The anti‐HIV drug nelfinavir mesylate (Viracept) is a potent inhibitor of cell fusion caused by the SARSCoV‐2 spike (S) glycoprotein warranting further evaluation as an antiviral against COVID‐19 infections
Musarrat, Farhana, Chouljenko, Vladimir, Dahal, Achyut, Nabi, Rafiq, Chouljenko, Tamara, Jois, Seetharama D., Kousoulas, Konstantin G.
Published in Journal of medical virology (01.10.2020)
Published in Journal of medical virology (01.10.2020)
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Journal Article
EGFR trafficking: effect of dimerization, dynamics, and mutation
Schultz, Destiny F, Billadeau, Daniel D, Jois, Seetharama D
Published in Frontiers in oncology (11.09.2023)
Published in Frontiers in oncology (11.09.2023)
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Journal Article
Click Conjugation of Boron Dipyrromethene (BODIPY) Fluorophores to EGFR-Targeting Linear and Cyclic Peptides
Williams, Tyrslai M, Kaufman, Nichole E M, Zhou, Zehua, Singh, Sitanshu S, Jois, Seetharama D, Vicente, Maria da Graça H
Published in Molecules (Basel, Switzerland) (23.01.2021)
Published in Molecules (Basel, Switzerland) (23.01.2021)
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Journal Article
(-)-Oleocanthal as a Dual c-MET-COX2 Inhibitor for the Control of Lung Cancer
Siddique, Abu Bakar, Kilgore, Phillip C S R, Tajmim, Afsana, Singh, Sitanshu S, Meyer, Sharon A, Jois, Seetharama D, Cvek, Urska, Trutschl, Marjan, Sayed, Khalid A El
Published in Nutrients (11.06.2020)
Published in Nutrients (11.06.2020)
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Journal Article
Peptides and peptidomimetics as therapeutic agents for Covid-19
Dahal, Achyut, Sonju, Jafrin Jobayer, Kousoulas, Konstantin G, Jois, Seetharama D
Published in Peptide Science (01.01.2022)
Published in Peptide Science (01.01.2022)
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Journal Article
Web Resource
Design of cyclic and d‐amino acids containing peptidomimetics for inhibition of protein‐protein interactions of HER2‐HER3
Pallerla, Sandeep, Naik, Himgauri, Singh, Sitanshu, Gauthier, Ted, Sable, Rushikesh, Jois, Seetharama D.
Published in Journal of peptide science (01.02.2018)
Published in Journal of peptide science (01.02.2018)
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Journal Article
Structure, Self-Assembly, and Dual Role of a β-Defensin-like Peptide from the Chinese Soft-Shelled Turtle Eggshell Matrix
Lakshminarayanan, Rajamani, Vivekanandan, Subramanian, Samy, Ramar Perumal, Banerjee, Yajnavalka, Chi-Jin, Emma Ooi, Teo, Kay Wah, Jois, Seetharama D. S, Kini, R. Manjunatha, Valiyaveettil, Suresh
Published in Journal of the American Chemical Society (09.04.2008)
Published in Journal of the American Chemical Society (09.04.2008)
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Journal Article
Protein Folding Determinants: Structural Features Determining Alternative Disulfide Pairing in α- and χ/λ-Conotoxins
Kang, Tse Siang, Radić, Zoran, Talley, Todd T, Jois, Seetharama D. S, Taylor, Palmer, Kini, R. Manjunatha
Published in Biochemistry (Easton) (20.03.2007)
Published in Biochemistry (Easton) (20.03.2007)
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Journal Article
An N 6 -methyladenosine at the transited codon 273 of p53 pre-mRNA promotes the expression of R273H mutant protein and drug resistance of cancer cells
Uddin, Mohammad B, Roy, Kartik R, Hosain, Salman B, Khiste, Sachin K, Hill, Ronald A, Jois, Seetharama D, Zhao, Yunfeng, Tackett, Alan J, Liu, Yong-Yu
Published in Biochemical pharmacology (01.02.2019)
Published in Biochemical pharmacology (01.02.2019)
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Journal Article
A pH-sensitive liposome formulation of a peptidomimetic-Dox conjugate for targeting HER2 + cancer
Sonju, Jafrin Jobayer, Dahal, Achyut, Singh, Sitanshu S., Gu, Xin, Johnson, William D., Muthumula, Chandra Mohan Reddy, Meyer, Sharon A., Jois, Seetharama D.
Published in International journal of pharmaceutics (25.01.2022)
Published in International journal of pharmaceutics (25.01.2022)
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Journal Article
1,3‐diarylpyrazolones as potential anticancer agents for non‐small cell lung cancer: Synthesis and antiproliferative activity evaluation
Dahal, Achyut, Lo, Mary, Singh, Sitanshu, Vo, Huu, ElHage, Denzel, Jois, Seetharama D., Murru, Siva
Published in Chemical biology & drug design (01.04.2022)
Published in Chemical biology & drug design (01.04.2022)
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Journal Article
Pseurotin A as a novel suppressor of hormone dependent breast cancer progression and recurrence by inhibiting PCSK9 secretion and interaction with LDL receptor
Abdelwahed, Khaldoun S., Siddique, Abu Bakar, Mohyeldin, Mohamed M., Qusa, Mohammed H., Goda, Amira A., Singh, Sitanshu S., Ayoub, Nehad M., King, Judy Ann, Jois, Seetharama D., El Sayed, Khalid A.
Published in Pharmacological research (01.08.2020)
Published in Pharmacological research (01.08.2020)
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Journal Article
Lyophilized liposomal formulation of a peptidomimetic-Dox conjugate for HER2 positive breast and lung cancer
Sonju, Jafrin Jobayer, Shrestha, Prajesh, Dahal, Achyut, Gu, Xin, Johnson, William D., Zhang, Dachuan, Muthumula, Chandra Mohan Reddy, Meyer, Sharon A., Mattheolabakis, George, Jois, Seetharama D.
Published in International journal of pharmaceutics (25.05.2023)
Published in International journal of pharmaceutics (25.05.2023)
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Journal Article
Synthesis of BODIPY-Peptide Conjugates for Fluorescence Labeling of EGFR Overexpressing Cells
Zhao, Ning, Williams, Tyrslai M, Zhou, Zehua, Fronczek, Frank R, Sibrian-Vazquez, Martha, Jois, Seetharama D, Vicente, M. Graça H
Published in Bioconjugate chemistry (17.05.2017)
Published in Bioconjugate chemistry (17.05.2017)
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