Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Judge, Russell A., Sridar, Janani, Tunyasuvunakool, Kathryn, Jain, Rinku, Wang, John C. K., Ouch, Christna, Xu, Jun, Mafi, Amirhossein, Nile, Aaron H., Remarcik, Clint, Smith, Corey L., Ghosh, Crystal, Xu, Chen, Stoll, Vincent, Jumper, John, Singh, Amoolya H., Eaton, Dan, Hao, Qi
Published in Nature communications (20.09.2022)
Published in Nature communications (20.09.2022)
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Journal Article
Author Correction: Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Judge, Russell A., Sridar, Janani, Tunyasuvunakool, Kathryn, Jain, Rinku, Wang, John C. K., Ouch, Christna, Xu, Jun, Mafi, Amirhossein, Nile, Aaron H., Remarcik, Clint, Smith, Corey L., Ghosh, Crystal, Xu, Chen, Stoll, Vincent, Jumper, John, Singh, Amoolya H., Eaton, Dan, Hao, Qi
Published in Nature communications (28.09.2022)
Published in Nature communications (28.09.2022)
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Journal Article
Cryo-EM structure of human PAPP-A2 and mechanism of substrate recognition
Sridar, Janani, Mafi, Amirhossein, Judge, Russell A., Xu, Jun, Kong, Kailyn A., Wang, John C. K., Stoll, Vincent S., Koukos, Georgios, Simon, Reyna J., Eaton, Dan, Bratkowski, Matthew, Hao, Qi
Published in Communications chemistry (28.10.2023)
Published in Communications chemistry (28.10.2023)
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Journal Article
Selective MCL-1 inhibitor ABBV-467 is efficacious in tumor models but is associated with cardiac troponin increases in patients
Yuda, Junichiro, Will, Christine, Phillips, Darren C., Abraham, Linu, Alvey, Cory, Avigdor, Abraham, Buck, Wayne, Besenhofer, Lauren, Boghaert, Erwin, Cheng, Dong, Cojocari, Dan, Doyle, Kelly, Hansen, T. Matthew, Huang, Kevin, Johnson, Eric F., Judd, Andrew S., Judge, Russell A., Kalvass, John C., Kunzer, Aaron, Lam, Lloyd T., Li, Rachel, Martin, Ruth L., Mastracchio, Anthony, Mitten, Mike, Petrich, Adam, Wang, Jin, Ward, James E., Zhang, Haichao, Wang, Xilu, Wolff, Johannes E., Bell-McGuinn, Katherine M., Souers, Andrew J.
Published in Communications medicine (25.10.2023)
Published in Communications medicine (25.10.2023)
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Journal Article
Neutron structure of the cyclic glucose-bound xylose isomerase E186Q mutant
Munshi, Parthapratim, Snell, Edward H., van der Woerd, Mark J., Judge, Russell A., Myles, Dean A. A., Ren, Zhong, Meilleur, Flora
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
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Journal Article
CD40/anti-CD40 antibody complexes which illustrate agonist and antagonist structural switches
Argiriadi, Maria A, Benatuil, Lorenzo, Dubrovska, Ievgeniia, Egan, David A, Gao, Lei, Greischar, Amy, Hardman, Jennifer, Harlan, John, Iyer, Ramesh B, Judge, Russell A, Lake, Marc, Perron, Denise C, Sadhukhan, Ramkrishna, Sielaff, Bernhard, Sousa, Silvino, Wang, Rui, McRae, Bradford L
Published in BMC molecular and cell biology (05.08.2019)
Published in BMC molecular and cell biology (05.08.2019)
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Journal Article
Minimising the payload solvent exposed hydrophobic surface area optimises the antibody-drug conjugate properties
