Expeditious synthesis of novel NK1 antagonists based on a 1,2,4-trisubstituted cyclohexane
Dirat, O, Elliott, JM, Jelley, RA, Jones, AB, Reader, M
Published in Tetrahedron letters (20.02.2006)
Published in Tetrahedron letters (20.02.2006)
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Selective, orally active gamma-aminobutyric acid(A) alpha 5 receptor inverse agonists as cognition enhancers
Sternfeld, F, Carling, RW, Jelley, RA, Ladduwahetty, T, Merchant, KJ, Moore, KW, Reeve, AJ, Street, LJ, O'Connor, D, Sohal, B, Atack, Cook, S, Seabrook, G, Wafford, K, Tattersall, FD, Collinson, N, Dawson, GR, Castro, JL, MacLeod, AM
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Synthesis and biological evaluation of 3-heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4-a]phthalazines and analogues as subtype-selective inverse agonists for the GABA(A)alpha 5 benzodiazepine binding site
Street, LJ, Sternfeld, F, Jelley, RA, Reeve, AJ, Carling, RW, Moore, KW, McKernan, RM, Sohal, B, Cook, S, Pike, A, Dawson, GR, Bromidge, FA, Wafford, KA, Seabrook, GR, Thompson, SA, Marshall, G, Pillai, GV, Castro, JL, Atack, MacLeod, AM
Published in Journal of medicinal chemistry (01.07.2004)
Published in Journal of medicinal chemistry (01.07.2004)
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Journal Article
Synthesis and Conformational Dynamics of Tricyclic Pyridones Containing a Fused Seven-Membered Ring
Gibson, Karl R, Hitzel, Laure, Mortishire-Smith, Russell J, Gerhard, Ute, Jelley, Richard A, Reeve, Austin J, Rowley, Michael, Nadin, Alan, Owens, Andrew P
Published in Journal of organic chemistry (27.12.2002)
Published in Journal of organic chemistry (27.12.2002)
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Synthesis and Serotonergic Activity of 3-[2-(Pyrrolidin-1-yl)ethyl]indoles: Potent Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Receptor
Sternfeld, Francine, Guiblin, Alexander R, Jelley, Richard A, Matassa, Victor G, Reeve, Austin J, Hunt, Peter A, Beer, Margaret S, Heald, Anne, Stanton, Josephine A, Sohal, Bindi, Watt, Alan P, Street, Leslie J
Published in Journal of medicinal chemistry (25.02.1999)
Published in Journal of medicinal chemistry (25.02.1999)
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Journal Article
Synthesis and Serotonergic Activity of N,N-Dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine and Analogs: Potent Agonists for 5-HT1D Receptors
Street, Leslie J, Baker, Raymond, Davey, William B, Guiblin, Alexander R, Jelley, Richard A, Reeve, Austin J, Routledge, Helen, Sternfeld, Francine, Watt, Alan P
Published in Journal of medicinal chemistry (01.05.1995)
Published in Journal of medicinal chemistry (01.05.1995)
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Journal Article
3-(Piperazinylpropyl)indoles: Selective, Orally Bioavailable h5-HT1D Receptor Agonists as Potential Antimigraine Agents
Chambers, Mark S, Street, Leslie J, Goodacre, Simon, Hobbs, Sarah C, Hunt, Peter, Jelley, Richard A, Matassa, Victor G, Reeve, Austin J, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Rathbone, Denise, Watt, Alan P, MacLeod, Angus M
Published in Journal of medicinal chemistry (25.02.1999)
Published in Journal of medicinal chemistry (25.02.1999)
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Journal Article
Selective, Orally Active 5-HT1D Receptor Agonists as Potential Antimigraine Agents
MacLeod, Angus M, Street, Leslie J, Reeve, Austin J, Jelley, Richard A, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Watt, Alan P, Rathbone, Denise, Matassa, Victor G
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Journal Article
3-[2-(Pyrrolidin-1-yl)ethyl]indoles and 3-[3-(Piperidin-1-yl)propyl]indoles: Agonists for the h5-HT1D Receptor with High Selectivity over the h5-HT1B Subtype
Castro, José L, Street, Leslie J, Guiblin, Alexander R, Jelley, Richard A, Russell, Michael G. N, Sternfeld, Francine, Beer, Margaret S, Stanton, Josephine A, Matassa, Victor G
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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The chemical evolution of N,N-dimethyl-2-[5-(1,2,4-triazol-4-yl)-1H-indol-3-yl]ethylamine (L-741,604) and analogues: Potent and selective agonists for 5-HT1D receptors
Sternfeld, Francine, Baker, Raymond, Broughton, Howard B., Guiblin, Alexander R., Jelley, Richard A., Matassa, Victor G., Reeve, Austin J., Beer, Margaret S., Stanton, Josephine A., Hargreaves, Richard J., Shepheard, Sara L., Longmore, Jeanette, Razzaque, Zerin, Graham, Michael I., Sohal, Bindi, Street, Leslie J.
Published in Bioorganic & medicinal chemistry letters (06.08.1996)
Published in Bioorganic & medicinal chemistry letters (06.08.1996)
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