Discovery of a chemical probe for PRDM9
Allali-Hassani, Abdellah, Szewczyk, Magdalena M., Ivanochko, Danton, Organ, Shawna L., Bok, Jabez, Ho, Jessica Sook Yuin, Gay, Florence P. H., Li, Fengling, Blazer, Levi, Eram, Mohammad S., Halabelian, Levon, Dilworth, David, Luciani, Genna M., Lima-Fernandes, Evelyne, Wu, Qin, Loppnau, Peter, Palmer, Nathan, Talib, S. Zakiah A., Brown, Peter J., Schapira, Matthieu, Kaldis, Philipp, O’Hagan, Ronan C., Guccione, Ernesto, Barsyte-Lovejoy, Dalia, Arrowsmith, Cheryl H., Sanders, John M., Kattar, Solomon D., Bennett, D. Jonathan, Nicholson, Benjamin, Vedadi, Masoud
Published in Nature communications (17.12.2019)
Published in Nature communications (17.12.2019)
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Structure-Guided Discovery of Aminoquinazolines as Brain-Penetrant and Selective LRRK2 Inhibitors
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Published in Journal of medicinal chemistry (13.01.2022)
Published in Journal of medicinal chemistry (13.01.2022)
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Discovery and Optimization of N‑Heteroaryl Indazole LRRK2 Inhibitors
Logan, Kaitlyn M., Kaplan, Will, Simov, Vladimir, Zhou, Hua, Li, Derun, Torres, Luis, Morriello, Gregori J., Acton, John J., Pio, Barbara, Chen, Yi-Heng, Keylor, Mitchell H., Johnson, Rebecca, Kattar, Solomon D., Chau, Ryan, Yan, Xin, Ardolino, Michael, Zarate, Cayetana, Otte, Karin M., Palte, Rachel L., Xiong, Tina, McMinn, Spencer E., Lin, Shishi, Neelamkavil, Santhosh F., Liu, Ping, Su, Jing, Hegde, Laxminarayan G., Woodhouse, Janice D., Moy, Lily Y., Ciaccio, Paul J., Piesvaux, Jennifer, Zebisch, Matthias, Henry, Clare, Barker, John, Wood, Harold B., Kennedy, Matthew E., DiMauro, Erin F., Fell, Matthew J., Fuller, Peter H.
Published in Journal of medicinal chemistry (26.09.2024)
Published in Journal of medicinal chemistry (26.09.2024)
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Discovery of MK-1468: A Potent, Kinome-Selective, Brain-Penetrant Amidoisoquinoline LRRK2 Inhibitor for the Potential Treatment of Parkinson’s Disease
Kattar, Solomon D., Gulati, Anmol, Margrey, Kaila A., Keylor, Mitchell H., Ardolino, Michael, Yan, Xin, Johnson, Rebecca, Palte, Rachel L., McMinn, Spencer E., Nogle, Lisa, Su, Jing, Xiao, Dong, Piesvaux, Jennifer, Lee, Susi, Hegde, Laxminarayan G., Woodhouse, Janice D., Faltus, Robert, Moy, Lily Y., Xiong, Tina, Ciaccio, Paul J., Pearson, Kara, Patel, Mayankbhai, Otte, Karin M., Leyns, Cheryl E.G., Kennedy, Matthew E., Bennett, David Jonathan, DiMauro, Erin F., Fell, Matthew J., Fuller, Peter H.
Published in Journal of medicinal chemistry (09.11.2023)
Published in Journal of medicinal chemistry (09.11.2023)
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Discovery of a new series of PI3K-δ inhibitors from Virtual Screening
Fradera, Xavier, Deng, Qiaolin, Achab, Abdelganhi, Garcia, Yudith, Kattar, Solomon D., McGowan, Meredeth A., Methot, Joey L., Wilson, Kevin, Zhou, Hua, Shaffer, Lynsey, Goldenblatt, Peter, Tong, Vincent, Augustin, Martin A, Altman, Michael D., Lesburg, Charles A., Shah, Sanjiv, Katz, Jason D.
