ASP5878, a Novel Inhibitor of FGFR1, 2, 3, and 4, Inhibits the Growth of FGF19-Expressing Hepatocellular Carcinoma
Futami, Takashi, Okada, Hidetsugu, Kihara, Rumi, Kawase, Tatsuya, Nakayama, Ayako, Suzuki, Tomoyuki, Kameda, Minoru, Shindoh, Nobuaki, Terasaka, Tadashi, Hirano, Masaaki, Kuromitsu, Sadao
Published in Molecular cancer therapeutics (01.01.2017)
Published in Molecular cancer therapeutics (01.01.2017)
Get full text
Journal Article
ASP5878, a selective FGFR inhibitor, to treat FGFR3‐dependent urothelial cancer with or without chemoresistance
Kikuchi, Aya, Suzuki, Tomoyuki, Nakazawa, Taisuke, Iizuka, Masateru, Nakayama, Ayako, Ozawa, Tohru, Kameda, Minoru, Shindoh, Nobuaki, Terasaka, Tadashi, Hirano, Masaaki, Kuromitsu, Sadao
Published in Cancer science (01.02.2017)
Published in Cancer science (01.02.2017)
Get full text
Journal Article
Asymmetric phase-transfer catalysis of homo- and heterochiral quaternary ammonium salts: development and application of conformationally flexible chiral phase-transfer catalysts
Ooi, Takashi, Uematsu, Yukitaka, Kameda, Minoru, Maruoka, Keiji
Published in Tetrahedron (04.12.2006)
Published in Tetrahedron (04.12.2006)
Get full text
Journal Article
Facile synthesis of l-Dopa tert-butyl ester by catalytic enantioselective phase-transfer alkylation
Ooi, Takashi, Kameda, Minoru, Tannai, Hidenori, Maruoka, Keiji
Published in Tetrahedron letters (01.10.2000)
Published in Tetrahedron letters (01.10.2000)
Get full text
Journal Article
Design of N-Spiro C2-Symmetric Chiral Quaternary Ammonium Bromides as Novel Chiral Phase-Transfer Catalysts: Synthesis and Application to Practical Asymmetric Synthesis of α-Amino Acids
OOI, Takashi, KAMEDA, Minoru, MARUOKA, Keiji
Published in Journal of the American Chemical Society (30.04.2003)
Published in Journal of the American Chemical Society (30.04.2003)
Get full text
Journal Article
Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity
Kuriwaki, Ikumi, Kameda, Minoru, Iikubo, Kazuhiko, Hisamichi, Hiroyuki, Kawamoto, Yuichiro, Kikuchi, Shigetoshi, Moritomo, Hiroyuki, Terasaka, Tadashi, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Kikuchi, Aya, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (01.04.2022)
Published in Bioorganic & medicinal chemistry (01.04.2022)
Get full text
Journal Article
Design of N-Spiro C 2-Symmetric Chiral Quaternary Ammonium Bromides as Novel Chiral Phase-Transfer Catalysts: Synthesis and Application to Practical Asymmetric Synthesis of α-Amino Acids
Ooi, Takashi, Kameda, Minoru, Maruoka, Keiji
Published in Journal of the American Chemical Society (30.04.2003)
Published in Journal of the American Chemical Society (30.04.2003)
Get full text
Journal Article
Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2
Kuriwaki, Ikumi, Kameda, Minoru, Hisamichi, Hiroyuki, Kikuchi, Shigetoshi, Iikubo, Kazuhiko, Kawamoto, Yuichiro, Moritomo, Hiroyuki, Kondoh, Yutaka, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Suzuki, Tomoyuki, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (15.05.2020)
Published in Bioorganic & medicinal chemistry (15.05.2020)
Get full text
Journal Article
Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency
Kuriwaki, Ikumi, Kameda, Minoru, Iikubo, Kazuhiko, Hisamichi, Hiroyuki, Kawamoto, Yuichiro, Kikuchi, Shigetoshi, Moritomo, Hiroyuki, Kondoh, Yutaka, Terasaka, Tadashi, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Nakazawa, Taisuke, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (01.03.2021)
Published in Bioorganic & medicinal chemistry (01.03.2021)
Get full text
Journal Article