Analysis of Quinolinequinone Analogs with Promising Cytotoxic Activity against Breast Cancer
Yilmaz Goler, Ayse Mine, Tarbin Jannuzzi, Ayse, Biswas, Abanish, Mondal, Subodh, Basavanakatti, Vinay N., Jayaprakash Venkatesan, Raghusrinivasan, Yıldırım, Hatice, Yıldız, Mahmut, Çelik Onar, Hülya, Bayrak, Nilüfer, Jayaprakash, Venkatesan, TuYuN, Amaç Fatih
Published in Chemistry & biodiversity (01.09.2023)
Published in Chemistry & biodiversity (01.09.2023)
Get full text
Journal Article
Farnesyl Transferase Inhibitors as Potential Anticancer Agents
Bagchi, Sounak, Rathee, Parth, Jayaprakash, Venkatesan, Banerjee, Sugato
Published in Mini reviews in medicinal chemistry (01.01.2018)
Published in Mini reviews in medicinal chemistry (01.01.2018)
Get more information
Journal Article
Exploring the Anticancer Effects of Brominated Plastoquinone Analogs with Promising Cytotoxic Activity in MCF-7 Breast Cancer Cells via Cell Cycle Arrest and Oxidative Stress Induction
Jannuzzi, Ayse Tarbin, Yilmaz Goler, Ayse Mine, Bayrak, Nilüfer, Yıldız, Mahmut, Yıldırım, Hatice, Karademir Yilmaz, Betul, Shilkar, Deepak, Venkatesan, Raghusrinivasan Jayaprakash, Jayaprakash, Venkatesan, TuYuN, Amaç Fatih
Published in Pharmaceuticals (Basel, Switzerland) (22.06.2022)
Published in Pharmaceuticals (Basel, Switzerland) (22.06.2022)
Get full text
Journal Article
In Silico Drug Repurposing Studies for the Discovery of Novel Salicyl-AMP Ligase (MbtA)Inhibitors
Rakshit, Gourav, Biswas, Abanish, Jayaprakash, Venkatesan
Published in Pathogens (Basel) (01.12.2023)
Published in Pathogens (Basel) (01.12.2023)
Get full text
Journal Article
Highly Active Small Aminated Quinolinequinones against Drug-Resistant Staphylococcus aureus and Candida albicans
Yıldırım, Hatice, Bayrak, Nilüfer, Yıldız, Mahmut, Yılmaz, Fatıma Nur, Mataracı-Kara, Emel, Shilkar, Deepak, Jayaprakash, Venkatesan, TuYuN, Amaç Fatih
Published in Molecules (Basel, Switzerland) (03.05.2022)
Published in Molecules (Basel, Switzerland) (03.05.2022)
Get full text
Journal Article
SELEX based aptamers with diagnostic and entry inhibitor therapeutic potential for SARS-CoV-2
Halder, Sayanti, Thakur, Abhishek, Keshry, Supriya Suman, Jana, Pradip, Karothia, Divyanshi, Das Jana, Indrani, Acevedo, Orlando, Swain, Rajeeb K., Mondal, Arindam, Chattopadhyay, Soma, Jayaprakash, Venkatesan, Dev, Abhimanyu
Published in Scientific reports (04.09.2023)
Published in Scientific reports (04.09.2023)
Get full text
Journal Article
A novel druggable interprotomer pocket in the capsid of rhino- and enteroviruses
Abdelnabi, Rana, Geraets, James A, Ma, Yipeng, Mirabelli, Carmen, Flatt, Justin W, Domanska, Aušra, Delang, Leen, Jochmans, Dirk, Kumar, Timiri Ajay, Jayaprakash, Venkatesan, Sinha, Barij Nayan, Leyssen, Pieter, Butcher, Sarah J, Neyts, Johan
Published in PLoS biology (11.06.2019)
Published in PLoS biology (11.06.2019)
Get full text
Journal Article
Rationally Designed Novel Phenyloxazoline Synthase Inhibitors: Chemical Synthesis and Biological Evaluation to Accelerate the Discovery of New Antimycobacterial Antibiotics
Shyam, Mousumi, Bhattacharje, Gourab, Daniel, Chris, Kumar, Amrendra, Yadav, Pragya, Mukherjee, Piyali, Singh, Samsher, Das, Amit Kumar, Narender, Tadigoppula, Singh, Amit, Jayaprakash, Venkatesan, Bhakta, Sanjib
Published in Molecules (Basel, Switzerland) (01.12.2023)
Published in Molecules (Basel, Switzerland) (01.12.2023)
Get full text
Journal Article
