Muscarinic acetylcholine receptors: novel opportunities for drug development
Kruse, Andrew C, Kobilka, Brian K, Gautam, Dinesh, Sexton, Patrick M, Christopoulos, Arthur, Wess, Jürgen
Published in Nature reviews. Drug discovery (01.07.2014)
Published in Nature reviews. Drug discovery (01.07.2014)
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Journal Article
β-Arrestins as Important Regulators of Glucose and Energy Homeostasis
Pydi, Sai P, Barella, Luiz F, Zhu, Lu, Meister, Jaroslawna, Rossi, Mario, Wess, Jürgen
Published in Annual review of physiology (10.02.2022)
Published in Annual review of physiology (10.02.2022)
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Journal Article
Key Metabolic Functions of β-Arrestins: Studies with Novel Mouse Models
Pydi, Sai P., Barella, Luiz F., Meister, Jaroslawna, Wess, Jürgen
Published in Trends in endocrinology and metabolism (01.02.2021)
Published in Trends in endocrinology and metabolism (01.02.2021)
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Journal Article
β-Cell-intrinsic β-arrestin 1 signaling enhances sulfonylurea-induced insulin secretion
Barella, Luiz F, Rossi, Mario, Zhu, Lu, Cui, Yinghong, Mei, Fang C, Cheng, Xiaodong, Chen, Wei, Gurevich, Vsevolod V, Wess, Jürgen
Published in The Journal of clinical investigation (03.09.2019)
Published in The Journal of clinical investigation (03.09.2019)
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Journal Article
Gigantism and Acromegaly Due to Xq26 Microduplications and GPR101 Mutation
Trivellin, Giampaolo, Daly, Adrian F, Faucz, Fabio R, Yuan, Bo, Rostomyan, Liliya, Larco, Darwin O, Schernthaner-Reiter, Marie Helene, Szarek, Eva, Leal, Letícia F, Caberg, Jean-Hubert, Castermans, Emilie, Villa, Chiara, Dimopoulos, Aggeliki, Chittiboina, Prashant, Xekouki, Paraskevi, Shah, Nalini, Metzger, Daniel, Lysy, Philippe A, Ferrante, Emanuele, Strebkova, Natalia, Mazerkina, Nadia, Zatelli, Maria Chiara, Lodish, Maya, Horvath, Anelia, de Alexandre, Rodrigo Bertollo, Manning, Allison D, Levy, Isaac, Keil, Margaret F, Sierra, Maria de la Luz, Palmeira, Leonor, Coppieters, Wouter, Georges, Michel, Naves, Luciana A, Jamar, Mauricette, Bours, Vincent, Wu, T. John, Choong, Catherine S, Bertherat, Jerome, Chanson, Philippe, Kamenický, Peter, Farrell, William E, Barlier, Anne, Quezado, Martha, Bjelobaba, Ivana, Stojilkovic, Stanko S, Wess, Jurgen, Costanzi, Stefano, Liu, Pengfei, Lupski, James R, Beckers, Albert, Stratakis, Constantine A
Published in The New England journal of medicine (18.12.2014)
Published in The New England journal of medicine (18.12.2014)
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Web Resource
Beta-cell M 3 muscarinic acetylcholine receptors as potential targets for novel antidiabetic drugs
Zhu, Lu, Rossi, Mario, Doliba, Nicolai M, Wess, Jürgen
Published in International immunopharmacology (01.04.2020)
Published in International immunopharmacology (01.04.2020)
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Journal Article
Beta-cell M3 muscarinic acetylcholine receptors as potential targets for novel antidiabetic drugs
Zhu, Lu, Rossi, Mario, Doliba, Nicolai M., Wess, Jürgen
Published in International immunopharmacology (01.04.2020)
Published in International immunopharmacology (01.04.2020)
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Journal Article
Ultrasonic vocalizations induced by sex and amphetamine in M2, M4, M5 muscarinic and D2 dopamine receptor knockout mice
Wang, Haoran, Liang, Shuyin, Burgdorf, Jeffrey, Wess, Jurgen, Yeomans, John
Published in PloS one (02.04.2008)
Published in PloS one (02.04.2008)
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Journal Article
Muscarinic acetylcholine receptor regulates self-renewal of early erythroid progenitors
Trivedi, Gaurang, Inoue, Daichi, Chen, Cynthia, Bitner, Lillian, Chung, Young Rock, Taylor, Justin, Gönen, Mithat, Wess, Jürgen, Abdel-Wahab, Omar, Zhang, Lingbo
Published in Science translational medicine (25.09.2019)
Published in Science translational medicine (25.09.2019)
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Journal Article
Deletion of M1 Muscarinic Acetylcholine Receptors Increases Amyloid Pathology In Vitro and In Vivo
Davis, Albert A, Fritz, Jason J, Wess, Jurgen, Lah, James J, Levey, Allan I
Published in The Journal of neuroscience (24.03.2010)
Published in The Journal of neuroscience (24.03.2010)
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Journal Article
Allosteric modulation of β-cell M 3 muscarinic acetylcholine receptors greatly improves glucose homeostasis in lean and obese mice
Zhu, Lu, Rossi, Mario, Cohen, Amanda, Pham, Jonathan, Zheng, Hongchao, Dattaroy, Diptadip, Mukaibo, Taro, Melvin, James E, Langel, Jennifer L, Hattar, Samer, Matschinsky, Franz M, Appella, Daniel H, Doliba, Nicolai M, Wess, Jürgen
Published in Proceedings of the National Academy of Sciences - PNAS (10.09.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (10.09.2019)
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Journal Article
Cholinergic Projections to the Substantia Nigra Pars Reticulata Inhibit Dopamine Modulation of Basal Ganglia through the M 4 Muscarinic Receptor
Moehle, Mark S, Pancani, Tristano, Byun, Nellie, Yohn, Samantha E, Wilson, 3rd, George H, Dickerson, Johnathan W, Remke, Daniel H, Xiang, Zixiu, Niswender, Colleen M, Wess, Jürgen, Jones, Carrie K, Lindsley, Craig W, Rook, Jerri M, Conn, P Jeffrey
Published in Neuron (Cambridge, Mass.) (20.12.2017)
Published in Neuron (Cambridge, Mass.) (20.12.2017)
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Journal Article
Hepatic β-arrestin 2 is essential for maintaining euglycemia
Zhu, Lu, Rossi, Mario, Cui, Yinghong, Lee, Regina J, Sakamoto, Wataru, Perry, Nicole A, Urs, Nikhil M, Caron, Marc G, Gurevich, Vsevolod V, Godlewski, Grzegorz, Kunos, George, Chen, Minyong, Chen, Wei, Wess, Jürgen
Published in The Journal of clinical investigation (01.08.2017)
Published in The Journal of clinical investigation (01.08.2017)
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Journal Article
M1 muscarinic allosteric modulators slow prion neurodegeneration and restore memory loss
Bradley, Sophie J, Bourgognon, Julie-Myrtille, Sanger, Helen E, Verity, Nicholas, Mogg, Adrian J, White, David J, Butcher, Adrian J, Moreno, Julie A, Molloy, Colin, Macedo-Hatch, Timothy, Edwards, Jennifer M, Wess, Jurgen, Pawlak, Robert, Read, David J, Sexton, Patrick M, Broad, Lisa M, Steinert, Joern R, Mallucci, Giovanna R, Christopoulos, Arthur, Felder, Christian C, Tobin, Andrew B
Published in The Journal of clinical investigation (01.02.2017)
Published in The Journal of clinical investigation (01.02.2017)
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