Heteroaryl compounds, compositions thereof, and their use as protein kinase inhibitors
PERRIN-NINKOVIC, SOPHIE, HUANG, DEHUA, RIGGS, JENNIFER R, SHEVLIN, GRAZIELLA ISABEL, PAPA, PATRICK WILLIAM, MEDEROS, MARIA MERCEDES DELGADO, HARRIS, ROY LEONARD LLL, ALBERS, RONALD J, PARNES, JASON SIMON, LEE, BRANDON G, SCHWARZ, KIMBERLEY LYN, TEHRANI, LIDA RADNIA, SAPIENZA, JOHN JOSEPH, PACKARD, GARRICK K, MORTENSEN, DEBORAH SUE
Year of Publication 11.02.2015
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Year of Publication 11.02.2015
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Pyrazino[2,3-b]pyrazine mTOR kinase inhibitor for oncology indications and diseases associated with the mTOR/PI3K/AKT pathway
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, HARRIS ROY L, FULTZ KIMBERLY, SHEVLIN GRAZIELLA, LEE BRANDEN, SANKAR SABITA, PACKARD GARRICK, SAPIENZA JOHN, RIGGS JENNIFER, NARLA RAMA K, MADAKAMUTIL LOUI, PAPA PATRICK, PARNES JASON, MORTENSEN DEBORAH, ELSNER JAN, XU WEIMING, TEHRANI LIDA
Year of Publication 13.08.2013
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Year of Publication 13.08.2013
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Pyrazino[2,3-b]pyrazine mTOR kinase inhibitor for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, HARRIS ROY L, FULTZ KIMBERLY, SHEVLIN GRAZIELLA, LEE BRANDEN, SANKAR SABITA, PACKARD GARRICK, SAPIENZA JOHN, RIGGS JENNIFER, NARLA RAMA K, MADAKAMUTIL LOUI, PAPA PATRICK, PARNES JASON, MORTENSEN DEBORAH, ELSNER JAN, XU WEIMING, TEHRANI LIDA
Year of Publication 23.07.2013
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Year of Publication 23.07.2013
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MTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE MTOR/P13K/AKT PATHWAY
Garrick PACKARD, Weiming XU, Kimberly FULTZ, Sophie PERRIN-NINKOVIC, John SAPIENZA, Roy L. HARRIS, Rama K. NARLA, Loui MADAKAMUTIL, Deborah MORTENSEN, Branden LEE, Sabita SANKAR, Jason PARNES, Lida TEHRANI, Jingjing ZHAO, Patrick PAPA, Jennifer RIGGS, Jan ELSNER, Graziella SHEVLIN
Year of Publication 19.12.2018
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Year of Publication 19.12.2018
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3,4-Dihydropyrazino[2,3-b]pyrazin-2(1H)-one compounds as MTOR kinase inhibitors for oncology indications and diseases associated with the MTOR/P13K/AKT pathway
MORTENSEN, DEBORAH, PERRIN-NINKOVIC, SOPHIE, SHEVLIN, GRAZIELLA I, ZHAO, JINGJING, NARLA, RAMA K, TEHRANI, LIDA, MADAKAMUTIL, LOUI, SAPIENZA, JOHN, PARNES, JASON, FULTZ, KIMBERLY ELIZABETH, HARRIS, ROY, XU, WEIMING, SANKAR, SABITA, ELSNER, JAN, RIGGS, JENNIFER, PAPA, PATRICK, LEE, BRANDEN, PACKARD, GARRICK K
Year of Publication 11.06.2014
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Year of Publication 11.06.2014
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Methods of treatment using heteroaryl compounds and compositions thereof
CLAREEN STEVEN SPENCER, MORTENSEN DEBORAH SUE, PARNES JASON SIMON, SAPIENZA JOHN JOSEPH, RIGGS JENNIFER R, PAPA PATRICK WILLIAM, MCKENNA JEFFREY MARK, DELGADO MEDEROS MARIA MERCEDES, SCHWARZ KIMBERLY LYN, ALBERS RONALD J, HEGDE SAYEE GAJANAN
Year of Publication 26.02.2013
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Year of Publication 26.02.2013
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mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY
MORTENSEN, DEBORAH, PERRIN-NINKOVIC, SOPHIE, FULTZ KIMBERLY, ZHAO, JINGJING, SHEVLIN, GRAZIELLA, NARLA, RAMA K, TEHRANI, LIDA, PACKARD, GARRICK, SAPIENZA, JOHN, PARNES, JASON, HARRIS, ROY, L, XU, WEIMING, SANKAR, SABITA, ELSNER, JAN, MADAKAMUTIL LOUI, RIGGS, JENNIFER, PAPA, PATRICK, LEE, BRANDEN
Year of Publication 25.01.2013
