Cabozantinib (XL184), a novel MET and VEGFR2 inhibitor, simultaneously suppresses metastasis, angiogenesis, and tumor growth
Yakes, F Michael, Chen, Jason, Tan, Jenny, Yamaguchi, Kyoko, Shi, Yongchang, Yu, Peiwen, Qian, Fawn, Chu, Felix, Bentzien, Frauke, Cancilla, Belinda, Orf, Jessica, You, Andrew, Laird, A Douglas, Engst, Stefan, Lee, Lillian, Lesch, Justin, Chou, Yu-Chien, Joly, Alison H
Published in Molecular cancer therapeutics (01.12.2011)
Published in Molecular cancer therapeutics (01.12.2011)
Get full text
Journal Article
Abstract 4999: Cellular mechanism of action of bispecific T-cell engager (BiTE®) antibody constructs targeting Folate Receptor 1
Bailis, Julie M., Orf, Jessica N., Sternjak, Alexander, Belmontes, Brian, Case, Ryan, Grinberg, Natalia, Chang, Wesley, Hinkle, Beth, Friedrich, Matthias
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Get full text
Journal Article
Metastatic Properties and Genomic Amplification of the Tyrosine Kinase Gene ACK1
Edward Htun van der Horst, Yan Y. Degenhardt, Strelow, Astrid, Slavin, Anthony, Lawrence Chinn, Jessica Orf, Rong, Minqing, Li, Shyun, Lei-Hoon See, Ken Q. C. Nguyen, Hoey, Timothy, Wesche, Holger, Powers, Scott, McKnight, Steven L.
Published in Proceedings of the National Academy of Sciences - PNAS (01.11.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (01.11.2005)
Get full text
Journal Article
Single-Cell Analyses Inform Mechanisms of Myeloid-Targeted Therapies in Colon Cancer
Zhang, Lei, Li, Ziyi, Skrzypczynska, Katarzyna M., Fang, Qiao, Zhang, Wei, O’Brien, Sarah A., He, Yao, Wang, Lynn, Zhang, Qiming, Kim, Aeryon, Gao, Ranran, Orf, Jessica, Wang, Tao, Sawant, Deepali, Kang, Jiajinlong, Bhatt, Dev, Lu, Daniel, Li, Chi-Ming, Rapaport, Aaron S., Perez, Kristy, Ye, Yingjiang, Wang, Shan, Hu, Xueda, Ren, Xianwen, Ouyang, Wenjun, Shen, Zhanlong, Egen, Jackson G., Zhang, Zemin, Yu, Xin
Published in Cell (16.04.2020)
Published in Cell (16.04.2020)
Get full text
Journal Article
Comparison of cesium and X-ray irradiation for generation of bone marrow chimeras
Eng, Jason Samuel, Orf, Jessica, Perez, Kristy, Sawant, Deepali, DeVoss, Jason J
Published in The Journal of immunology (1950) (01.05.2020)
Published in The Journal of immunology (1950) (01.05.2020)
Get full text
Journal Article
Activity of tumor-associated macrophage depletion by CSF1R blockade is highly dependent on the tumor model and timing of treatment
O’Brien, Sarah A., Orf, Jessica, Skrzypczynska, Katarzyna M., Tan, Hong, Kim, Jennie, DeVoss, Jason, Belmontes, Brian, Egen, Jackson G.
Published in Cancer Immunology, Immunotherapy (01.08.2021)
Published in Cancer Immunology, Immunotherapy (01.08.2021)
Get full text
Journal Article
Abstract 1586: Oncolytic virus HSV-1/ICP34.5-/ICP47-/mFLT3L/mIL12 promotes systemic anti-tumor responses and cooperates with immuno-modulatory agents in multiple mouse syngeneic tumor models
Cooke, Keegan, Meisen, Walter H., Mitchell, Petia, Estrada, Juan, Zhan, Jinghui, Orf, Jessica, Li, Peng, de Zafra, Christina, Qing, Jing, DeVoss, Jason
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Get full text
Journal Article
Abstract 2803: CSF-1 receptor-mediated macrophage depletion can induce immunomodulatory resistance mechanisms in murine tumor models
O'Brien, Sarah A., Skrzypczynska, Katarzyna, Orf, Jessica, Belmontes, Brian, Tan, Hong, Lu, Daniel, Driver, Ian, Egen, Jackson
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Get full text
Journal Article
Brief report: STING expressed in tumor and non-tumor compartments has distinct roles in regulating anti-tumor immunity
Kim, Jennie C., Liu, Xian, Fitzgerald, Karen, Eng, Jason S., Orf, Jessica, O’Brien, Sarah A., Belmontes, Brian, Casbon, Amy-Jo, Novitskiy, Sergey V., Tarbell, Kristin V., DeVoss, Jason, Egen, Jackson G.
