Quantification of Active Site Density and Turnover Frequency: From Single-Atom Metal to Nanoparticle Electrocatalysts
Bae, Geunsu, Kim, Haesol, Choi, Hansol, Jeong, Pyeonghwa, Kim, Dong Hyun, Kwon, Han Chang, Lee, Kug-Seung, Choi, Minkee, Oh, Hyung-Suk, Jaouen, Frédéric, Choi, Chang Hyuck
Published in JACS Au (24.05.2021)
Published in JACS Au (24.05.2021)
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Journal Article
Characterization of LDD-2633 as a Novel RET Kinase Inhibitor with Anti-Tumor Effects in Thyroid Cancer
Lee, Hyo Jeong, Jeong, Pyeonghwa, Moon, Yeongyu, Choi, Jungil, Heo, Jeong Doo, Kim, Yong-Chul, Han, Sun-Young
Published in Pharmaceuticals (Basel, Switzerland) (06.01.2021)
Published in Pharmaceuticals (Basel, Switzerland) (06.01.2021)
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Journal Article
Chemical characterization and biological activity data for a novel indirubin derivative, LDD-1819
Kim, Woong-Hee, Jeong, Pyeonghwa, Kim, Seon-Wook, Cho, Haaglim, Lee, Jeong-min, Seo, Shinae, Shen, Haihong, Ahn, Youngkeun, Jung, Da-Woon, Kim, Yong-Chul, Williams, Darren R.
Published in Data in brief (01.08.2019)
Published in Data in brief (01.08.2019)
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Journal Article
Methotrexate recognition by the human reduced folate carrier SLC19A1
Wright, Nicholas J., Fedor, Justin G., Zhang, Han, Jeong, Pyeonghwa, Suo, Yang, Yoo, Jiho, Hong, Jiyong, Im, Wonpil, Lee, Seok-Yong
Published in Nature (London) (29.09.2022)
Published in Nature (London) (29.09.2022)
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Journal Article
Methotrexate recognition by the human reduced folate carrier SLC19A1
Fedor, Justin G., Wright, Nicholas J., Zhang, Han, Jeong, Pyeonghwa, Suo, Yang, Yoo, Jiho, Hong, Jiyong, Im, Wonpil, Lee, Seok-Yong
Published in Biophysical journal (10.02.2023)
Published in Biophysical journal (10.02.2023)
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Journal Article
Cryo-EM structure determination of the human reduced folate carrier SLC19A1 in complex with methotrexate
Wright, Nicholas J., Fedor, Justin G., Zhang, Han, Jeong, Pyeonghwa, Suo, Yang, Yoo, Jiho, Hong, Jiyong, Im, Wonpil, Lee, Seok-Yong
Published in Biophysical journal (10.02.2023)
Published in Biophysical journal (10.02.2023)
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Journal Article
Discovery of benzimidazole-indazole derivatives as potent FLT3-tyrosine kinase domain mutant kinase inhibitors for acute myeloid leukemia
Ko, Bongki, Jang, Yongsoo, Kim, Min Ha, Lam, Thai Thi, Seo, Hye Kyung, Jeong, Pyeonghwa, Choi, Munkyung, Kang, Keon Wook, Lee, So-Deok, Park, Jin-Hee, Kim, Myungjin, Han, Sun-Young, Kim, Yong-Chul
Published in European journal of medicinal chemistry (15.12.2023)
Published in European journal of medicinal chemistry (15.12.2023)
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Journal Article
Discovery of orally active indirubin-3′-oxime derivatives as potent type 1 FLT3 inhibitors for acute myeloid leukemia
Jeong, Pyeonghwa, Moon, Yeongyu, Lee, Je-Heon, Lee, So-Deok, Park, Jiyeon, Lee, Jungeun, Kim, Jiheon, Lee, Hyo Jeong, Kim, Na Yoon, Choi, Jungil, Heo, Jeong Doo, Shin, Ji Eun, Park, Hyun Woo, Kim, Yoon-Gyoon, Han, Sun-Young, Kim, Yong-Chul
Published in European journal of medicinal chemistry (01.06.2020)
Published in European journal of medicinal chemistry (01.06.2020)
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Journal Article
Discovery of indirubin-3′-aminooxy-acetamide derivatives as potent and selective FLT3/D835Y mutant kinase inhibitors for acute myeloid leukemia
Lee, Je-Heon, Shin, Ji Eun, Kim, WooChan, Jeong, Pyeonghwa, Kim, Myung Jin, Oh, Su Jin, Lee, Hyo Jeong, Park, Hyun Woo, Han, Sun-Young, Kim, Yong-Chul
Published in European journal of medicinal chemistry (05.07.2022)
Published in European journal of medicinal chemistry (05.07.2022)
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Journal Article
Synthesis and evaluation of cyclopentane-based muraymycin analogs targeting MraY
Kwak, Seung-Hwa, Lim, Won Young, Hao, Aili, Mashalidis, Ellene H., Kwon, Do-Yeon, Jeong, Pyeonghwa, Kim, Mi Jung, Lee, Seok-Yong, Hong, Jiyong
Published in European journal of medicinal chemistry (05.04.2021)
Published in European journal of medicinal chemistry (05.04.2021)
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Journal Article
