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[18F]BTK-1: A Novel Positron Emission Tomography Tracer for Imaging Bruton’s Tyrosine Kinase
Skaddan, Marc B., Wooten, Dustin W., Wilcox, Kyle C., Voorbach, Martin J., Reuter, David R., Jia, Zhaozhong J., Foster-Duke, Kelly D., Hickson, Jonathan A., Vaidyanathan, Srirajan, Reed, Aimee D., Tovcimak, Ann E., Guo, Qi, Comley, Robert A., Lee, Lance, Finnema, Sjoerd J., Mudd, Sarah R.
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Design, synthesis and structure–Activity relationships of benzoxazinone-Based factor Xa inhibitors
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Published in Bioorganic & medicinal chemistry letters (10.02.2003)
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1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 3: Design, synthesis and sar of orally bioavailable benzamidine-P4 inhibitors
JIA, Zhaozhong J, YANHONG WU, HOLLENNBACH, Stanley J, LAMBING, Joseph L, SCARBOROUGH, Robert M, ZHU, Bing-Yan, WENRONG HUANG, PENGLIE ZHANG, YONGHONG SONG, WOOLFREY, John, SINHA, Uma, ARFSTEN, Ann E, EDWARDS, Susan T, HUTCHALEELAHA, Athiwat
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
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PYRIMIDINES FOR DEGRADING BRUTON'S TYROSINE KINASE
BERENGER BIANNIC, ELIZABETH L NOEY, JOSHUA N PAYETTE, OKANO AKINORI, SHAHAB MORTEZAEI, BIAN ZHIGUO, JASON P BURKE, ASHLEY M ADAMS, VENKAT REDDY MALI, ALEXEY A RIVKIN, ZHAO XIANRUI, MATTHEW H KATCHER, VIOLETA L MARIN, JIANG XINGYU, JIA ZHAOZHONG J, KEVIN R WOLLER, SPENCER O SHOLZ, JEFFERY A ZABLOCKI
Year of Publication 04.10.2023
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Year of Publication 04.10.2023
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브루톤 티로신 키나제의 억제제
CHEN WEI, ATALLAH GORDANA BABIC, JIA ZHAOZHONG J, POZZAN ALFONSO, RAVEGLIA LUCAL FRANCESCO, ZANALETTI RICCARDO
Year of Publication 05.03.2018
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Year of Publication 05.03.2018
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1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides as potent factor xa inhibitors. Part 2: A survey of P4 motifs
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Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors incorporating substituted biphenyl P4 motifs
PENGLIE ZHANG, LIANG BAO, LAMBING, Joseph L, HOLLENBACH, Stanley J, SCARBOROUGH, Robert M, ZHU, Bing-Yan, ZUCKETT, Jingmei F, GOLDMAN, Erick A, JIA, Zhaozhong J, ARFSTEN, Ann, EDWARDS, Susan, SINHA, Uma, HUTCHALEELAHA, Athiwat, PARK, Gary
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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Design, synthesis, and SAR of anthranilamide-based factor Xa inhibitors with improved functional activity
PENGLIE ZHANG, LIANG BAO, HOLLENBACH, Stanley J, SCARBOROUGH, Robert M, ZHU, Bing-Yan, ZUCKETT, Jingmei F, JIA, Zhaozhong J, WOOLFREY, John, ARFSTEN, Ann, EDWARDS, Susan, SINHA, Uma, HUTCHALEELAHA, Athiwat, LAMBING, Joseph L
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Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P1 Structure-activity relationships of the substituted 1-(2-naphthyl)-1H-pyrazole-5-carboxylamides
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Published in Bioorganic & medicinal chemistry letters (01.06.2002)
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N, N-Dialkylated 4-(4-arylsulfonylpiperazine-1-carbonyl)-benzamidines and 4-((4-arylsulfonyl)-2-oxo-piperazin-1-ylmethyl)-benzamidines as potent factor Xa inhibitors
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Inhibition of Purified Factor Xa Amidolytic Activity May Not Be Predictive of Inhibition of In Vivo Thrombosis: Implications for Identification of Therapeutically Active Inhibitors
Sinha, Uma, Lin, Pei Hua, Edwards, Susan T, Wong, Paul W, Zhu, Bingyan, Scarborough, Robert M, Su, Ting, Jia, Zhaozhong J, Song, Yonghong, Zhang, Penglie, Clizbe, Lane, Park, Gary, Reed, Andrea, Hollenbach, Stanley J, Malinowski, John, Arfsten, Ann E
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Published in Arteriosclerosis, thrombosis, and vascular biology (01.06.2003)
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26-DIAMINO-PYRIMIDIN-5-YL-CARBOXAMIDES AS SYK OR JAK KINASES INHIBITORS
ROSE JACK W, PANDEY ANJALI, HUANG WOLIN, MEHROTRA MUKUND, JIA ZHAOZHONG J, SONG YONGHONG, XU QING, KANE BRIAN, BAUER SHAWN M, VENKATARAMANI CHANDRASEKAR
Year of Publication 11.05.2017
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Year of Publication 11.05.2017
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