Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors
Fucini, Raymond V., Hanan, Emily J., Romanowski, Michael J., Elling, Robert A., Lew, Willard, Barr, Kenneth J., Zhu, Jiang, Yoburn, Joshua C., Liu, Yang, Fahr, Bruce T., Fan, Junfa, Lu, Yafan, Pham, Phuongly, Choong, Ingrid C., VanderPorten, Erica C., Bui, Minna, Purkey, Hans E., Evanchik, Marc J., Yang, Wenjin
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Journal Article
Modifications of the isonipecotic acid fragment of SNS-032 : Analogs with improved permeability and lower efflux ratio
JUNFA FAN, FAHR, Bruce, CHOONG, Ingrid C, STOCKETT, David, CHAN, Erica, CHEETI, Sravanthi, SERAFIMOVA, Iana, YAFAN LU, PHAM, Phuongly, WALKER, Duncan H, HOCH, Ute
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
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Journal Article
A diaminocyclohexyl analog of SNS-032 with improved permeability and bioavailability properties
Choong, Ingrid C., Serafimova, Iana, Fan, Junfa, Stockett, David, Chan, Erica, Cheeti, Sravanthi, Lu, Yafan, Fahr, Bruce, Pham, Phuongly, Arkin, Michelle R., Walker, Duncan H., Hoch, Ute
Published in Bioorganic & medicinal chemistry (01.11.2008)
Published in Bioorganic & medicinal chemistry (01.11.2008)
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Journal Article
Syntheses of β,β-Difluorotryptamines
Deng, Wei-Ping, Nam, Ghilsoo, Fan, Junfa, Kirk, Kenneth L
Published in Journal of organic chemistry (04.04.2003)
Published in Journal of organic chemistry (04.04.2003)
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Journal Article
Optimization of novel reversible Bruton’s tyrosine kinase inhibitors identified using Tethering-fragment-based screens
Hopkins, Brian T., Bame, Eris, Bell, Noah, Bohnert, Tonika, Bowden-Verhoek, Jon K., Bui, Minna, Cancilla, Mark T., Conlon, Patrick, Cullen, Patrick, Erlanson, Daniel A., Fan, Junfa, Fuchs-Knotts, Tarra, Hansen, Stig, Heumann, Stacey, Jenkins, Tracy J., Marcotte, Douglas, McDowell, Bob, Mertsching, Elisabeth, Negrou, Ella, Otipoby, Kevin L., Poreci, Urjana, Romanowski, Michael J., Scott, Daniel, Silvian, Laura, Yang, Wenjin, Zhong, Min
Published in Bioorganic & medicinal chemistry (01.07.2019)
Published in Bioorganic & medicinal chemistry (01.07.2019)
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Journal Article
Utilizing structure based drug design and metabolic soft spot identification to optimize the in vitro potency and in vivo pharmacokinetic properties leading to the discovery of novel reversible Bruton’s tyrosine kinase inhibitors
Hopkins, Brian T., Bame, Eris, Bell, Noah, Bohnert, Tonika, Bowden-Verhoek, Jon K., Bui, Minna, Cancilla, Mark T., Conlon, Patrick, Cullen, Patrick, Erlanson, Daniel A., Fan, Junfa, Fuchs-Knotts, Tarra, Hansen, Stig, Heumann, Stacey, Jenkins, Tracy J., Gua, Chuck, Liu, Ying, Liu, YuTing, Lulla, Mukush, Marcotte, Douglas, Marx, Isaac, McDowell, Bob, Mertsching, Elisabeth, Negrou, Ella, Romanowski, Michael J., Scott, Daniel, Silvian, Laura, Yang, Wenjin, Zhong, Min
Published in Bioorganic & medicinal chemistry (15.08.2021)
Published in Bioorganic & medicinal chemistry (15.08.2021)
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Journal Article
Synthesis of ( E)- and ( Z)-α,β-difluorourocanic acid
Hajduch, Jan, Dolenský, Bohumil, Yoshida, Shinichi, Fan, Junfa, Kirk, Kenneth L.
Published in Journal of fluorine chemistry (01.02.2008)
Published in Journal of fluorine chemistry (01.02.2008)
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Journal Article
In vitro properties of antimicrobial bromotyrosine alkaloids
Pick, Neora, Rawat, Mamta, Arad, Dorit, Lan, Jiong, Fan, Junfa, Kende, Andrew S, Av-Gay, Yossef
Published in Journal of medical microbiology (01.04.2006)
Published in Journal of medical microbiology (01.04.2006)
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Journal Article
CXCR7 antagonists
Fan, Junfa, Lui, Rebecca M, Zhang, Penglie, McMahon, Jeffrey P, Zeng, Yibin, Powers, Jay P, Krasinski, Antoni, Lange, Christopher W
Year of Publication 05.12.2023
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Year of Publication 05.12.2023
Patent
Substituted tetrahydropyrans as CCR2 modulators
Fan, Junfa, Lui, Rebecca M, Zhang, Penglie, McMahon, Jeffrey P, Zeng, Yibin, Powers, Jay P, Kalisiak, Jaroslaw, Mali, Venkat Reddy, Tanaka, Hiroko
Year of Publication 06.08.2024
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Year of Publication 06.08.2024
Patent
CCR2 MODULATORS
MALI, VENKAT REDDY, TANAKA, HIROKO, LUI, REBECCA M, ZENG, YIBIN, FAN, JUNFA, MCMAHON, JEFFREY P, KALISIAK, JAROSLAW, ZHANG, PENGLIE, POWERS, JAY P
Year of Publication 21.05.2024
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Year of Publication 21.05.2024
Patent
Inhibitors of CXCR2
Fan, Junfa, Zhang, Penglie, Malathong, Viengkham, Mali, Venkat, Yu, Chao, Kalisiak, Jaroslaw, Dragoli, Dean R, Tanaka, Hiroko, Yang, Ju, Chen, Xi, Leleti, Manmohan Reddy, McMahon, Jeffrey
Year of Publication 02.04.2024
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Year of Publication 02.04.2024
Patent
Inhibitors of cxcr2
Fan, Junfa, Leleti, Manmohan, Zhang, Penglie, Mcmahon, Jeffrey, Malathong, Viengkham, Mali, Venkat, Yu, Chao, Kalisiak, Jaroslaw, Dragoli, Dean, Yang, Ju, Chen, Xi, Tankaka, Hiroko
Year of Publication 22.03.2024
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Year of Publication 22.03.2024
Patent
Substituted anilines as CCR(4) antagonists
Fan, Junfa, McMahon, Jeffrey P, Li, Yandong, Charvat, Trevor T, Lange, Christopher W, Mali, Venkat Reddy, Punna, Sreenivas, Powers, Jay, Yang, Ju, Leleti, Manmohan Reddy
Year of Publication 30.01.2024
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Year of Publication 30.01.2024
Patent
CCR2 MODULATORS
POWERS, Jay, ZHANG, Penglie, KALISIAK, Jaroslaw, LUI, Rebecca, MALI, Venkat, ZENG, Yibin, FAN, Junfa, MCMAHON, Jeffrey, TANAKA, Hiroko
Year of Publication 28.02.2023
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Year of Publication 28.02.2023
Patent
Ccr2 modulators
Fan, Junfa, Zhang, Penglie, Mcmahon, Jeffrey, Mali, Venkat, Zeng, Yibin, Kalisiak, Jaroslaw, Tanaka, Hiroko, Powers, Jay, Lui, Rebecca
Year of Publication 27.01.2023
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Year of Publication 27.01.2023
Patent