Hobson, Adrian D, Zhu, Haizhong, Qiu, Wei, Judge, Russell A, Longenecker, Kenton
Published in MedChemComm (20.03.2024)
Published in MedChemComm (20.03.2024)
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Journal Article
Microgravity and Macromolecular Crystallography
Kundrot, Craig E, Judge, Russell A, Pusey, Marc L, Snell, Edward H
Published in Crystal growth & design (01.01.2001)
Published in Crystal growth & design (01.01.2001)
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Journal Article
Structure-Guided Design of a Series of MCL‑1 Inhibitors with High Affinity and Selectivity
Bruncko, Milan, Wang, Le, Sheppard, George S, Phillips, Darren C, Tahir, Stephen K, Xue, John, Erickson, Scott, Fidanze, Steve, Fry, Elizabeth, Hasvold, Lisa, Jenkins, Gary J, Jin, Sha, Judge, Russell A, Kovar, Peter J, Madar, David, Nimmer, Paul, Park, Chang, Petros, Andrew M, Rosenberg, Saul H, Smith, Morey L, Song, Xiaohong, Sun, Chaohong, Tao, Zhi-Fu, Wang, Xilu, Xiao, Yu, Zhang, Haichao, Tse, Chris, Leverson, Joel D, Elmore, Steven W, Souers, Andrew J
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Journal Article
Inhibition of MALT1 and BCL2 Induces Synergistic Antitumor Activity in Models of B-Cell Lymphoma
Plotnik, Joshua P., Richardson, Adam E., Yang, Haopeng, Rojas, Estela, Bontcheva, Velitchka, Dowell, Colleen, Parsons, Sydney, Wilson, Ashley, Ravanmehr, Vida, Will, Christine, Jung, Paul, Zhu, Haizhong, Partha, Sarathy Karunan, Panchal, Sanjay C., Mali, Raghuveer Singh, Kohlhapp, Frederick J., McClure, Ryan A., Ramathal, Cyril Y., George, Mariam D., Jhala, Manisha, Elsen, Nathaniel L., Qiu, Wei, Judge, Russell A., Pan, Chin, Mastracchio, Anthony, Henderson, Jared, Meulbroek, Jonathan A., Green, Michael R., Pappano, William N.
Published in Molecular cancer therapeutics (02.07.2024)
Published in Molecular cancer therapeutics (02.07.2024)
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Journal Article
The Effect of Temperature and Solution pH on the Nucleation of Tetragonal Lysozyme Crystals
Judge, Russell A., Jacobs, Randolph S., Frazier, Tyralynn, Snell, Edward H., Pusey, Marc L.
Published in Biophysical journal (01.09.1999)
Published in Biophysical journal (01.09.1999)
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Journal Article
Discovery of a Potent and Selective BCL‑XL Inhibitor with in Vivo Activity
Tao, Zhi-Fu, Hasvold, Lisa, Wang, Le, Wang, Xilu, Petros, Andrew M, Park, Chang H, Boghaert, Erwin R, Catron, Nathaniel D, Chen, Jun, Colman, Peter M, Czabotar, Peter E, Deshayes, Kurt, Fairbrother, Wayne J, Flygare, John A, Hymowitz, Sarah G, Jin, Sha, Judge, Russell A, Koehler, Michael F. T, Kovar, Peter J, Lessene, Guillaume, Mitten, Michael J, Ndubaku, Chudi O, Nimmer, Paul, Purkey, Hans E, Oleksijew, Anatol, Phillips, Darren C, Sleebs, Brad E, Smith, Brian J, Smith, Morey L, Tahir, Stephen K, Watson, Keith G, Xiao, Yu, Xue, John, Zhang, Haichao, Zobel, Kerry, Rosenberg, Saul H, Tse, Chris, Leverson, Joel D, Elmore, Steven W, Souers, Andrew J
Published in ACS medicinal chemistry letters (09.10.2014)
Published in ACS medicinal chemistry letters (09.10.2014)
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Journal Article
Tetragonal Chicken Egg White Lysozyme Solubility in Sodium Chloride Solutions
