Structure and dynamics of the active human parathyroid hormone receptor-1
Zhao, Li-Hua, Ma, Shanshan, Sutkeviciute, Ieva, Shen, Dan-Dan, Zhou, X Edward, de Waal, Parker W, Li, Chen-Yao, Kang, Yanyong, Clark, Lisa J, Jean-Alphonse, Frederic G, White, Alex D, Yang, Dehua, Dai, Antao, Cai, Xiaoqing, Chen, Jian, Li, Cong, Jiang, Yi, Watanabe, Tomoyuki, Gardella, Thomas J, Melcher, Karsten, Wang, Ming-Wei, Vilardaga, Jean-Pierre, Xu, H Eric, Zhang, Yan
Published in Science (American Association for the Advancement of Science) (12.04.2019)
Published in Science (American Association for the Advancement of Science) (12.04.2019)
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Sustained cyclic AMP production by parathyroid hormone receptor endocytosis
Ferrandon, Sébastien, Feinstein, Timothy N, Castro, Marian, Wang, Bin, Bouley, Richard, Potts, John T, Gardella, Thomas J, Vilardaga, Jean-Pierre
Published in Nature chemical biology (01.10.2009)
Published in Nature chemical biology (01.10.2009)
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Journal Article
Noncanonical Control of Vasopressin Receptor Type 2 Signaling by Retromer and Arrestin
Feinstein, Timothy N., Yui, Naofumi, Webber, Matthew J., Wehbi, Vanessa L., Stevenson, Hilary P., King, J. Darwin, Hallows, Kenneth R., Brown, Dennis, Bouley, Richard, Vilardaga, Jean-Pierre
Published in The Journal of biological chemistry (27.09.2013)
Published in The Journal of biological chemistry (27.09.2013)
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Journal Article
Noncanonical GPCR signaling arising from a PTH receptor–arrestin–Gβγ complex
Wehbi, Vanessa L., Stevenson, Hilary P., Feinstein, Timothy N., Calero, Guillermo, Romero, Guillermo, Vilardaga, Jean-Pierre
Published in Proceedings of the National Academy of Sciences - PNAS (22.01.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (22.01.2013)
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Journal Article
Gq/11-dependent regulation of endosomal cAMP generation by parathyroid hormone class B GPCR
White, Alex D., Jean-Alphonse, Frederic G., Fang, Fei, Peña, Karina A., Liu, Shi, König, Gabriele M., Inoue, Asuka, Aslanoglou, Despoina, Gellman, Samuel H., Kostenis, Evi, Xiao, Kunhong, Vilardaga, Jean-Pierre
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2020)
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.2020)
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Journal Article
Allosteric interactions in the parathyroid hormone GPCR-arrestin complex formation
Clark, Lisa J, Krieger, James, White, Alex D, Bondarenko, Vasyl, Lei, Saifei, Fang, Fei, Lee, Ji Young, Doruker, Pemra, Böttke, Thore, Jean-Alphonse, Frederic, Tang, Pei, Gardella, Thomas J, Xiao, Kunhong, Sutkeviciute, Ieva, Coin, Irene, Bahar, Ivet, Vilardaga, Jean-Pierre
Published in Nature chemical biology (01.10.2020)
Published in Nature chemical biology (01.10.2020)
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Journal Article
Design and validation of the first cell‐impermeant melatonin receptor agonist
Gbahou, Florence, Cecon, Erika, Viault, Guillaume, Gerbier, Romain, Jean‐Alphonse, Frederic, Karamitri, Angeliki, Guillaumet, Gérald, Delagrange, Philippe, Friedlander, Robert M, Vilardaga, Jean‐Pierre, Suzenet, Franck, Jockers, Ralf
Published in British journal of pharmacology (01.07.2017)
Published in British journal of pharmacology (01.07.2017)
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Journal Article
Precise druggability of the PTH type 1 receptor
Sutkeviciute, Ieva, Lee, Ji Young, White, Alex D, Maria, Christian Santa, Peña, Karina A, Savransky, Sofya, Doruker, Pemra, Li, Hongchun, Lei, Saifei, Kaynak, Burak, Tu, Chialing, Clark, Lisa J, Sanker, Subramaniam, Gardella, Thomas J, Chang, Wenhan, Bahar, Ivet, Vilardaga, Jean-Pierre
