, Vassilakopoulos, Theodoros P, Samal, Priyanka, Ku, Matthew, Ma, Xiwen, Corona, Kelly, Chamoun, Kamal, Shah, Jatin, Shacham, Sharon, Kauffman, Michael G, Canales, Miguel
Published in Journal of hematology and oncology (16.07.2021)
Published in Journal of hematology and oncology (16.07.2021)
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Selinexor, a novel selective inhibitor of nuclear export, reduces SARS-CoV-2 infection and protects the respiratory system in vivo
Kashyap, Trinayan, Murray, Jackelyn, Walker, Christopher J., Chang, Hua, Tamir, Sharon, Hou, Bing, Shacham, Sharon, Kauffman, Michael G., Tripp, Ralph A., Landesman, Yosef
Published in Antiviral research (01.08.2021)
Published in Antiviral research (01.08.2021)
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A Phase II Study of the Efficacy and Safety of Oral Selinexor in Recurrent Glioblastoma
Lassman, Andrew B, Wen, Patrick Y, van den Bent, Martin J, Plotkin, Scott R, Walenkamp, Annemiek M E, Green, Adam L, Li, Kai, Walker, Christopher J, Chang, Hua, Tamir, Sharon, Henegar, Leah, Shen, Yao, Alvarez, Mariano J, Califano, Andrea, Landesman, Yosef, Kauffman, Michael G, Shacham, Sharon, Mau-Sørensen, Morten
Published in Clinical cancer research (01.02.2022)
Published in Clinical cancer research (01.02.2022)
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