Forsythe, Elizabeth L, Judge, Russell A, Pusey, Marc L
Published in Journal of chemical and engineering data (01.05.1999)
Published in Journal of chemical and engineering data (01.05.1999)
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Journal Article
Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure-Based Drug Design
Hobson, Adrian D, Judge, Russell A, Aguirre, Ana L, Brown, Brian S, Cui, Yifang, Ding, Ping, Dominguez, Eric, DiGiammarino, Enrico, Egan, David A, Freiberg, Gail M, Gopalakrishnan, Sujatha M, Harris, Christopher M, Honore, Marie P, Kage, Karen L, Kapecki, Nicolas J, Ling, Christopher, Ma, Junli, Mack, Helmut, Mamo, Mulugeta, Maurus, Stefan, McRae, Bradford, Moore, Nigel S, Mueller, Bernhard K, Mueller, Reinhold, Namovic, Marian T, Patel, Kaushal, Pratt, Steve D, Putman, C. Brent, Queeney, Kara L, Sarris, Kathy K, Schaffter, Lisa M, Stoll, Vincent, Vasudevan, Anil, Wang, Lei, Wang, Lu, Wirthl, William, Yach, Kimberly
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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Journal Article
An anti-PD-1-GITR-L bispecific agonist induces GITR clustering-mediated T cell activation for cancer immunotherapy
Chan, Sarah, Belmar, Nicole, Ho, Sun, Rogers, Bryan, Stickler, Marcia, Graham, Michelle, Lee, Eileen, Tran, Ninian, Zhang, Dong, Gupta, Priyanka, Sho, Mien, MacDonough, Tracy, Woolley, Andrew, Kim, Han, Zhang, Hong, Liu, Wei, Zheng, Pingping, Dezso, Zoltan, Halliwill, Kyle, Ceccarelli, Michele, Rhodes, Susan, Thakur, Archana, Forsyth, Charles M, Xiong, Mengli, Tan, Siu Sze, Iyer, Ramesh, Lake, Marc, Digiammarino, Enrico, Zhou, Li, Bigelow, Lance, Longenecker, Kenton, Judge, Russell A, Liu, Cassie, Trumble, Max, Remis, Jonathan P, Fox, Melvin, Cairns, Belinda, Akamatsu, Yoshiko, Hollenbaugh, Diane, Harding, Fiona, Alvarez, Hamsell M
Published in Nature cancer (01.03.2022)
Published in Nature cancer (01.03.2022)
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Journal Article
Targeting lysine specific demethylase 4A (KDM4A) tandem TUDOR domain – A fragment based approach
Upadhyay, Anup K., Judge, Russell A., Li, Leiming, Pithawalla, Ron, Simanis, Justin, Bodelle, Pierre M., Marin, Violeta L., Henry, Rodger F., Petros, Andrew M., Sun, Chaohong
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
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Journal Article
Expanding the Repertoire for "Large Small Molecules": Prodrug ABBV-167 Efficiently Converts to Venetoclax with Reduced Food Effect in Healthy Volunteers
Salem, Ahmed Hamed, Tao, Zhi-Fu, Bueno, Orlando F, Chen, Jie, Chen, Shuang, Edalji, Rohinton, Elmore, Steven W, Fournier, Keith M, Harper, Kaid C, Hong, Richard, Jenkins, Gary J, Ji, Jianguo, Judge, Russell A, Kalvass, John C, Klix, Russell C, Ku, Yi-Yin, Leverson, Joel D, Marks, Richard A, Marsh, Kennan C, Menon, Rajeev M, Park, Chang H, Phillips, Darren C, Pu, Yu-Ming, Rosenberg, Saul H, Sanzgiri, Yeshwant D, Sheikh, Ahmad Y, Shi, Yi, Stolarik, Deanne, Suleiman, Ahmed A, Wang, Xilu, Zhang, Geoff G Z, Catron, Nathaniel D, Souers, Andrew J
Published in Molecular cancer therapeutics (01.06.2021)
Published in Molecular cancer therapeutics (01.06.2021)
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