Development of novel benznidazole formulations: Physicochemical characterization and in vivo evaluation on parasitemia reduction in Chagas disease
Palmeiro-Roldán, Ricardo, Fonseca-Berzal, Cristina, Gómez-Barrio, Alicia, Arán, Vicente J., Escario, José A., Torrado-Durán, Susana, Torrado-Santiago, Santiago
Published in International journal of pharmaceutics (10.09.2014)
Published in International journal of pharmaceutics (10.09.2014)
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Journal Article
5-Nitroindazole-based compounds: further studies for activity optimization as anti-Trypanosoma cruzi agents
Fonseca-Berzal, Cristina, Ibáñez-Escribano, Alexandra, de Castro, Sonia, Escario, José A., Gómez-Barrio, Alicia, Arán, Vicente J.
Published in Acta tropica (01.10.2022)
Published in Acta tropica (01.10.2022)
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Journal Article
Selective activity of 2,4-diaryl-1,2,3,4-tetrahydroquinolines on Trypanosoma cruzi epimastigotes and amastigotes expressing β-galactosidase
Fonseca-Berzal, Cristina, Merchán Arenas, Diego R., Romero Bohórquez, Arnold R., Escario, José A., Kouznetsov, Vladimir V., Gómez-Barrio, Alicia
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
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Journal Article
In vitro phenotypic screening of 7-chloro-4-amino(oxy)quinoline derivatives as putative anti-Trypanosoma cruzi agents
Fonseca-Berzal, Cristina, Rojas Ruiz, Fernando A, Escario, José A, Kouznetsov, Vladimir V, Gómez-Barrio, Alicia
Published in Bioorganic & medicinal chemistry letters (15.02.2014)
Published in Bioorganic & medicinal chemistry letters (15.02.2014)
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Journal Article
Novel solid dispersions of benznidazole: Preparation, dissolution profile and biological evaluation as alternative antichagasic drug delivery system
Fonseca-Berzal, Cristina, Palmeiro-Roldán, Ricardo, Escario, José A., Torrado, Susana, Arán, Vicente J., Torrado-Santiago, Santiago, Gómez-Barrio, Alicia
Published in Experimental parasitology (01.02.2015)
Published in Experimental parasitology (01.02.2015)
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Journal Article
Novel Imidazo[4,5-c][1,2,6]thiadiazine 2,2-dioxides as antiproliferative trypanosoma cruzi drugs: Computational screening from neural network, synthesis and in vivo biological properties
Guerra, Angela, Gonzalez-Naranjo, Pedro, Campillo, Nuria E., Varela, Javier, Lavaggi, María L., Merlino, Alicia, Cerecetto, Hugo, González, Mercedes, Gomez-Barrio, Alicia, Escario, José A., Fonseca-Berzal, Cristina, Yaluf, Gloria, Paniagua-Solis, Jorge, Páez, Juan A.
Published in European journal of medicinal chemistry (18.08.2017)
Published in European journal of medicinal chemistry (18.08.2017)
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Journal Article
Bond-based bilinear indices for computational discovery of novel trypanosomicidal drug-like compounds through virtual screening
Castillo-Garit, Juan Alberto, del Toro-Cortés, Oremia, Vega, Maria C., Rolón, Miriam, Rojas de Arias, Antonieta, Casañola-Martin, Gerardo M., Escario, José A., Gómez-Barrio, Alicia, Marrero-Ponce, Yovani, Torrens, Francisco, Abad, Concepción
Published in European journal of medicinal chemistry (26.05.2015)
Published in European journal of medicinal chemistry (26.05.2015)
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Journal Article
Biological approaches to characterize the mode of action of two 5-nitroindazolinone prototypes on Trypanosoma cruzi bloodstream trypomastigotes
FONSECA-BERZAL, CRISTINA, DA SILVA, CRISTIANE FRANÇA, MENNA-BARRETO, RUBEM F. S., BATISTA, MARCOS MEUSER, ESCARIO, JOSÉ A., ARÁN, VICENTE J., GÓMEZ-BARRIO, ALICIA, SOEIRO, MARIA DE NAZARÉ C.
