Design, synthesis, and biological activity of novel, potent, and highly selective fused pyrimidine-2-carboxamide-4-one-based matrix metalloproteinase (MMP)-13 zinc-binding inhibitors
Nara, Hiroshi, Sato, Kenjiro, Kaieda, Akira, Oki, Hideyuki, Kuno, Haruhiko, Santou, Takashi, Kanzaki, Naoyuki, Terauchi, Jun, Uchikawa, Osamu, Kori, Masakuni
Published in Bioorganic & medicinal chemistry (01.12.2016)
Published in Bioorganic & medicinal chemistry (01.12.2016)
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Discovery of Novel, Highly Potent, and Selective Matrix Metalloproteinase (MMP)-13 Inhibitors with a 1,2,4-Triazol-3-yl Moiety as a Zinc Binding Group Using a Structure-Based Design Approach
Nara, Hiroshi, Kaieda, Akira, Sato, Kenjiro, Naito, Takako, Mototani, Hideyuki, Oki, Hideyuki, Yamamoto, Yoshio, Kuno, Haruhiko, Santou, Takashi, Kanzaki, Naoyuki, Terauchi, Jun, Uchikawa, Osamu, Kori, Masakuni
Published in Journal of medicinal chemistry (26.01.2017)
Published in Journal of medicinal chemistry (26.01.2017)
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Journal Article
Identification of 2,6-Disubstituted 3H‑Imidazo[4,5‑b]pyridines as Therapeutic Agents for Dysferlinopathies through Phenotypic Screening on Patient-Derived Induced Pluripotent Stem Cells
Takada, Hiroyuki, Kaieda, Akira, Tawada, Michiko, Nagino, Tomoko, Sasa, Katsunori, Oikawa, Tatsuo, Oki, Akiko, Sameshima, Tomoya, Miyamoto, Kazumasa, Miyamoto, Makoto, Kokubu, Yuko, Tozawa, Ryuichi, Sakurai, Hidetoshi, Saito, Bunnai
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Novel HDAC6 Inhibitors Increase Tubulin Acetylation and Rescue Axonal Transport of Mitochondria in a Model of Charcot–Marie–Tooth Type 2F
Adalbert, Robert, Kaieda, Akira, Antoniou, Christina, Loreto, Andrea, Yang, Xiuna, Gilley, Jonathan, Hoshino, Takashi, Uga, Keiko, Makhija, Mahindra T, Coleman, Michael P
Published in ACS chemical neuroscience (05.02.2020)
Published in ACS chemical neuroscience (05.02.2020)
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Journal Article
Identification of 2,6-Disubstituted 3 H -Imidazo[4,5- b ]pyridines as Therapeutic Agents for Dysferlinopathies through Phenotypic Screening on Patient-Derived Induced Pluripotent Stem Cells
Takada, Hiroyuki, Kaieda, Akira, Tawada, Michiko, Nagino, Tomoko, Sasa, Katsunori, Oikawa, Tatsuo, Oki, Akiko, Sameshima, Tomoya, Miyamoto, Kazumasa, Miyamoto, Makoto, Kokubu, Yuko, Tozawa, Ryuichi, Sakurai, Hidetoshi, Saito, Bunnai
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Journal Article
Structure-based design, synthesis, and biological evaluation of imidazo[1,2-b]pyridazine-based p38 MAP kinase inhibitors
Kaieda, Akira, Takahashi, Masashi, Takai, Takafumi, Goto, Masayuki, Miyazaki, Takahiro, Hori, Yuri, Unno, Satoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Itono, Sachiko, Takagi, Terufumi, Hamada, Teruki, Shirasaki, Mikio, Okada, Kengo, Snell, Gyorgy, Bragstad, Ken, Sang, Bi-Ching, Uchikawa, Osamu, Miwatashi, Seiji
Published in Bioorganic & medicinal chemistry (01.02.2018)
Published in Bioorganic & medicinal chemistry (01.02.2018)
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Journal Article
Structure‐Based Design, Synthesis, and Biological Evaluation of ImidazoPyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 2
Kaieda, Akira, Takahashi, Masashi, Fukuda, Hiromi, Okamoto, Rei, Morimoto, Shinji, Gotoh, Masayuki, Miyazaki, Takahiro, Hori, Yuri, Unno, Satoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Itono, Sachiko, Takagi, Terufumi, Sugimoto, Hiroshi, Okada, Kengo, Weston, Lane, Bi‐Ching Sang, Kumar Saikatendu, Matsunaga, Shinichiro, Miwatashi, Seiji
Published in ChemMedChem (01.12.2019)
Published in ChemMedChem (01.12.2019)
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Journal Article
Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5‐b]Pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 2
Kaieda, Akira, Takahashi, Masashi, Fukuda, Hiromi, Okamoto, Rei, Morimoto, Shinji, Gotoh, Masayuki, Miyazaki, Takahiro, Hori, Yuri, Unno, Satoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Itono, Sachiko, Takagi, Terufumi, Sugimoto, Hiroshi, Okada, Kengo, Lane, Weston, Sang, Bi‐Ching, Saikatendu, Kumar, Matsunaga, Shinichiro, Miwatashi, Seiji
Published in ChemMedChem (17.12.2019)
Published in ChemMedChem (17.12.2019)
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Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazopyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 1
Kaieda, Akira, Takahashi, Masashi, Fukuda, Hiromi, Okamoto, Rei, Morimoto, Shinji, Gotoh, Masayuki, Miyazaki, Takahiro, Hori, Yuri, Unno, Satoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Itono, Sachiko, Takagi, Terufumi, Sugimoto, Hiroshi, Okada, Kengo, Snell, Gyorgy, Bertsch, Ryan, Nguyen, Jasmine, Bi‐Ching Sang, Miwatashi, Seiji
Published in ChemMedChem (01.05.2019)
Published in ChemMedChem (01.05.2019)
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Journal Article
Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4,5‐b]pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 1
Kaieda, Akira, Takahashi, Masashi, Fukuda, Hiromi, Okamoto, Rei, Morimoto, Shinji, Gotoh, Masayuki, Miyazaki, Takahiro, Hori, Yuri, Unno, Satoko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Itono, Sachiko, Takagi, Terufumi, Sugimoto, Hiroshi, Okada, Kengo, Snell, Gyorgy, Bertsch, Ryan, Nguyen, Jasmine, Sang, Bi‐Ching, Miwatashi, Seiji
Published in ChemMedChem (17.05.2019)
Published in ChemMedChem (17.05.2019)
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Journal Article
헤테로시클릭 화합물
IKEURA YOSHINORI, YOSHIDA YOSHINORI, NARA HIROSHI, KAIEDA AKIRA, KONDO SHIGERU, MIKI KENJI
Year of Publication 11.12.2020
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Year of Publication 11.12.2020
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Year of Publication 03.10.2019
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Year of Publication 03.10.2019
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HETEROCYCLIC COMPOUND
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Year of Publication 28.01.2021
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HETEROCYCLIC COMPOUND
NARA, Hiroshi, YOSHIKAWA, Masato, KAIEDA, Akira, ISHII, Naoki, DAINI, Masaki
Year of Publication 02.03.2017
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Year of Publication 02.03.2017
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HETEROCYCLIC COMPOUND
HANYA, Yuki, ICHIKAWA, Takashi, KAWASAKI, Masanori, IMAEDA, Toshihiro, KIKUCHI, Fumiaki, OYABU, Norio, FUKUDA, Hiromi, SHIOKAWA, Zenyu, YOSHIKAWA, Takeshi, NEGORO, Nobuyuki, KAIEDA, Akira
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Year of Publication 11.04.2019
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NARA, Hiroshi, YOSHIKAWA, Masato, KAIEDA, Akira, ISHII, Naoki, HIDAKA, Kousuke, TOYOFUKU, Masashi, DAINI, Masaki
Year of Publication 26.01.2017
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Year of Publication 26.01.2017
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HETEROCYCLIC COMPOUND
TOYOFUKU, MASASHI, HIDAKA, KOUSUKE, ISHII, NAOKI, YOSHIKAWA, MASATO, DAINI, MASAKI, KAIEDA, AKIRA, NARA, HIROSHI
Year of Publication 03.03.2016
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Year of Publication 03.03.2016
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IMAEDA, TOSHIHIRO, DAINI, MASAKI, KIKUCHI, FUMIAKI, NARA, HIROSHI, KAIEDA, AKIRA, KAMEI, TAKU
Year of Publication 05.12.2013
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Year of Publication 05.12.2013
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