An Assessment of the Effects of Serotonin 6 (5-HT6) Receptor Antagonists in Rodent Models of Learning
Lindner, Mark D, Hodges, Jr, Donald B, Hogan, John B, Orie, Anitra F, Corsa, Jason A, Barten, Donna M, Polson, Craig, Robertson, Barbara J, Guss, Valerie L, Gillman, Kevin W, Starrett, Jr, John E, Gribkoff, Valentin K
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
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Journal Article
Donepezil primarily attenuates scopolamine-induced deficits in psychomotor function, with moderate effects on simple conditioning and attention, and small effects on working memory and spatial mapping
Lindner, Mark D, Hogan, John B, Hodges, Jr, Donald B, Orie, Anitra F, Chen, Ping, Corsa, Jason A, Leet, John E, Gillman, Kevin W, Rose, Gregory M, Jones, Kelli M, Gribkoff, Valentin K
Published in Psychopharmacology (01.11.2006)
Published in Psychopharmacology (01.11.2006)
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Journal Article
2-(N-Benzyl-N-phenylsulfonamido)alkyl amide derivatives as γ-secretase inhibitors
Parker, Michael F., Barten, Donna M., Bergstrom, Carl P., Bronson, Joanne J., Corsa, Jason A., Dee, Michael F., Gai, Yonghua, Guss, Valerie L., Higgins, Mendi A., Keavy, Daniel J., Loo, Alice, Mate, Robert A., Marcin, Larry R., McElhone, Katharine E., Polson, Craig T., Roberts, Susan B., Macor, John E.
Published in Bioorganic & medicinal chemistry letters (15.11.2012)
Published in Bioorganic & medicinal chemistry letters (15.11.2012)
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Journal Article
Discovery of (S) -2 -( (S) -2 -(3,5 -difluorophenyl ) -2-hydroxyacetamido ) -N-( (S,Z) -3 -methyl -4 -oxo -4,5 -dihydro -3H-benzo[d|[1,2 ]diazepin -5 -yl )propanamide (BMS -433796 ) : A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer's disease
PRASAD, C. V. C, MING ZHENG, LOO, Alice, JIAN WANG, SLECZKA, Bogdan G, DANGLER, Charles, ROBERTSON, Barbara J, HENDRICK, Joseph P, ROBERTS, Susan B, BARTEN, Donna M, VIG, Shikha, BERGSTROM, Carl, SMITH, David W, QI GAO, YEOLA, Suresh, POLSON, Craig T, CORSA, Jason A, GUSS, Valerie L
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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Journal Article
Carbamate-appended N-alkylsulfonamides as inhibitors of γ-secretase
Bergstrom, Carl P., Sloan, Charles P., Lau, Wai-Yu, Smith, David W., Zheng, Ming, Hansel, Steven B., Polson, Craig T., Corsa, Jason A., Barten, Donna M., Felsenstein, Kevin M., Roberts, Susan B.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Journal Article
Amino-caprolactam derivatives as γ-secretase inhibitors
Parker, Michael F., Bronson, Joanne J., Barten, Donna M., Corsa, Jason A., Du, Wengsheng, Felsenstein, Kevin M., Guss, Valerie L., Izzarelli, Darcy, Loo, Alice, McElhone, Kate E., Marcin, Larry R., Padmanabha, Ramesh, Pak, Roger, Polson, Craig T., Toyn, Jeremy H., Varma, Sam, Wang, Jian, Wong, Victoria, Zheng, Ming, Roberts, Susan B.
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Journal Article
Soluble Aβ and cognitive function in aged F-344 rats and Tg2576 mice
Lindner, Mark D., Hogan, John B., Krause, Rudolph G., Machet, Frederic, Bourin, Clotilde, Hodges, Donald B., Corsa, Jason A., Barten, Donna M., Toyn, Jeremy H., Stock, David A., Rose, Gregory M., Gribkoff, Valentin K.
Published in Behavioural brain research (02.10.2006)
Published in Behavioural brain research (02.10.2006)
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Journal Article
2,3-Benzodiazepin-1,4-diones as peptidomimetic inhibitors of γ-secretase
Prasad, C.V.C., Vig, Shikha, Smith, David W., Gao, Qi, Polson, Craig T., Corsa, Jason A., Guss, Valerie L., Loo, Alice, Barten, Donna M., Zheng, Ming, Felsenstein, Kevin M., Roberts, Susan B.
