Search Results - "Jourdan, Fabrice" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Quinazolinone-Based Anticancer Agents: Synthesis, Antiproliferative SAR, Antitubulin Activity, and Tubulin Co-crystal Structure

Quinazolinone-Based Anticancer Agents: Synthesis, Antiproliferative SAR, Antitubulin Activity, and Tubulin Co-crystal Structure

by Dohle, Wolfgang, Jourdan, Fabrice L, Menchon, Grégory, Prota, Andrea E, Foster, Paul A, Mannion, Pascoe, Hamel, Ernest, Thomas, Mark P, Kasprzyk, Philip G, Ferrandis, Eric, Steinmetz, Michel O, Leese, Mathew P, Potter, Barry V. L
Published in Journal of medicinal chemistry (08.02.2018)

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Optimisation of Tetrahydroisoquinoline-Based Chimeric Microtubule Disruptors

Optimisation of Tetrahydroisoquinoline-Based Chimeric Microtubule Disruptors

by Dohle, Wolfgang, Leese, Mathew P., Jourdan, Fabrice L., Chapman, Christopher J., Hamel, Ernest, Ferrandis, Eric, Potter, Barry V. L.
Published in ChemMedChem (01.08.2014)

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Synthesis, Anti-tubulin and Antiproliferative SAR of Steroidomimetic Dihydroisoquinolinones

Synthesis, Anti-tubulin and Antiproliferative SAR of Steroidomimetic Dihydroisoquinolinones

by Leese, Mathew P., Jourdan, Fabrice L., Major, Meriel R., Dohle, Wolfgang, Thomas, Mark P., Hamel, Ernest, Ferrandis, Eric, Mahon, Mary F., Newman, Simon P., Purohit, Atul, Potter, Barry V. L.
Published in ChemMedChem (01.04.2014)

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Structure–Activity Relationships of C-17 Cyano-Substituted Estratrienes as Anticancer Agents

Structure–Activity Relationships of C-17 Cyano-Substituted Estratrienes as Anticancer Agents

by Leese, Mathew P, Jourdan, Fabrice L, Gaukroger, Keira, Mahon, Mary F, Newman, Simon P, Foster, Paul A, Stengel, Chloe, Regis-Lydi, Sandra, Ferrandis, Eric, Fiore, Anna Di, De Simone, Giuseppina, Supuran, Claudiu T, Purohit, Atul, Reed, Michael J, Potter, Barry V. L
Published in Journal of medicinal chemistry (13.03.2008)

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Tetrahydroisoquinolinone-Based Steroidomimetic and Chimeric Microtubule Disruptors

Tetrahydroisoquinolinone-Based Steroidomimetic and Chimeric Microtubule Disruptors

by Leese, Mathew P., Jourdan, Fabrice L., Major, Meriel R., Dohle, Wolfgang, Hamel, Ernest, Ferrandis, Eric, Fiore, Ann, Kasprzyk, Philip G., Potter, Barry V. L.
Published in ChemMedChem (01.01.2014)

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Synthesis, Antitubulin, and Antiproliferative SAR of C3/C1-Substituted Tetrahydroisoquinolines

Synthesis, Antitubulin, and Antiproliferative SAR of C3/C1-Substituted Tetrahydroisoquinolines

by Dohle, Wolfgang, Leese, Mathew P., Jourdan, Fabrice L., Major, Meriel R., Bai, Ruoli, Hamel, Ernest, Ferrandis, Eric, Kasprzyk, Philip G., Fiore, Ann, Newman, Simon P., Purohit, Atul, Potter, Barry V. L.
Published in ChemMedChem (01.02.2014)

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Cover Picture: Tetrahydroisoquinolinone-Based Steroidomimetic and Chimeric Microtubule Disruptors (ChemMedChem 1/2014)

Cover Picture: Tetrahydroisoquinolinone-Based Steroidomimetic and Chimeric Microtubule Disruptors (ChemMedChem 1/2014)

by Leese, Mathew P., Jourdan, Fabrice L., Major, Meriel R., Dohle, Wolfgang, Hamel, Ernest, Ferrandis, Eric, Fiore, Ann, Kasprzyk, Philip G., Potter, Barry V. L.
Published in ChemMedChem (01.01.2014)

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AMPA AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS

AMPA AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS

by CHEN GANG, JOURDAN FABRICE LOIC, AMERIKS MICHAEL K, LIN DAVID WEI, BERRY CYNTHIA G.B, RAVULA SUCHITRA, SAVALL BRADLEY M, SWANSON DEVIN M, PENA PINON MIGUEL ANGEL, WU DONGPEI, ZHANG WEI, LEBOLD TERRY PATRICK
Year of Publication 08.02.2024

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Patent

1,3,5‐Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu2/3 Receptors

1,3,5‐Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu2/3 Receptors

by Van Gool, Michiel, Alonso De Diego, Sergio A., Delgado, Oscar, Trabanco, Andrés A., Jourdan, Fabrice, Macdonald, Gregor J., Somers, Marijke, Ver Donck, Luc
Published in ChemMedChem (21.06.2017)

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Journal Article

1,3,5-Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu 2/3 Receptors

1,3,5-Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu 2/3 Receptors

by Van Gool, Michiel, Alonso De Diego, Sergio A, Delgado, Oscar, Trabanco, Andrés A, Jourdan, Fabrice, Macdonald, Gregor J, Somers, Marijke, Ver Donck, Luc
Published in ChemMedChem (21.06.2017)

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Synthesis, Antitubulin, and Antiproliferative SAR of Analogues of 2-Methoxyestradiol-3,17-O,O-bis-sulfamate

