Intranasal administration of a stapled relaxin‐3 mimetic has anxiolytic‐ and antidepressant‐like activity in rats
Marwari, Subhi, Poulsen, Anders, Shih, Norrapat, Lakshminarayanan, Rajamani, Kini, R. Manjunatha, Johannes, Charles William, Dymock, Brian William, Dawe, Gavin Stewart
Published in British journal of pharmacology (01.10.2019)
Published in British journal of pharmacology (01.10.2019)
Get full text
Journal Article
Design-Rules for Stapled Alpha-Helical Peptides with On-Target In Vivo Activity: Application to Mdm2/X dual antagonists
Chandramohan, Arun, Josien, Hubert, Yuen, Tsz Ying, Duggal, Ruchia, Spiegelberg, Diana, Yan, Lin, Angela Juang, Yu-Chi, Ge, Lan, Aronica, Pietro, Kaan, Kristal, Lim, Yee Hwee, Peier, Andrea, Sherborne, Brad, Hochman, Jerome, Lin, Songnian, Biswas, Kaustav, Henry, Brian, Nestor, Marika, Verma, Chandra S, Lane, David, Sawyer, Tomi, Garbaccio, Robert, Kannan, Srinivasaraghavan, Brown, Christopher J., Johannes, Charles W, Partridge, Anthony William
Published in Nature communications (26.02.2023)
Published in Nature communications (26.02.2023)
Get full text
Journal Article
Hydrocarbon stapled B chain analogues of relaxin-3 retain biological activity
Jayakody, Tharindunee, Marwari, Subhi, Lakshminarayanan, Rajamani, Tan, Francis Chee Kuan, Johannes, Charles William, Dymock, Brian William, Poulsen, Anders, Herr, Deron Raymond, Dawe, Gavin Stewart
Published in Peptides (New York, N.Y. : 1980) (01.10.2016)
Published in Peptides (New York, N.Y. : 1980) (01.10.2016)
Get full text
Journal Article
Cascade fluorofunctionalisation of 2,3-unsubstituted indoles by means of electrophilic fluorination
Tuan Minh Nguyen, Duong, Hung A., Richard, Jean-Alexandre, Johannes, Charles William, Fu Pincheng, Ye, Danson Kwong Jia, Shuying, Eileen Lau
Published in Chemical communications (Cambridge, England) (21.11.2013)
Published in Chemical communications (Cambridge, England) (21.11.2013)
Get full text
Journal Article
Cascade fluorofunctionalisation of 2,3-unsubstituted indoles by means of electrophilic fluorinationElectronic supplementary information (ESI) available: Full experimental procedures, compound characterisation and copies of NMR spectra. See DOI: 10.1039/c3cc46564k
Nguyen, Tuan Minh, Duong, Hung A, Richard, Jean-Alexandre, Johannes, Charles William, Pincheng, Fu, Kwong Jia Ye, Danson, Shuying, Eileen Lau
Year of Publication 17.10.2013
Year of Publication 17.10.2013
Get full text
Journal Article
C-TERMINAL EXTENDED P53 ACTIVATOR CROSSLINKED PEPTIDOMIMETIC MACROCYCLES AGAINST MDM2/MDMX
YUEN, Tsz Ying, KANNAN, Srinivasaraghavan, BROWN, Christopher, J, CHANDRAMOHAN, Arun, JOHANNES, Charles, William, JOSIEN, Hubert, VERMA, Chandra Shekhar, PARTRIDGE, Anthony, W, YAN, Lin
Year of Publication 09.10.2024
Get full text
Year of Publication 09.10.2024
Patent
P53 PEPTIDOMIMETIC MACROCYCLES
YUEN, Tsz Ying, KANNAN, Srinivasaraghavan, JOHANNES, Charles William, CHANDRAMOHAN, Arun, JOSIEN, Hubert, VERMA, Chandra Shekhar, YAN, Lin, BROWN, Christopher, PARTRIDGE, Anthony William
Year of Publication 03.08.2023
Get full text
Year of Publication 03.08.2023
Patent
P53 PEPTIDOMIMETIC MACROCYCLES
YUEN, Tsz Ying, KANNAN, Srinivasaraghavan, JOHANNES, Charles William, CHANDRAMOHAN, Arun, JOSIEN, Hubert, VERMA, Chandra Shekhar, YAN, Lin, BROWN, Christopher, PARTRIDGE, Anthony William
Year of Publication 15.06.2023
Get full text
Year of Publication 15.06.2023
Patent
STAPLED PEPTIDES
YUEN, Tsz Ying, FERRER GAGO, Fernando Jose, JOHANNES, Charles William
Year of Publication 30.10.2019
Get full text
Year of Publication 30.10.2019
Patent
STAPLED PEPTIDES
YUEN, Tsz Ying, FERRER GAGO, Fernando Jose, JOHANNES, Charles William
Year of Publication 27.09.2018
Get full text
Year of Publication 27.09.2018
Patent
CELL PERMEABLE MACROCYCLIC PEPTIDES USEFUL FOR EIF4E CAP-BINDING SITE INHIBITION
KAAN, Hung Yi, VERMA, Chandra Shekhar, YAN, Lin, FROSI, Yuri, YADAHALLI, Shilpa Siddappa, YUEN, Tsz Ying, KANNAN, Srinivasaraghavan, LANE, David Philip, JOHANNES, Charles William, LUKAMTO, Daniel Hartoyo, ARONICA, Pietro, SAWYER, Tomi, LI, Jianguo, BROWN, Christopher, PARTRIDGE, Anthony William
Year of Publication 27.04.2023
Get full text
Year of Publication 27.04.2023
Patent
ChemInform Abstract: Cascade Fluorofunctionalization of 2,3-Unsubstituted Indoles by Means of Electrophilic Fluorination
Nguyen, Tuan Minh, Duong, Hung A., Richard, Jean-Alexandre, Johannes, Charles William, Pincheng, Fu, Ye, Danson Kwong Jia, Shuying, Eileen Lau
Published in ChemInform (01.04.2014)
Published in ChemInform (01.04.2014)
Get full text
Journal Article
PHOSPHORUS-CONTAINING CATALYSTS
PODICHETTY, ANIL, JONG, HOWARD, YANG, YONG, JOHANNES, CHARLES WILLIAM, LIM, YEE HWEE, CHIA, SAEI WENG, GEORGE ROBINS, EDWARD
Year of Publication 30.03.2016
Get full text
Year of Publication 30.03.2016
Patent