Published in Nature chemical biology (01.03.2022)
Published in Nature chemical biology (01.03.2022)
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Journal Article
Lighting up multiprotein complexes: lessons from GPCR oligomerization
Ciruela, Francisco, Vilardaga, Jean-Pierre, Fernández-Dueñas, Víctor
Published in Trends in biotechnology (Regular ed.) (01.08.2010)
Published in Trends in biotechnology (Regular ed.) (01.08.2010)
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Journal Article
Altered Selectivity of Parathyroid Hormone (PTH) and PTH-Related Protein (PTHrP) for Distinct Conformations of the PTH/PTHrP Receptor
Dean, Thomas, Vilardaga, Jean-Pierre, Potts, John T, Gardella, Thomas J
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2008)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2008)
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Journal Article
Actin-Sorting Nexin 27 (SNX27)-Retromer Complex Mediates Rapid Parathyroid Hormone Receptor Recycling
McGarvey, Jennifer C., Xiao, Kunhong, Bowman, Shanna L., Mamonova, Tatyana, Zhang, Qiangmin, Bisello, Alessandro, Sneddon, W. Bruce, Ardura, Juan A., Jean-Alphonse, Frederic, Vilardaga, Jean-Pierre, Puthenveedu, Manojkumar A., Friedman, Peter A.
Published in The Journal of biological chemistry (20.05.2016)
Published in The Journal of biological chemistry (20.05.2016)
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Journal Article
Endosomal GPCR signaling turned off by negative feedback actions of PKA and v-ATPase
Gidon, Alexandre, Al-Bataineh, Mohammad M, Jean-Alphonse, Frederic G, Stevenson, Hilary P, Watanabe, Tomoyuki, Louet, Claire, Khatri, Ashok, Calero, Guillermo, Pastor-Soler, Núria M, Gardella, Thomas J, Vilardaga, Jean-Pierre
Published in Nature chemical biology (01.09.2014)
Published in Nature chemical biology (01.09.2014)
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Journal Article
A FlAsH-based FRET approach to determine G protein-coupled receptor activation in living cells
Lohse, Martin J, Hoffmann, Carsten, Gaietta, Guido, Bünemann, Moritz, Adams, Stephen R, Oberdorff-Maass, Silke, Behr, Björn, Vilardaga, Jean-Pierre, Tsien, Roger Y, Ellisman, Mark H
Published in Nature methods (01.03.2005)
Published in Nature methods (01.03.2005)
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Journal Article
Optical techniques to analyze real-time activation and signaling of G-protein-coupled receptors
Lohse, Martin J, Nikolaev, Viacheslav O, Hein, Peter, Hoffmann, Carsten, Vilardaga, Jean-Pierre, Bünemann, Moritz
Published in Trends in pharmacological sciences (Regular ed.) (01.03.2008)
Published in Trends in pharmacological sciences (Regular ed.) (01.03.2008)
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Journal Article
Real-time optical recording of β1-adrenergic receptor activation reveals supersensitivity of the Arg389 variant to carvedilol
Rochais, Francesca, Vilardaga, Jean-Pierre, Nikolaev, Viacheslav O., Bünemann, Moritz, Lohse, Martin J., Engelhardt, Stefan
Published in The Journal of clinical investigation (02.01.2007)
Published in The Journal of clinical investigation (02.01.2007)
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Journal Article
Structural insights into emergent signaling modes of G protein–coupled receptors
Sutkeviciute, Ieva, Vilardaga, Jean-Pierre
Published in The Journal of biological chemistry (14.08.2020)
Published in The Journal of biological chemistry (14.08.2020)
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