Synthesis, Antitubulin, and Antiproliferative SAR of Analogues of 2-Methoxyestradiol-3,17-O,O-bis-sulfamate

by Jourdan, Fabrice, Leese, Mathew P, Dohle, Wolfgang, Hamel, Ernest, Ferrandis, Eric, Newman, Simon P, Purohit, Atul, Reed, Michael J, Potter, Barry V. L
Published in Journal of medicinal chemistry (08.04.2010)

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Structure–Activity Relationships of C-17-Substituted Estratriene-3-O-sulfamates as Anticancer Agents

Structure–Activity Relationships of C-17-Substituted Estratriene-3-O-sulfamates as Anticancer Agents

by Jourdan, Fabrice, Leese, Mathew P, Dohle, Wolfgang, Ferrandis, Eric, Newman, Simon P, Chander, Surinder, Purohit, Atul, Potter, Barry V. L
Published in Journal of medicinal chemistry (14.07.2011)

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Chimeric microtubule disruptors

Chimeric microtubule disruptors

by Leese, Mathew P., Jourdan, Fabrice, Kimberley, Meriel R., Cozier, Gyles E., Thiyagarajan, Nethaji, Stengel, Chloe, Regis-Lydi, Sandra, Foster, Paul A., Newman, Simon P., Acharya, K. Ravi, Ferrandis, Eric, Purohit, Atul, Reed, Michael J., Potter, Barry V. L.
Published in Chemical communications (Cambridge, England) (01.01.2010)

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Steroidomimetic Tetrahydroisoquinolines for the Design of New Microtubule Disruptors

Steroidomimetic Tetrahydroisoquinolines for the Design of New Microtubule Disruptors

by Leese, Mathew P, Jourdan, Fabrice, Dohle, Wolfgang, Kimberley, Meriel R, Thomas, Mark P, Bai, Ruoli, Hamel, Ernest, Ferrandis, Eric, Potter, Barry V. L
Published in ACS medicinal chemistry letters (12.01.2012)

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Journal Article

Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling

Effects of C-17 heterocyclic substituents on the anticancer activity of 2-ethylestra-1,3,5(10)-triene-3-O-sulfamates: synthesis, in vitro evaluation and computational modelling

by Jourdan, Fabrice, Bubert, Christian, Leese, Mathew P., Smith, Andrew, Ferrandis, Eric, Regis-Lydi, Sandra, Newman, Simon P., Purohit, Atul, Reed, Michael J., Potter, Barry V. L.
Published in Organic & biomolecular chemistry (01.01.2008)

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Purification and Characterization of the Fe II - and α-Ketoglutarate-Dependent Xanthine Hydroxylase from Aspergillus nidulans

Purification and Characterization of the Fe II - and α-Ketoglutarate-Dependent Xanthine Hydroxylase from Aspergillus nidulans

by Montero-Morán, Gabriela M., Li, Meng, Rendòn-Huerta, Erika, Jourdan, Fabrice, Lowe, David J., Stumpff-Kane, Andrew W., Feig, Michael, Scazzocchio, Claudio, Hausinger, Robert P.
Published in Biochemistry (Easton) (08.05.2007)

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아자벤즈이미다졸 및 AMPA 수용체 조절제로서의 이의 용도

아자벤즈이미다졸 및 AMPA 수용체 조절제로서의 이의 용도

by CHEN GANG, JOURDAN FABRICE LOIC, AMERIKS MICHAEL K, LIN DAVID WEI, BERRY CYNTHIA G.B, RAVULA SUCHITRA, SAVALL BRADLEY M, SWANSON DEVIN M, PENA PINON MIGUEL ANGEL, WU DONGPEI, ZHANG WEI, LEBOLD TERRY PATRICK
Year of Publication 20.12.2017

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Patent

Abstract 756: Optimization of tetrahydroisoquinoline-based microtubule disruptors as anticancer agents

Abstract 756: Optimization of tetrahydroisoquinoline-based microtubule disruptors as anticancer agents

by Leese, Mathew P., Jourdan, Fabrice L., Ferrandis, Eric, Regis-Lydi, Sandra, Kasprzyk, Philip G., Fiore, Ann, Newman, Simon P., Stengel, Chloe, Reed, Michael J., Purohit, Atul, Potter, Barry VL
Published in Cancer research (Chicago, Ill.) (15.04.2010)

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Journal Article

Chimeric microtubule disruptorsElectronic supplementary information (ESI) available: Synthetic, spectroscopic and crystallographic details are provided [crystallographic data pdb accession code 2WD2.pdb]. See DOI: 10.1039/c002558e

Chimeric microtubule disruptorsElectronic supplementary information (ESI) available: Synthetic, spectroscopic and crystallographic details are provided [crystallographic data pdb accession code 2WD2.pdb]. See DOI: 10.1039/c002558e

by Leese, Mathew P, Jourdan, Fabrice, Kimberley, Meriel R, Cozier, Gyles E, Thiyagarajan, Nethaji, Stengel, Chloe, Regis-Lydi, Sandra, Foster, Paul A, Newman, Simon P, Acharya, K. Ravi, Ferrandis, Eric, Purohit, Atul, Reed, Michael J, Potter, Barry V. L
Year of Publication 13.04.2010

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A left-handed α-helix containing both L- and D-amino acids: The solution structure of the antimicrobial lipodepsipeptide tolaasin

A left-handed α-helix containing both L- and D-amino acids: The solution structure of the antimicrobial lipodepsipeptide tolaasin

by Jourdan, Fabrice, Lazzaroni, Silvia, Méndez, Blanca López, Lo Cantore, Pietro, de Julio, Marianna, Amodeo, Pietro, Iacobellis, Nicola S., Evidente, Antonio, Motta, Andrea
Published in Proteins, structure, function, and bioinformatics (01.09.2003)

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