Published in Parasitology (01.09.2016)
Published in Parasitology (01.09.2016)
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Journal Article
Drug repositioning for novel antitrichomonas from known antiprotozoan drugs using hierarchical screening
Meneses-Marcel, Alfredo, Marrero-Ponce, Yovani, Ibáñez-Escribano, Alexandra, Gómez-Barrio, Alicia, Escario, José A, Barigye, Stephen J, Terán, Enrique, García-Jacas, Cesar R, Machado-Tugores, Yanetsy, Nogal-Ruiz, Juan J, Arán-Redó, Vicente J
Published in Future medicinal chemistry (01.04.2018)
Published in Future medicinal chemistry (01.04.2018)
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Journal Article
Selective activity of polyene macrolides produced by genetically modified Streptomyces on Trypanosoma cruzi
Rolón, Miriam, Seco, Elena M., Vega, Celeste, Nogal, Juan J., Escario, José A., Gómez-Barrio, Alicia, Malpartida, Francisco
Published in International journal of antimicrobial agents (01.08.2006)
Published in International journal of antimicrobial agents (01.08.2006)
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Journal Article
Ligand-based discovery of novel trypanosomicidal drug-like compounds: In silico identification and experimental support
Castillo-Garit, Juan Alberto, Vega, Maria Celeste, Rolón, Miriam, Marrero-Ponce, Yovani, Gómez-Barrio, Alicia, Escario, José A., Bello, Alfredo Alvarez, Montero, Alina, Torrens, Francisco, Pérez-Giménez, Facundo, Arán, Vicente J., Abad, Concepción
Published in European journal of medicinal chemistry (01.08.2011)
Published in European journal of medicinal chemistry (01.08.2011)
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Journal Article
Identification In Silico and In Vitro of Novel Trypanosomicidal Drug-Like Compounds
Castillo-Garit, Juan A., del Toro-Cortés, Oremia, Kouznetsov, Vladimir V., Puentes, Cristian Ochoa, Romero Bohórquez, Arnold R., Vega, Maria C., Rolón, Miriam, Escario, José A., Gómez-Barrio, Alicia, Marrero-Ponce, Yovani, Torrens, Francisco, Abad, Concepción
Published in Chemical biology & drug design (01.07.2012)
Published in Chemical biology & drug design (01.07.2012)
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Journal Article
Activity profile of two 5-nitroindazole derivatives over the moderately drug-resistant Trypanosoma cruzi Y strain (DTU TcII): in vitro and in vivo studies
Fonseca-Berzal, Cristina, da Silva, Cristiane França, Batista, Denise da Gama Jaen, de Oliveira, Gabriel Melo, Cumella, José, Batista, Marcos Meuser, Peres, Raiza Brandão, Silva da Gama Nefertiti, Aline, Escario, José A., Gómez-Barrio, Alicia, Arán, Vicente J., Soeiro, Maria de Nazaré Correia
Published in Parasitology (01.09.2020)
Published in Parasitology (01.09.2020)
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Journal Article
Biological Characterization of Trypanosoma cruzi Strains
Rafael A Martínez-Díaz, José A Escario, Juan J Nogal-Ruiz, Alicia Gómez-Barrio
Published in Memórias do Instituto Oswaldo Cruz (01.01.2001)
Published in Memórias do Instituto Oswaldo Cruz (01.01.2001)
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Journal Article
Antiparasitic properties of homoallylamines and related compounds
Gómez-Barrio, Alicia, Montero-Pereira, David, Nogal-Ruiz, Juan, Escario, José, Muelas-Serrano, Susana, Kouznetsov, Vladimir, Vargas Méndez, Leonor, Urbina Gonzáles, Juan, Ochoa, Carmen
Published in Acta parasitologica (01.03.2006)
Published in Acta parasitologica (01.03.2006)
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Journal Article
Antiprotozoan lead discovery by aligning dry and wet screening: Prediction, synthesis, and biological assay of novel quinoxalinones
Martins Alho, Miriam A., Marrero-Ponce, Yovani, Barigye, Stephen J., Meneses-Marcel, Alfredo, Machado Tugores, Yanetsy, Montero-Torres, Alina, Gómez-Barrio, Alicia, Nogal, Juan J., García-Sánchez, Rory N., Vega, María Celeste, Rolón, Miriam, Martínez-Fernández, Antonio R., Escario, José A., Pérez-Giménez, Facundo, Garcia-Domenech, Ramón, Rivera, Norma, Mondragón, Ricardo, Mondragón, Mónica, Ibarra-Velarde, Froylán, Lopez-Arencibia, Atteneri, Martín-Navarro, Carmen, Lorenzo-Morales, Jacob, Cabrera-Serra, Maria Gabriela, Piñero, Jose, Tytgat, Jan, Chicharro, Roberto, Arán, Vicente J.
Published in Bioorganic & medicinal chemistry (01.03.2014)
Published in Bioorganic & medicinal chemistry (01.03.2014)
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Journal Article
Saponinas esteroidales de la planta Agave brittoniana (Agavaceae) con actividad contra el parásito Trichomona vaginalis
José Orestes Guerra, Alfredo Meneses, Ana María Simonet, Francisco Antonio Macías, Clara Nogueiras, Alicia Gómez, José A. Escario
Published in Revista de biología tropical (01.12.2008)
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Published in Revista de biología tropical (01.12.2008)
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