An Aromatic Microdomain at the Cannabinoid CB1 Receptor Constitutes an Agonist/Inverse Agonist Binding Region
McAllister, Sean D, Rizvi, Gulrukh, Anavi-Goffer, Sharon, Hurst, Dow P, Barnett-Norris, Judy, Lynch, Diane L, Reggio, Patricia H, Abood, Mary E
Published in Journal of medicinal chemistry (20.11.2003)
Published in Journal of medicinal chemistry (20.11.2003)
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Journal Article
N-(Piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide (SR141716A) Interaction with LYS 3.28(192) Is Crucial for Its Inverse Agonism at the Cannabinoid CB1 Receptor
Dow P. Hurst, Diane L. Lynch, Judy Barnett-Norris, Stephen M. Hyatt, Herbert H. Seltzman, Miao Zhong, Zhao-Hui Song, Jingjiang Nie, Deborah Lewis, Patricia H. Reggio
Published in Molecular pharmacology (01.12.2002)
Published in Molecular pharmacology (01.12.2002)
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Helix 8 Leu in the CB1 Cannabinoid Receptor Contributes to Selective Signal Transduction Mechanisms
Anavi-Goffer, Sharon, Fleischer, Daniel, Hurst, Dow P., Lynch, Diane L., Barnett-Norris, Judy, Shi, Shanping, Lewis, Deborah L., Mukhopadhyay, Somnath, Howlett, Allyn C., Reggio, Patricia H., Abood, Mary E.
Published in The Journal of biological chemistry (24.08.2007)
Published in The Journal of biological chemistry (24.08.2007)
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Journal Article
Cysteine 2.59(89) in the Second Transmembrane Domain of Human CB2 Receptor Is Accessible within the Ligand Binding Crevice: Evidence for Possible CB2 Deviation from a Rhodopsin Template
Rundong Zhang, Dow P. Hurst, Judy Barnett-Norris, Patricia H. Reggio, Zhao-Hui Song
Published in Molecular pharmacology (01.07.2005)
Published in Molecular pharmacology (01.07.2005)
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Agonist alkyl tail interaction with cannabinoid CB1 receptor V6.43/I6.46 groove induces a helix 6 active conformation
Barnett-Norris, Judy, Hurst, Dow P., Buehner, Kurt, Ballesteros, Juan A., Guarnieri, Frank, Reggio, Patricia H.
Published in International journal of quantum chemistry (2002)
Published in International journal of quantum chemistry (2002)
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Journal Article
Structural mimicry in class A G protein-coupled receptor rotamer toggle switches: the importance of the F3.36(201)/W6.48(357) interaction in cannabinoid CB1 receptor activation
McAllister, Sean D, Hurst, Dow P, Barnett-Norris, Judy, Lynch, Diane, Reggio, Patricia H, Abood, Mary E
Published in The Journal of biological chemistry (12.11.2004)
Published in The Journal of biological chemistry (12.11.2004)
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Journal Article
A critical role for a tyrosine residue in the cannabinoid receptors for ligand recognition
McAllister, Sean D., Tao, Qing, Barnett-Norris, Judy, Buehner, Kurt, Hurst, Dow P., Guarnieri, Frank, Reggio, Patricia H., Nowell Harmon, Katharine W., Cabral, Guy A., Abood, Mary E.
Published in Biochemical pharmacology (15.06.2002)
Published in Biochemical pharmacology (15.06.2002)
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Journal Article
Helix 8 Leu in the CB sub(1) Cannabinoid Receptor Contributes to Selective Signal Transduction Mechanisms
Anavi-Goffer, Sharon, Fleischer, Daniel, Hurst, Dow P, Lynch, Diane L, Barnett-Norris, Judy, Shi, Shanping, Lewis, Deborah L, Mukhopadhyay, Somnath, Howlett, Allyn C, Reggio, Patricia H, Abood, Mary E
Published in The Journal of biological chemistry (01.08.2007)
Get full text
Published in The Journal of biological chemistry (01.08.2007)
Journal Article
Structural Mimicry in Class A G Protein-coupled Receptor Rotamer Toggle Switches: The Importance of the F3.36(201)/W6.48(357) Interaction in Cannabinoid CB sub(1) Receptor Activation
Mcallister, Sean D, Hurst, Dow P, Barnett-Norris, Judy, Lynch, Diane, Reggio, Patricia H, Abood, Mary E
Published in The Journal of biological chemistry (12.11.2004)
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Published in The Journal of biological chemistry (12.11.2004)
Journal Article
An aromatic microdomain at the cannabinoid CB(1) receptor constitutes an agonist/inverse agonist binding region
McAllister, Sean D, Rizvi, Gulrukh, Anavi-Goffer, Sharon, Hurst, Dow P, Barnett-Norris, Judy, Lynch, Diane L, Reggio, Patricia H, Abood, Mary E
Published in Journal of medicinal chemistry (20.11.2003)
Get full text
Published in Journal of medicinal chemistry (20.11.2003)
Journal Article
An Aromatic Microdomain at the Cannabinoid CB 1 Receptor Constitutes an Agonist/Inverse Agonist Binding Region
McAllister, Sean D., Rizvi, Gulrukh, Anavi-Goffer, Sharon, Hurst, Dow P., Barnett-Norris, Judy, Lynch, Diane L., Reggio, Patricia H., Abood, Mary E.
Published in Journal of medicinal chemistry (01.11.2003)
Published in Journal of medicinal chemistry (01.11.2003)
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Journal Article
The Bioactive Conformation of Aminoalkylindoles at the Cannabinoid CB1 and CB2 Receptors: Insights Gained from (E)- and (Z)-Naphthylidene Indenes
Reggio, Patricia H, Basu-Dutt, Sharmista, Barnett-Norris, Judy, Castro, Marie T, Hurst, Dow P, Seltzman, Herbert H, Roche, Michael J, Gilliam, Anne F, Thomas, Brian F, Stevenson, L. A, Pertwee, Roger G, Abood, Mary E
Published in Journal of medicinal chemistry (17.12.1998)
Published in Journal of medicinal chemistry (17.12.1998)
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Journal Article
N -(Piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1 H -pyrazole-3-carboxamide (SR141716A) Interaction with LYS 3.28(192) Is Crucial for Its Inverse Agonism at the Cannabinoid CB1 Receptor
Hurst, Dow P., Lynch, Diane L., Barnett-Norris, Judy, Hyatt, Stephen M., Seltzman, Herbert H., Zhong, Miao, Song, Zhao-Hui, Nie, Jingjiang, Lewis, Deborah, Reggio, Patricia H.
Published in Molecular pharmacology (01.12.2002)
Published in Molecular pharmacology (01.12.2002)
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Journal Article