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Journal Article
N-(5-Chloro-2-(hydroxymethyl)-N-alkyl-arylsulfonamides as γ-secretase inhibitors
Parker, Michael F., Barten, Donna M., Bergstrom, Carl P., Bronson, Joanne J., Corsa, Jason A., Deshpande, Milind S., Felsenstein, Kevin M., Guss, Valerie L., Hansel, Steven B., Johnson, Graham, Keavy, Daniel J., Lau, Wai Y., Mock, Jeremy, Prasad, C.V.C., Polson, Craig T., Sloan, Charles P., Smith, David W., Wallace, Owen B., Wang, Henry H., Williams, Andrew, Zheng, Ming
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Journal Article
Nitrogen-appended N-alkylsulfonamides as inhibitors of γ-secretase
Bergstrom, Carl P., Sloan, Charles P., Wang, Henry H., Parker, Michael F., Smith, David W., Zheng, Ming, Hansel, Steven B., Polson, Craig T., Barber, Lauren E., Bursuker, Isia, Guss, Valerie L., Corsa, Jason A., Barten, Donna M., Felsenstein, Kevin M., Roberts, Susan B.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Journal Article
The Amyloid-β Rise and γ-Secretase Inhibitor Potency Depend on the Level of Substrate Expression
Burton, Catherine R., Meredith, Jere E., Barten, Donna M., Goldstein, Margi E., Krause, Carol M., Kieras, Cathy J., Sisk, Lisa, Iben, Lawrence G., Polson, Craig, Thompson, Mark W., Lin, Xu-Alan, Corsa, Jason, Fiedler, Tracey, Pierdomenico, Maria, Cao, Yang, Roach, Arthur H., Cantone, Joseph L., Ford, Michael J., Drexler, Dieter M., Olson, Richard E., Yang, Michael G., Bergstrom, Carl P., McElhone, Kate E., Bronson, Joanne J., Macor, John E., Blat, Yuval, Grafstrom, Robert H., Stern, Andrew M., Seiffert, Dietmar A., Zaczek, Robert, Albright, Charles F., Toyn, Jeremy H.
Published in The Journal of biological chemistry (22.08.2008)
Published in The Journal of biological chemistry (22.08.2008)
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Journal Article
P-glycoprotein efflux and other factors limit brain amyloid beta reduction by beta-site amyloid precursor protein-cleaving enzyme 1 inhibitors in mice
Meredith, Jr, Jere E, Thompson, Lorin A, Toyn, Jeremy H, Marcin, Lawrence, Barten, Donna M, Marcinkeviciene, Jovita, Kopcho, Lisa, Kim, Young, Lin, Alan, Guss, Valerie, Burton, Catherine, Iben, Lawrence, Polson, Craig, Cantone, Joe, Ford, Michael, Drexler, Dieter, Fiedler, Tracey, Lentz, Kimberley A, Grace, Jr, James E, Kolb, Janet, Corsa, Jason, Pierdomenico, Maria, Jones, Kelli, Olson, Richard E, Macor, John E, Albright, Charles F
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
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Journal Article
Ex vivo occupancy of gamma-secretase inhibitors correlates with brain beta-amyloid peptide reduction in Tg2576 mice
Goldstein, Margi E, Cao, Yang, Fiedler, Tracey, Toyn, Jeremy, Iben, Lawrence, Barten, Donna M, Pierdomenico, Maria, Corsa, Jason, Prasad, C V C, Olson, Richard E, Li, Yu-Wen, Zaczek, Robert, Albright, Charles F
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
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Journal Article
P4‐020: Separation of Aβ Reduction from Notch Toxicity with Gamma Secretase Inhibitors in Rats
Meredith, Jere, Barten, Donna, Burton, Catherine, Corsa, Jason, Fiedler, Tracey, Guss, Valerie, Polson, Craig, Seiffert, Dietmar, Car, Bruce, Detnon, R. Rex, Hanumegowda, Umesh, Lentz, Kimberley, Clarke, Wendy, Macor, John, Zaczek, Robert, Houston, John, Olson, Richard, Albright, Charlie
Published in Alzheimer's & dementia (01.07.2010)
Published in Alzheimer's & dementia (01.07.2010)
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Journal Article
Separation of Aβ Reduction from Notch Toxicity with Gamma Secretase Inhibitors in Rats