Novel Thioxothiazolo[3,4‑a]quinazolin-5(4H)‑one Derivatives as BKCa Channel Activators for Urinary Incontinence
Bae, Eun Jung, Jo, Heeji, Kim, Seong Soon, Shin, Dae-Seop, Yang, Jung Yoon, Bae, Myung Ae, Jeong, Pyeonghwa, Park, Chul-Seung, Ahn, Jin Hee
Published in ACS medicinal chemistry letters (14.07.2022)
Published in ACS medicinal chemistry letters (14.07.2022)
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Journal Article
Novel Thioxothiazolo[3,4- a ]quinazolin-5(4 H )-one Derivatives as BK Ca Channel Activators for Urinary Incontinence
Bae, Eun Jung, Jo, Heeji, Kim, Seong Soon, Shin, Dae-Seop, Yang, Jung Yoon, Bae, Myung Ae, Jeong, Pyeonghwa, Park, Chul-Seung, Ahn, Jin Hee
Published in ACS medicinal chemistry letters (14.07.2022)
Published in ACS medicinal chemistry letters (14.07.2022)
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Journal Article
Activation mechanism and novel binding sites of the BK Ca channel activator CTIBD
Lee, Narasaem, Kim, Subin, Lee, Na Young, Jo, Heeji, Jeong, Pyeonghwa, Pagire, Haushabhau S, Pagire, Suvarna H, Ahn, Jin Hee, Jin, Mi Sun, Park, Chul-Seung
Published in Life science alliance (01.10.2024)
Published in Life science alliance (01.10.2024)
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Journal Article
A novel indirubin derivative that increases somatic cell plasticity and inhibits tumorigenicity
Kim, Woong-Hee, Jeong, Pyeonghwa, Kim, Seon-Wook, Cho, Haaglim, Lee, Jeong-min, Seo, Shinae, Shen, Haihong, Ahn, Youngkeun, Jung, Da-Woon, Kim, Yong-Chul, Williams, Darren R.
Published in Bioorganic & medicinal chemistry (01.07.2019)
Published in Bioorganic & medicinal chemistry (01.07.2019)
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Journal Article
Activation mechanism and novel binding sites of the BKCa channel activator CTIBD
Lee, Narasaem, Kim, Subin, Lee, Na Young, Jo, Heeji, Jeong, Pyeonghwa, Pagire, Haushabhau S, Pagire, Suvarna H, Ahn, Jin Hee, Jin, Mi Sun, Park, Chul-Seung
Published in Life science alliance (01.10.2024)
Published in Life science alliance (01.10.2024)
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Journal Article
Benserazide, the first allosteric inhibitor of Coxsackievirus B3 3C protease
Kim, Bo-Kyoung, Cho, Joong-Heui, Jeong, Pyeonghwa, Lee, Youngjin, Lim, Jia Jia, Park, Kyoung Ryoung, Eom, Soo Hyun, Kim, Yong-Chul
Published in FEBS letters (08.07.2015)
Published in FEBS letters (08.07.2015)
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Journal Article
Discovery of a FLT3 inhibitor LDD1937 as an anti-leukemic agent for acute myeloid leukemia
Lee, Hyo Jeong, Lee, Jungeun, Jeong, Pyeonghwa, Choi, Jungil, Baek, Juhwa, Ahn, Su Jin, Moon, Yeongyu, Heo, Jeong Doo, Choi, Young Hee, Chin, Young-Won, Kim, Yong-Chul, Han, Sun-Young
Published in Oncotarget (02.01.2018)
Published in Oncotarget (02.01.2018)
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Journal Article
Discovery of Novel Biased Opioid Receptor Ligands through Structure‐Based Pharmacophore Virtual Screening and Experiment
Jeong, Pyeonghwa, Kim, Soo‐Kyung, Li, Quanjie, Oh, Su‐jin, Son, Seonil, Chen, Guangju, Tan, Hongwei, Kim, Siwon, Park, Jong‐Hyun, Park, Ki Duk, Kim, Yeo Ok, Yoon, Myung Ha, Kim, Yong‐Chul, Goddard, William A.
Published in ChemMedChem (17.10.2019)
Published in ChemMedChem (17.10.2019)
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Journal Article
Correction: Discovery of a FLT3 inhibitor LDD1937 as an anti-leukemic agent for acute myeloid leukemia
Lee, Hyo Jeong, Lee, Jungeun, Jeong, Pyeonghwa, Choi, Jungil, Baek, Juhwa, Ahn, Su Lin, Moon, Yeongyu, Heo, Jeong Doo, Choi, Young Hee, Chin, Young-Won, Kim, Yong-Chul, Han, Sun-Young
Published in Oncotarget (13.04.2018)
Published in Oncotarget (13.04.2018)
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Journal Article
A one-step protocol to generate impermeable fluorescent HaloTag substrates for in situ live cell application and super-resolution imaging
Roßmann, Kilian, Sun, Siqi, Olesen, Christina Holmboe, Kowald, Maria, Tapp, Eleni, Pabst, Ulrich, Bieck, Marie, Birke, Ramona, Shields, Brenda C, Jeong, PyeongHwa, Hong, Jiyong, Tadross, Michael R, Levitz, Joshua, Lehmann, Martin, Lipstein, Noa, Broichhagen, Johannes
Published in bioRxiv (23.09.2024)
Published in bioRxiv (23.09.2024)
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