SB‐334867‐A: the first selective orexin‐1 receptor antagonist
Smart, D, Sabido‐David, C, Brough, S J, Jewitt, F, Johns, A, Porter, R A, Jerman, J C
Published in British journal of pharmacology (01.03.2001)
Published in British journal of pharmacology (01.03.2001)
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Journal Article
Characterization of recombinant human orexin receptor pharmacology in a Chinese hamster ovary cell‐line using FLIPR
Smart, D, Jerman, J C, Brough, S J, Rushton, S L, Murdock, P R, Jewitt, F, Elshourbagy, N A, Ellis, C E, Middlemiss, D N, Brown, F
Published in British journal of pharmacology (01.09.1999)
Published in British journal of pharmacology (01.09.1999)
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Journal Article
Use of cryopreserved cells for enabling greater flexibility in compound profiling
Wigglesworth, M J, Lawless, K J, Standing, D J, Mackenzie, E K, Kitchen, V R, McKay, F, Ward, E, Brough, S J, Stylianou, M, Jewitt, F R, McLaren-Douglas, A M, Jowet, M I, Tamayama, N, Finnigan, D, Ding, J, Wise, A
Published in Journal of biomolecular screening (01.06.2008)
Published in Journal of biomolecular screening (01.06.2008)
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Journal Article
The hypocretins are weak agonists at recombinant human orexin‐1 and orexin‐2 receptors
Smart, D, Jerman, J C, Brough, S J, Neville, W A, Jewitt, F, Porter, R A
Published in British journal of pharmacology (01.04.2000)
Published in British journal of pharmacology (01.04.2000)
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Journal Article
Evidence for antagonist activity of the dopamine D3 receptor partial agonist, BP 897, at human dopamine D3 receptor
Wood, Martyn D, Boyfield, Izzy, Nash, David J, Jewitt, Frances R, Avenell, Kim Y, Riley, Graham J
Published in European journal of pharmacology (27.10.2000)
Published in European journal of pharmacology (27.10.2000)
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Journal Article
Pharmacological Actions of a Novel, High-Affinity, and Selective Human Dopamine D3 Receptor Antagonist, SB-277011-A
Charlie Reavill, Stephen G. Taylor, Martyn D. Wood, Tracey Ashmeade, Nigel E. Austin, Kim Y. Avenell, Izzy Boyfield, Clive L. Branch, Jackie Cilia, Martyn C. Coldwell, Michael S. Hadley, A. Jackie Hunter, Phil Jeffrey, Frances Jewitt, Christopher N. Johnson, Declan N. C. Jones, Andrew D. Medhurst, Derek N. Middlemiss, David J. Nash, Graham J. Riley, Carol Routledge, Geoff Stemp, Kevin M. Thewlis, Brenda Trail, Antonio K. K. Vong, Jim J. Hagan
Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
Journal Article
1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor
PORTER, Roderick A, CHAN, Wai N, JEWITT, A. Frances, JEFFREY, Phillip, AUSTIN, Nigel, COULTON, Steven, JOHNS, Amanda, HADLEY, Michael S, WIDDOWSON, Katherine, JERMAN, Jeffrey C, BROUGH, Stephen J, COLDWELL, Martyn, SMART, Darren
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
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Journal Article
Characterisation of an endogenous bombesin receptor in CHO/DG44 cells
Brough, Stephen J, Jerman, Jeffrey C, Jewitt, Frances, Smart, Darren
Published in European journal of pharmacology (15.12.2000)
Published in European journal of pharmacology (15.12.2000)
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Journal Article
Pharmacological actions of a novel, high-affinity, and selective human dopamine D(3) receptor antagonist, SB-277011-A
Reavill, C, Taylor, S G, Wood, M D, Ashmeade, T, Austin, N E, Avenell, K Y, Boyfield, I, Branch, C L, Cilia, J, Coldwell, M C, Hadley, M S, Hunter, A J, Jeffrey, P, Jewitt, F, Johnson, C N, Jones, D N, Medhurst, A D, Middlemiss, D N, Nash, D J, Riley, G J, Routledge, C, Stemp, G, Thewlis, K M, Trail, B, Vong, A K, Hagan, J J
Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2000)
Journal Article