Meredith, Jere, Barten, Donna, Burton, Catherine, Corsa, Jason, Fiedler, Tracey, Guss, Valerie, Polson, Craig, Seiffert, Dietmar, Car, Bruce, Detnon, R. Rex, Hanumegowda, Umesh, Lentz, Kimberley, Clarke, Wendy, Macor, John, Zaczek, Robert, Houston, John, Olson, Richard, Albright., Charlie
Published in Alzheimer's & dementia (01.07.2010)
Published in Alzheimer's & dementia (01.07.2010)
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Journal Article
Ex Vivo Occupancy of γ-Secretase Inhibitors Correlates with Brain β-Amyloid Peptide Reduction in Tg2576 Mice
Margi E. Goldstein, Yang Cao, Tracey Fiedler, Jeremy Toyn, Lawrence Iben, Donna M. Barten, Maria Pierdomenico, Jason Corsa, C. V. C. Prasad, Richard E. Olson, Yu-Wen Li, Robert Zaczek, Charles F. Albright
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2007)
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Journal Article
P-Glycoprotein Efflux and Other Factors Limit Brain Amyloid β Reduction by β-Site Amyloid Precursor Protein-Cleaving Enzyme 1 Inhibitors in Mice
Jere E. Meredith, Jr, Lorin A. Thompson, Jeremy H. Toyn, Lawrence Marcin, Donna M. Barten, Jovita Marcinkeviciene, Lisa Kopcho, Young Kim, Alan Lin, Valerie Guss, Catherine Burton, Lawrence Iben, Craig Polson, Joe Cantone, Michael Ford, Dieter Drexler, Tracey Fiedler, Kimberley A. Lentz, James E. Grace, Jr, Janet Kolb, Jason Corsa, Maria Pierdomenico, Kelli Jones, Richard E. Olson, John E. Macor, Charles F. Albright
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2008)
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Journal Article
The Amyloid-β Rise and γ-Secretase Inhibitor Potency Depend on the Level of Substrate Expression
Catherine R. Burton, Jere E. Meredith, Donna M. Barten, Margi E. Goldstein, Carol M. Krause, Cathy J. Kieras, Lisa Sisk, Lawrence G. Iben, Craig Polson, Mark W. Thompson, Xu-Alan Lin, Jason Corsa, Tracey Fiedler, Maria Pierdomenico, Yang Cao, Arthur H. Roach, Joseph L. Cantone, Michael J. Ford, Dieter M. Drexler, Richard E. Olson, Michael G. Yang, Carl P. Bergstrom, Kate E. McElhone, Joanne J. Bronson, John E. Macor, Yuval Blat, Robert H. Grafstrom, Andrew M. Stern, Dietmar A. Seiffert, Robert Zaczek, Charles F. Albright, Jeremy H. Toyn
Published in The Journal of biological chemistry (22.08.2008)
Published in The Journal of biological chemistry (22.08.2008)
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Journal Article
Soluble Abeta and cognitive function in aged F-344 rats and Tg2576 mice
Lindner, Mark D, Hogan, John B, Krause, Rudolph G, Machet, Frederic, Bourin, Clotilde, Hodges, Jr, Donald B, Corsa, Jason A, Barten, Donna M, Toyn, Jeremy H, Stock, David A, Rose, Gregory M, Gribkoff, Valentin K
Published in Behavioural brain research (02.10.2006)
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Published in Behavioural brain research (02.10.2006)
Journal Article
Discovery of (S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((S,Z)-3-methyl-4-oxo-4,5-dihydro-3H-benzo[d][1,2]diazepin-5-yl)propanamide (BMS-433796): a gamma-secretase inhibitor with Abeta lowering activity in a transgenic mouse model of Alzheimer's disease
Prasad, C V C, Zheng, Ming, Vig, Shikha, Bergstrom, Carl, Smith, David W, Gao, Qi, Yeola, Suresh, Polson, Craig T, Corsa, Jason A, Guss, Valerie L, Loo, Alice, Wang, Jian, Sleczka, Bogdan G, Dangler, Charles, Robertson, Barbara J, Hendrick, Joseph P, Roberts, Susan B, Barten, Donna M
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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Published in Bioorganic & medicinal chemistry letters (15.07.2007)
Journal Article