Published in Cancer Immunology, Immunotherapy (01.05.2023)
Published in Cancer Immunology, Immunotherapy (01.05.2023)
Get full text
Journal Article
Abstract P4-07-12: Development of Triple-negative breast cancer (TNBC) syngeneic models and TROP2-directed antibody-drug conjugate (ADC) surrogate to model therapeutic combinations
Chou, Chih-Chien, Kardos, Jordan, Yang, Becky, Orf, Jessica, Dave, Rutwij, Lai, Yurong, Lee, Chingwei V., Papalia, Giuseppe A., Boyd, Kelli, Diehl, Lauri, Scholler, Nathalie
Published in Cancer research (Chicago, Ill.) (01.03.2023)
Published in Cancer research (Chicago, Ill.) (01.03.2023)
Get full text
Journal Article
Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor for treating acute myeloid leukemia
Keegan, Kathleen, Li, Cong, Li, Zhihong, Ma, Ji, Ragains, Mark, Coberly, Suzanne, Hollenback, David, Eksterowicz, John, Liang, Lingming, Weidner, Margaret, Huard, Justin, Wang, Xianghong, Alba, Grace, Orf, Jessica, Lo, Mei-Chu, Zhao, Sharon, Ngo, Rachel, Chen, Ada, Liu, Lily, Carlson, Timothy, Quéva, Christophe, McGee, Lawrence R, Medina, Julio, Kamb, Alexander, Wickramasinghe, Dineli, Dai, Kang
Published in Molecular cancer therapeutics (01.04.2014)
Published in Molecular cancer therapeutics (01.04.2014)
Get full text
Journal Article
Abstract LB-249: Characterization of a novel potent and selective CDK4/6 inhibitor and a resistance mechanism
Dai, Kang, Li, Cong, Liang, Lingming, Rong, Minqing, Orf, Jessica, Keegan, Kathy, Li, Zhihong, Fu, Jiasheng, Ma, Ji, Carlson, Tim, McGee, Larry, Medina, Julio, Kamb, Alexander, Wickramasinghe, Dineli
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Get full text
Journal Article
Abstract 711: Small molecule compounds that target cell division cycle 7 (Cdc7) kinase inhibit cell proliferation and tumor growth
Bailis, Julie, Fang, Li, Orf, Jessica, Heller, Scott, Bush, Tammy, Bourbeau, Matthew, Escobar, Sonia, Frohn, Michael, Harrington, Paul, Hsieh, Faye, Pickrell, Alexander, Sham, Kelvin, Siegmund, Aaron, Tan, Helming, Zalameda, Leeanne, Allen, John, Wickramasinghe, Dineli
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article
Discovery of amide replacements that improve activity and metabolic stability of a bis-amide smoothened antagonist hit
Brown, Matthew L., Aaron, Wade, Austin, Richard J., Chong, Angela, Huang, Tom, Jiang, Ben, Kaizerman, Jacob A., Lee, Gary, Lucas, Brian S., McMinn, Dustin L., Orf, Jessica, Rong, Minqing, Toteva, Maria M., Xu, Guifen, Ye, Qiuping, Zhong, Wendy, DeGraffenreid, Michael R., Wickramasinghe, Dineli, Powers, Jay P., Hungate, Randall, Johnson, Michael G.
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Get full text
Journal Article
Abstract A244: Characterization of a novel potent and selective CDK4/6 inhibitor and a resistance mechanism
Dai, Kang, Li, Cong, Liang, Lingming, Rong, Minqing, Orf, Jessica, Keegan, Kathy, Li, Zhihong, Fu, Jiasheng, Ma, Ji, Carlson, Timothy, McGee, Larry, Medina, Julio, Kamb, Alexander, Wickramasinghe, Dineli
Published in Molecular cancer therapeutics (12.11.2011)
Published in Molecular cancer therapeutics (12.11.2011)
Get full text
Journal Article
Abstract A279: Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor
Dai, Kang, Keegan, Kathleen, Li, Zhihong, Ji, Ma, Li, Cong, Eksterowicz, John, Suzanne, Coberly, Hollenback, David, Weidner, Margret, Huard, Justin, Liang, Lingming, Alba, Grace, Orf, Jessica, Lo, Mei-Chu, Zhao, Sharon, Ngo, Rachel, Chen, Ada, Liu, Lily, Carlson, Timothy, McGee, Lawrence R., Medina, Julio, Kamb, Alexander, Wickramasinghe, Dineli
Published in Molecular cancer therapeutics (01.11.2013)
Published in Molecular cancer therapeutics (01.11.2013)
Get full text
Journal Article
Design of 1-piperazinyl-4-arylphthalazines as potent Smoothened antagonists
Lucas, Brian S., Aaron, Wade, An, Songzhu, Austin, Richard J., Brown, Matthew, Chan, Hon, Chong, Angela, Hungate, Randall, Huang, Tom, Jiang, Ben, Johnson, Michael G., Kaizerman, Jacob A., Lee, Gary, McMinn, Dustin L., Orf, Jessica, Powers, Jay P., Rong, Minqing, Toteva, Maria M., Uyeda, Craig, Wickramasinghe, Dineli, Xu, Guifen, Ye, Qiuping, Zhong, Wendy
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Get full text
Journal Article
Methylthioadenosine (MTA) Rescues Methylthioadenosine Phosphorylase (MTAP)-Deficient Tumors from Purine Synthesis Inhibition in Vivo via Non-Autonomous Adenine Supply
Ruefli-Brasse, Astrid, Sakamoto, Doreen, Orf, Jessica, Rong, Minqing, Shi, Jianxia, Carlson, Tim, Quon, Kim, Kamb, Alexander, Wickramasinghe, Dineli
Published in Journal of cancer therapy (2011)
Published in Journal of cancer therapy (2011)
Get full text
Journal Article