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Year of Publication 25.01.2013
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PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, HARRIS ROY L, LEE BRANDEN, SANKAR SABITA, PACKARD GARRICK, NARLA RAMA, SAPIENZA JOHN, SHEVLIN GRAZIELLA I, RIGGS JENNIFER, MADAKAMUTIL LOUI, PAPA PATRICK, PARNES JASON, MORTENSEN DEBORAH, ELSNER JAN, XU WEIMING, FULTZ KIMBERLY ELIZABETH, TEHRANI LIDA
Year of Publication 31.10.2013
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Year of Publication 31.10.2013
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Heteroaryl compounds, compositions thereof, and use thereof as protein kinase inhibitors
PARNES, JASON SIMON, ALBERS, RONALD J, LEE, BRANDEN G, HUANG, DEHUA, RIGGS, JENNIFER R, SAPIENZA, JOHN JOSEPH, SCHWARZ, KIMBERLY LYN, PAPA, PATRICK WILLIAM, MEDEROS, MARIA MERCEDES DELGADO, MORTENSEN, DEBORAH SUE
Year of Publication 17.05.2012
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Year of Publication 17.05.2012
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Heteroaryl compounds, compositions thereof, and methods of treatment therewith
PERRIN-NINKOVIC, SOPHIE, LEE, BRANDEN G, HUANG, DEHUA, RIGGS, JENNIFER R, SHEVLIN, GRAZIELLA ISABEL, PAPA, PATRICK WILLIAM, MEDEROS, MARIA MERCEDES DELGADO, ALBERS, RONALD J, PARNES, JASON SIMON, TEHRANI, LIDA RADNIA, HARRIS III, ROY LEONARD, SAPIENZA, JOHN JOSEPH, SCHWARZ, KIMBERLY LYN, PACKARD, GARRICK K, MORTENSEN, DEBORAH SUE
Year of Publication 18.07.2013
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Year of Publication 18.07.2013
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PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITOR FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, HARRIS ROY L, FULTZ KIMBERLY, SHEVLIN GRAZIELLA, LEE BRANDEN, SANKAR SABITA, PACKARD GARRICK, SAPIENZA JOHN, RIGGS JENNIFER, NARLA RAMA K, MADAKAMUTIL LOUI, PAPA PATRICK, PARNES JASON, MORTENSEN DEBORAH, ELSNER JAN, XU WEIMING, TEHRANI LIDA
Year of Publication 22.03.2012
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Year of Publication 22.03.2012
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HETEROARYLVERBINDUNGEN,ZUSAMMENSETZUNGEN DARAUS UND IHRE VERWENDUNG ALS PROTEINKINASEHEMMER
ALBERS, RONALD J, PARNES, JASON SIMON, LEE, BRANDEN G, HUANG, DEHUA, RIGGS, JENNIFER R, SAPIENZA, JOHN JOSEPH, SCHWARZ, KIMBERLY LYN, PAPA, PATRICK WILLIAM, MORTENSEN, DEBORAH SUE, MEDEROS, MARIA MERCEDES DELGADO
Year of Publication 15.03.2012
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Year of Publication 15.03.2012
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HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND USE THEREOF AS PROTEIN KINASE INHIBITORS
ALBERS, RONALD J, PARNES, JASON SIMON, HEDGE, SAYEE, G, RIGGS, JENNIFER R, MCKENNA, JEFFREY, M, SAPIENZA, JOHN JOSEPH, SCHWARZ, KIMBERLY LYN, PAPA, PATRICK WILLIAM, CLAREEN, STEVEN, S, MORTENSEN, DEBORAH SUE, MEDEROS, MARIA MERCEDES DELGADO
Year of Publication 14.03.2012
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Year of Publication 14.03.2012
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PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITOR FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY
PERRIN-NINKOVIC SOPHIE, ZHAO JINGJING, HARRIS ROY L, FULTZ KIMBERLY, SHEVLIN GRAZIELLA, LEE BRANDEN, SANKAR SABITA, PACKARD GARRICK, SAPIENZA JOHN, RIGGS JENNIFER, NARLA RAMA K, MADAKAMUTIL LOUI, PAPA PATRICK, PARNES JASON, MORTENSEN DEBORAH, ELSNER JAN, XU WEIMING, TEHRANI LIDA
Year of Publication 08.03.2012
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Year of Publication 08.03.2012
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