Novel Benzylidene Thiazolidinedione Derivatives as Partial PPARγ Agonists and their Antidiabetic Effects on Type 2 Diabetes
Yasmin, Sabina, Capone, Fabio, Laghezza, Antonio, Piaz, Fabrizio Dal, Loiodice, Fulvio, Vijayan, Viswanathan, Devadasan, Velmurugan, Mondal, Susanta K., Atlı, Özlem, Baysal, Merve, Pattnaik, Ashok K., Jayaprakash, Venkatesan, Lavecchia, Antonio
Published in Scientific reports (31.10.2017)
Published in Scientific reports (31.10.2017)
Get full text
Journal Article
Carbonic anhydrase inhibitory activity of phthalimide-capped benzene sulphonamide derivatives
Shilkar, Deepak, Mohd Siddique, Mohd Usman, Bua, Silvia, Yasmin, Sabina, Patil, Mrunali, Timiri, Ajay Kumar, Supuran, Claudiu T., Jayaprakash, Venkatesan
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Get full text
Journal Article
Quinazolinone derivative BNUA‐3 ameliorated [NDEA+2‐AAF]‐induced liver carcinogenesis in SD rats by modulating AhR‐CYP1B1‐Nrf2‐Keap1 pathway
Bose, Pritha, Siddique, Mohd. Usman M., Acharya, Reetuparna, Jayaprakash, Venkatesan, Sinha, Barij Nayan, Lapenna, Antonio, Pattanayak, Shakti P
Published in Clinical and experimental pharmacology & physiology (01.01.2020)
Published in Clinical and experimental pharmacology & physiology (01.01.2020)
Get full text
Journal Article
Scaffold Based Search on the Desferithiocin Archetype
Shyam, Mousumi, Dev, Abhimanyu, Sinha, Barij Nayan, Jayaprakash, Venkatesan
Published in Mini reviews in medicinal chemistry (01.01.2019)
Published in Mini reviews in medicinal chemistry (01.01.2019)
Get more information
Journal Article
Mycobactin analogue interacting with siderophore efflux-pump protein: insights from molecular dynamics simulations and whole-cell assays
Shyam, Mousumi, Thakur, Abhishek, Velez, Caroline, Daniel, Chris, Acevedo, Orlando, Bhakta, Sanjib, Jayaprakash, Venkatesan
Published in Frontiers in antibiotics (08.05.2024)
Published in Frontiers in antibiotics (08.05.2024)
Get full text
Journal Article
A Series of Ferulic Acid Amides Reveals Unexpected Peroxiredoxin 1 Inhibitory Activity with in vivo Antidiabetic and Hypolipidemic Effects
Yasmin, Sabina, Cerchia, Carmen, Badavath, Vishnu Nayak, Laghezza, Antonio, Dal Piaz, Fabrizio, Mondal, Susanta K., Atlı, Özlem, Baysal, Merve, Vadivelan, Sankaran, Shankar, S., Siddique, Mohd Usman Mohd, Pattnaik, Ashok Kumar, Singh, Ravi Pratap, Loiodice, Fulvio, Jayaprakash, Venkatesan, Lavecchia, Antonio
Published in ChemMedChem (04.02.2021)
Published in ChemMedChem (04.02.2021)
Get full text
Journal Article
Design, synthesis, optimization and antiviral activity of a class of hybrid dengue virus E protein inhibitors
Jadav, Surender Singh, Kaptein, Suzanne, Timiri, Ajaykumar, De Burghgraeve, Tine, Badavath, Vishnu Nayak, Ganesan, Ramesh, Sinha, Barij Nayan, Neyts, Johan, Leyssen, Pieter, Jayaprakash, Venkatesan
Published in Bioorganic & medicinal chemistry letters (15.04.2015)
Published in Bioorganic & medicinal chemistry letters (15.04.2015)
Get full text
Journal Article
Relevance of Machine Learning to Predict the Inhibitory Activity of Small Thiazole Chemicals on Estrogen Receptor
Jayaprakash, Venkatesan, Saravanan, Thangavelu, Ravindran, Karuppaiyan, Prabha, Thangavelu, Selvaraj, Jubie, Jayapalan, Sudeepan, Chaitanya, M V N L, Sivakumar, Thangavel
Published in Current computer-aided drug design (01.01.2023)
Published in Current computer-aided drug design (01.01.2023)
Get more information
Journal Article