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Published in Journal of the American Chemical Society (03.12.2008)
Published in Journal of the American Chemical Society (03.12.2008)
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Rational Design and Binding Mode Duality of MDM2–p53 Inhibitors
Gonzalez-Lopez de Turiso, Felix, Sun, Daqing, Rew, Yosup, Bartberger, Michael D, Beck, Hilary P, Canon, Jude, Chen, Ada, Chow, David, Correll, Tiffany L, Huang, Xin, Julian, Lisa D, Kayser, Frank, Lo, Mei-Chu, Long, Alexander M, McMinn, Dustin, Oliner, Jonathan D, Osgood, Tao, Powers, Jay P, Saiki, Anne Y, Schneider, Steve, Shaffer, Paul, Xiao, Shou-Hua, Yakowec, Peter, Yan, Xuelei, Ye, Qiuping, Yu, Dongyin, Zhao, Xiaoning, Zhou, Jing, Medina, Julio C, Olson, Steven H
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Published in Journal of medicinal chemistry (23.05.2013)
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Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model
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Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Total Synthesis of (+)-13-Deoxytedanolide
Julian, Lisa D, Newcom, Jason S, Roush, William R
Published in Journal of the American Chemical Society (04.05.2005)
Published in Journal of the American Chemical Society (04.05.2005)
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Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
McMinn, Dustin L., Rew, Yosup, Sudom, Athena, Caille, Seb, DeGraffenreid, Michael, He, Xiao, Hungate, Randall, Jiang, Ben, Jaen, Juan, Julian, Lisa D., Kaizerman, Jacob, Novak, Perry, Sun, Daqing, Tu, Hua, Ursu, Stefania, Walker, Nigel P.C., Yan, Xuelei, Ye, Qiuping, Wang, Zhulun, Powers, Jay P.
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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An Efficient and Scalable One-Pot Double Michael Addition-Dieckmann Condensation for the Synthesis of 4,4-Disubstituted Cyclohexane β-Keto Esters
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Published in Journal of organic chemistry (14.09.2007)
Published in Journal of organic chemistry (14.09.2007)
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CIS-morpholinone and other compounds as MDM2 inhibitors for the treatment of cancer
Yan, Xuelei, Beck, Hilary Plake, Olson, Steven H, Fox, Brian M, Julian, Lisa D, Degraffenreid, Michael R, Roveto, Philip M, Bartberger, Michael D, Sun, Daqing, Gonzalez Lopez De Turiso, Felix, Medina, Julio C, Rew, Yosup, Kayser, Frank
Year of Publication 09.08.2022
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Year of Publication 09.08.2022
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Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model
Julian, Lisa D, Wang, Zhulun, Bostick, Tracy, Caille, Seb, Choi, Rebekah, DeGraffenreid, Michael, Di, Yongmei, He, Xiao, Hungate, Randall W, Jaen, Juan C, Liu, Jinsong, Monshouwer, Mario, McMinn, Dustin, Rew, Yosup, Sudom, Athena, Sun, Daqing, Tu, Hua, Ursu, Stefania, Walker, Nigel, Yan, Xuelei, Ye, Qiuping, Powers, Jay P
Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Year of Publication 13.04.2021
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Year of Publication 13.04.2021
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CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
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Year of Publication 13.12.2018
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Year of Publication 13.12.2018
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Cis-morpholinone and other compounds as MDM2 inhibitors for the treatment of cancer
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Year of Publication 06.09.2018
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Year of Publication 06.09.2018
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Cis-morpholinone and other compounds as MDM2 inhibitors for the treatment of cancer
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Year of Publication 01.03.2018
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Year of Publication 01.03.2018
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CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
OLSON, Steven, H, KAYSER, Frank, BARTBERGER, Michael, D, BECK, Hilary, Plake, REW, Yosup, FOX, Brian, M, JULIAN, Lisa, D, YAN, Xuelei, SUN, Daqing, ROVETO, Philip, M, GONZALEZ LOPEZ DE TURISO, Felix, MEDINA, Julio, C, DEGRAFFENREID, Michael, R
Year of Publication 15.11.2017
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Year of Publication 15.11.2017
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CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
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Year of Publication 07.01.2016
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Year of Publication 07.01.2016
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CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
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Year of Publication 30.12.2015
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Year of Publication 30.12.2015
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