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
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Optimization of brain-penetrant picolinamide derived leucine-rich repeat kinase 2 (LRRK2) inhibitors
Gulati, Anmol, Yeung, Charles S, Lapointe, Blair, Kattar, Solomon D, Gunaydin, Hakan, Scott, Jack D, Childers, Kaleen K, Methot, Joey L, Simov, Vladimir, Kurukulasuriya, Ravi, Pio, Barbara, Morriello, Greg J, Liu, Ping, Tang, Haiqun, Neelamkavil, Santhosh, Wood, Harold B, Rada, Vanessa L, Ardolino, Michael J, Yan, Xin Cindy, Palte, Rachel, Otte, Karin, Faltus, Robert, Woodhouse, Janice, Hegde, Laxminarayan G, Ciaccio, Paul, Minnihan, Ellen C, DiMauro, Erin F, Fell, Matthew J, Fuller, Peter H, Ellis, J. Michael
Published in MedChemComm (21.07.2021)
Published in MedChemComm (21.07.2021)
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LRRK2 억제제로서의 N-연결된 이소퀴놀린 아미드, 제약 조성물 및 그의 용도
FULLER PETER H, YAN XIN, GULATI ANMOL, MARGREY KAILA A, KATTAR SOLOMON D, KEYLOR MITCHELL H
Year of Publication 30.06.2023
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Year of Publication 30.06.2023
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Parallel medicinal chemistry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1:2) optimization
Kattar, Solomon D., Surdi, Laura M., Zabierek, Anna, Methot, Joey L., Middleton, Richard E., Hughes, Bethany, Szewczak, Alexander A., Dahlberg, William K., Kral, Astrid M., Ozerova, Nicole, Fleming, Judith C., Wang, Hongmei, Secrist, Paul, Harsch, Andreas, Hamill, Julie E., Cruz, Jonathan C., Kenific, Candia M., Chenard, Melissa, Miller, Thomas A., Berk, Scott C., Tempest, Paul
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Neurofilaments Consist of Distinct Populations That Can Be Distinguished by C-Terminal Phosphorylation, Bundling, and Axonal Transport Rate in Growing Axonal Neurites
Yabe, Jason T, Chylinski, Teresa, Wang, Feng-Song, Pimenta, Aurea, Kattar, Solomon D, Linsley, Maria-Dawn, Chan, Walter K-H, Shea, Thomas B
Published in The Journal of neuroscience (01.04.2001)
Published in The Journal of neuroscience (01.04.2001)
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LRRK2 억제제로서의 N- 퀴나졸린-2-아민 유도체, 제약 조성물 및 그의 용도
FULLER PETER H, YU ELSIE C, GULATI ANMOL, JOHNSON REBECCA ELIZABETH, CHAU RYAN W, NEELAMKAVIL SANTHOSH F, KEYLOR MITCHELL H, MORRIELLO GREGORI J, YAN XIN, MARGREY KAILA A, ZARATE SAEZ CAYETANA CARMELA, ARDOLINO MICHAEL J, KATTAR SOLOMON D
Year of Publication 28.06.2022
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Year of Publication 28.06.2022
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Discovery of a new series of PI3K-6 inhibitors from Virtual Screening
Fradera, Xavier, Deng, Qiaolin, Achab, Abdelganhi, Garcia, Yudith, Kattar, Solomon D., McGowan, Meredeth A., Methot, Joey L., Wilson, Kevin, Zhou, Hua, Shaffer, Lynsey, Goldenblatt, Peter, Tong, Vincent, Augustin, Martin A., Altman, Michael D., Lesburg, Charles A., Shah, Sanjiv, Katz, Jason D.
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
Published in Bioorganic & medicinal chemistry letters (15.06.2021)
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AMINOPYRIMIDINES AS SYK INHIBITORS
DI FRANCESCO MARIA EMILIA, ZHOU HUA, GRIMM JONATHAN, CHILDERS KALEEN KONRAD, SCHELL ADAM J, ALTMAN MICHAEL D, HAIDLE ANDREW M, ELLIS JOHN MICHAEL, OTTE RYAN D, PETROCCHI ALESSIA, FISCHER CHRISTIAN, NORTHRUP ALAN B, KATTAR SOLOMON D
Year of Publication 07.03.2014
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Year of Publication 07.03.2014
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N-LINKED ISOQUINOLINE AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
Fuller, Peter H, Keylor, Mitchell H, Yan, Xin, Margrey, Kaila A, Gulati, Anmol, Kattar, Solomon D
Year of Publication 21.12.2023
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Year of Publication 21.12.2023
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SYSTEM AND METHOD FOR STATIC AND DYNAMIC MRI SHIMMING
MARGREY, Kaila, A, YAN, Xin, TORRES, Luis, GULATI, Anmol, FULLER, Peter, H, KEYLOR, Mitchell, H, KATTAR, Solomon, D
Year of Publication 07.08.2024
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Year of Publication 07.08.2024
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N-LINKED ISOQUINOLINE AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
YAN, XIN, GULATI, ANMOL, MARGREY, KAILA A, FULLER, PETER H, KATTAR, SOLOMON D, KEYLOR, MITCHELL H
Year of Publication 05.05.2022
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Year of Publication 05.05.2022
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HETEROARYL AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
Methot, Joey L, Ellis, J. Michael, Gunaydin, Hakan, Childers, Kaleen Konrad, Simov, Vladimir, Morriello, Gregori J, Kurukulasuriya, Ravi, Fuller, Peter H, Lapointe, Blair T, Gulati, Anmol, Neelamkavil, Santhosh, Yeung, Charles S, Kattar, Solomon D
Year of Publication 19.09.2024
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Year of Publication 19.09.2024
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HETEROAROYL AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
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Year of Publication 24.01.2024
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Year of Publication 24.01.2024
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N-(HETEROARYL) QUINAZOLIN-2-AMINE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
MARGREY, Kaila, A, YAN, Xin, GULATI, Anmol, NEELAMKAVIL, Santhosh, F, FULLER, Peter, H, ZARATE SAEZ, Cayetana Carmela, ARDOLINO, Michael, J, JOHNSON, Rebecca Elizabeth, KATTAR, Solomon, D, CHAU, Ryan, W, KEYLOR, Mitchell, H, YU, Elsie, C, MORRIELLO, Gregori, J
Year of Publication 22.11.2023
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Year of Publication 22.11.2023
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