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Jefferies, Harold B J, Cooke, Frank T, Jat, Parmjit, Boucheron, Christine, Koizumi, Tomonobu, Hayakawa, Masahiko, Kaizawa, Hiroyuki, Ohishi, Takahide, Workman, Paul, Waterfield, Michael D, Parker, Peter J
Published in EMBO reports (01.02.2008)
Published in EMBO reports (01.02.2008)
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PIKfyve Negatively Regulates Exocytosis in Neurosecretory Cells
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Published in Bioorganic & medicinal chemistry (15.10.2004)
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Design, synthesis and biological activity of YM-60828 derivatives: Potent and orally-bioavailable factor Xa inhibitors based on naphthoanilide and naphthalensulfonanilide templates
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Published in Bioorganic & medicinal chemistry (01.08.2002)
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A selective PIKfyve inhibitor blocks PtdIns(3,5)P 2 production and disrupts endomembrane transport and retroviral budding
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Published in EMBO reports (01.02.2008)
Published in EMBO reports (01.02.2008)
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Synthesis and biological evaluation of 4-morpholino-2-phenylquinazolines and related derivatives as novel PI3 kinase p110α inhibitors
Hayakawa, Masahiko, Kaizawa, Hiroyuki, Moritomo, Hiroyuki, Koizumi, Tomonobu, Ohishi, Takahide, Okada, Minoru, Ohta, Mitsuaki, Tsukamoto, Shin-ichi, Parker, Peter, Workman, Paul, Waterfield, Mike
Published in Bioorganic & medicinal chemistry (15.10.2006)
Published in Bioorganic & medicinal chemistry (15.10.2006)
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Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Synthesis and biological evaluation of sulfonylhydrazone-substituted imidazo[1,2- a]pyridines as novel PI3 kinase p110α inhibitors
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Published in Bioorganic & medicinal chemistry (01.09.2007)
Published in Bioorganic & medicinal chemistry (01.09.2007)
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Synthesis and biological evaluation of imidazo[1,2- a]pyridine derivatives as novel PI3 kinase p110α inhibitors
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Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
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Targeting PI3KC2β Impairs Proliferation and Survival in Acute Leukemia, Brain Tumours and Neuroendocrine Tumours
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Published in Anticancer research (01.08.2012)
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Published in Anticancer research (01.08.2012)
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Year of Publication 11.01.2017
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Year of Publication 27.09.2013
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Year of Publication 27.09.2013
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Year of Publication 03.12.2015
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QUINOXALINE COMPOUND
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Year of Publication 02.09.2013
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Year of Publication 02.09.2013
Patent
A selective PIKfyve inhibitor blocks PtdIns(3,5)P sub(2) production and disrupts endomembrane transport and retroviral budding
Jefferies, Harold B J, Cooke, Frank T, Jat, Parmjit, Boucheron, Christine, Koizumi, Tomonobu, Hayakawa, Masahiko, Kaizawa, Hiroyuki, Ohishi, Takahide, Workman, Paul, Waterfield, Michael D, Parker, Peter J
Published in EMBO reports (01.02.2008)
Published in EMBO reports (01.02.2008)
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Journal Article
A selective PIKfyve inhibitor blocks PtdIns(3,5)P(2) production and disrupts endomembrane transport and retroviral budding
Jefferies, Harold B J, Cooke, Frank T, Jat, Parmjit, Boucheron, Christine, Koizumi, Tomonobu, Hayakawa, Masahiko, Kaizawa, Hiroyuki, Ohishi, Takahide, Workman, Paul, Waterfield, Michael D, Parker, Peter J
Published in EMBO reports (01.02.2008)
Published in EMBO reports (01.02.2008)
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Journal Article
PYRAZOLOQUINOLINE COMPOUND
KAIZAWA, HIROYUKI, YAMAMOTO, SATOSHI, UKAI, ATSUSHI, KAMIJO, KAZUNORI, YAMAMOTO, HIROFUMI, SUGITA, MARI, SEO, RYUSHII
Year of Publication 15.03.2012
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Year of Publication 15.03.2012
Patent
QUINOXALINE COMPOUND
KAIZAWA, HIROYUKI, YAMAMOTO, SATOSHI, KAMIJO, KAZUNORI, YAMAMOTO, HIROFUMI, SEO, RYUSHI, SUGITA, MARI, TSUCHIYA, KAZUYUKI
Year of Publication 15.03.2012
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Year of Publication 15.03.2012
Patent